Table of Contents

Articles

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  A Novel Alcohol-Sensitive Position in the N-Methyl-d-Aspartate Receptor GluN2A Subunit M3 Domain Regulates Agonist Affinity and Ion Channel Gating

  Hong Ren, Yulin Zhao, Man Wu and Robert W. Peoples

  Molecular Pharmacology October 2013, 84 (4) 501-510; DOI: https://doi.org/10.1124/mol.113.085993
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  Brain-Derived Neurotrophic Factor–Mediated Downregulation of Brainstem K⁺–Cl^– Cotransporter and Cell-Type–Specific GABA Impairment for Activation of Descending Pain Facilitation

  Zhi Zhang, Xinxing Wang, Wei Wang, Yun-Gang Lu and Zhizhong Z. Pan

  Molecular Pharmacology October 2013, 84 (4) 511-520; DOI: https://doi.org/10.1124/mol.113.086496
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  Conserved Tryptophan Residues within Putative Transmembrane Domain 6 Affect Transport Function of Organic Anion Transporting Polypeptide 1B1

  Jiujiu Huang, Nan Li, Weifang Hong, Kai Zhan, Xuan Yu, Hong Huang and Mei Hong

  Molecular Pharmacology October 2013, 84 (4) 521-527; DOI: https://doi.org/10.1124/mol.113.085977
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  Muscarinic Receptors as Model Targets and Antitargets for Structure-Based Ligand Discovery

  Andrew C. Kruse, Dahlia R. Weiss, Mario Rossi, Jianxin Hu, Kelly Hu, Katrin Eitel, Peter Gmeiner, Jürgen Wess, Brian K. Kobilka and Brian K. Shoichet

  Molecular Pharmacology October 2013, 84 (4) 528-540; DOI: https://doi.org/10.1124/mol.113.087551
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  Inhibition of GluN2A-Containing N-Methyl-d-Aspartate Receptors by 2-Naphthoic Acid

  Han Yu and Gabriela K. Popescu

  Molecular Pharmacology October 2013, 84 (4) 541-550; DOI: https://doi.org/10.1124/mol.113.087189
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  Multiple Binding Sites for Small-Molecule Antagonists at the CC Chemokine Receptor 2

  Annelien J. M. Zweemer, Indira Nederpelt, Hilde Vrieling, Sarah Hafith, Maarten L. J. Doornbos, Henk de Vries, Jeffrey Abt, Raymond Gross, Dean Stamos, John Saunders, Martine J. Smit, Adriaan P. IJzerman and Laura H. Heitman

  Molecular Pharmacology October 2013, 84 (4) 551-561; DOI: https://doi.org/10.1124/mol.113.086850
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  Sorafenib/Regorafenib and Phosphatidyl Inositol 3 Kinase/Thymoma Viral Proto-Oncogene Inhibition Interact to Kill Tumor Cells

  Gangadharan B. Sajithlal, Hossein A. Hamed, Nichola Cruickshanks, Laurence Booth, Seyedmehrad Tavallai, Jahangir Syed, Steven Grant, Andrew Poklepovic and Paul Dent

  Molecular Pharmacology October 2013, 84 (4) 562-571; DOI: https://doi.org/10.1124/mol.113.088005
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  Paradoxical Activation of an Inwardly Rectifying Potassium Channel Mutant by Spermine: "(B)locking" Open the Bundle Crossing Gate

  Yury Y. Vilin, John-Jose Nunez, Robin Y. Kim, Gregory R. Dake and Harley T. Kurata

  Molecular Pharmacology October 2013, 84 (4) 572-581; DOI: https://doi.org/10.1124/mol.113.086603
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  Constitutive Knockout of Kalirin-7 Leads to Increased Rates of Cocaine Self-Administration

  Drew D. Kiraly, Natali E. Nemirovsky, Taylor P. LaRese, Seven E. Tomek, Stephanie L. Yahn, M. Foster Olive, Betty A. Eipper and Richard E. Mains

  Molecular Pharmacology October 2013, 84 (4) 582-590; DOI: https://doi.org/10.1124/mol.113.087106
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  Expression of Aryl Hydrocarbon Receptor Nuclear Translocator Enhances Cisplatin Resistance by Upregulating MDR1 Expression in Cancer Cells

  Ya-Yi Chan, Sriram Kalpana, Wei-Chiao Chang, Wen-Chang Chang and Ben-Kuen Chen

  Molecular Pharmacology October 2013, 84 (4) 591-602; DOI: https://doi.org/10.1124/mol.113.087197
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  Glutamate-Induced ATP Synthesis: Relationship between Plasma Membrane Na⁺/Ca²⁺ Exchanger and Excitatory Amino Acid Transporters in Brain and Heart Cell Models

  Simona Magi, Sara Arcangeli, Pasqualina Castaldo, Annamaria Assunta Nasti, Liberato Berrino, Elena Piegari, Renato Bernardini, Salvatore Amoroso and Vincenzo Lariccia

  Molecular Pharmacology October 2013, 84 (4) 603-614; DOI: https://doi.org/10.1124/mol.113.087775
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  Role of Human Hypoxanthine Guanine Phosphoribosyltransferase in Activation of the Antiviral Agent T-705 (Favipiravir)

  Lieve Naesens, Luke W. Guddat, Dianne T. Keough, André B. P. van Kuilenburg, Judith Meijer, Johan Vande Voorde and Jan Balzarini

  Molecular Pharmacology October 2013, 84 (4) 615-629; DOI: https://doi.org/10.1124/mol.113.087247
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  Fluorescence Correlation Spectroscopy Analysis of Serotonin, Adrenergic, Muscarinic, and Dopamine Receptor Dimerization: The Oligomer Number Puzzle

  Katharine Herrick-Davis, Ellinor Grinde, Ann Cowan and Joseph E. Mazurkiewicz

  Molecular Pharmacology October 2013, 84 (4) 630-642; DOI: https://doi.org/10.1124/mol.113.087072
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  C-Terminal Alternative Splicing of Ca_V1.3 Channels Distinctively Modulates Their Dihydropyridine Sensitivity

  Hua Huang, Dejie Yu and Tuck Wah Soong

  Molecular Pharmacology October 2013, 84 (4) 643-653; DOI: https://doi.org/10.1124/mol.113.087155