Table of Contents

Articles

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  Salicylate, a Catalytic Inhibitor of Topoisomerase II, Inhibits DNA Cleavage and Is Selective for the α Isoform

  Jason T. Bau, Zhili Kang, Caroline A. Austin and Ebba U. Kurz

  Molecular Pharmacology February 2014, 85 (2) 198-207; DOI: https://doi.org/10.1124/mol.113.088963
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  Binding of Mazindol and Analogs to the Human Serotonin and Dopamine Transporters

  Kasper Severinsen, Heidi Koldsø, Katrine Almind Vinberg Thorup, Christina Schjøth-Eskesen, Pernille Thornild Møller, Ove Wiborg, Henrik Helligsø Jensen, Steffen Sinning and Birgit Schiøtt

  Molecular Pharmacology February 2014, 85 (2) 208-217; DOI: https://doi.org/10.1124/mol.113.088922
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  Cross-Modulation and Molecular Interaction at the Ca_v3.3 Protein between the Endogenous Lipids and the T-Type Calcium Channel Antagonist TTA-A2.

  Magali Cazade, Cindy E. Nuss, Isabelle Bidaud, John J. Renger, Victor N. Uebele, Philippe Lory and Jean Chemin

  Molecular Pharmacology February 2014, 85 (2) 218-225; DOI: https://doi.org/10.1124/mol.113.089581
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  A Structural Explanation of the Effects of Dissociated Glucocorticoids on Glucocorticoid Receptor Transactivation

  Xavier Dezitter, Jérôme Fagart, Solenne Taront, Michel Fay, Bernadette Masselot, Dominique Hétuin, Pierre Formstecher, Marie-Edith Rafestin-Oblin and Thierry Idziorek

  Molecular Pharmacology February 2014, 85 (2) 226-236; DOI: https://doi.org/10.1124/mol.113.085860
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  Structural and Functional Analysis of G Protein–Coupled Receptor Kinase Inhibition by Paroxetine and a Rationally Designed Analog

  Kristoff T. Homan, Emily Wu, Michael W. Wilson, Puja Singh, Scott D. Larsen and John J. G. Tesmer

  Molecular Pharmacology February 2014, 85 (2) 237-248; DOI: https://doi.org/10.1124/mol.113.089631
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  Metformin Represses Drug-Induced Expression of CYP2B6 by Modulating the Constitutive Androstane Receptor Signaling

  Hui Yang, Brandy Garzel, Scott Heyward, Timothy Moeller, Paul Shapiro and Hongbing Wang

  Molecular Pharmacology February 2014, 85 (2) 249-260; DOI: https://doi.org/10.1124/mol.113.089763
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  Potent Antimycobacterial Activity of the Pyridoxal Isonicotinoyl Hydrazone Analog 2-Pyridylcarboxaldehyde Isonicotinoyl Hydrazone: A Lipophilic Transport Vehicle for Isonicotinic Acid Hydrazide

  Samantha Ellis, Danuta S. Kalinowski, Lisa Leotta, Michael L. H. Huang, Peter Jelfs, Vitali Sintchenko, Des R. Richardson and James A. Triccas

  Molecular Pharmacology February 2014, 85 (2) 269-278; DOI: https://doi.org/10.1124/mol.113.090357
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  Identification of Amino Acid Residues in the Ligand-Binding Domain of the Aryl Hydrocarbon Receptor Causing the Species-Specific Response to Omeprazole: Possible Determinants for Binding Putative Endogenous Ligands

  Kazuhiro Shiizaki, Seiichiroh Ohsako, Masanobu Kawanishi and Takashi Yagi

  Molecular Pharmacology February 2014, 85 (2) 279-289; DOI: https://doi.org/10.1124/mol.113.088856
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  Passenger Protein Determines Translocation Versus Retention in the Endoplasmic Reticulum for Aromatase Expression

  Jasmeet Kaur and Himangshu S. Bose

  Molecular Pharmacology February 2014, 85 (2) 290-300; DOI: https://doi.org/10.1124/mol.113.090431
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  The Second Extracellular Loop of the Adenosine A₁ Receptor Mediates Activity of Allosteric Enhancers

  Dylan P. Kennedy, Fiona M. McRobb, Susan A. Leonhardt, Michael Purdy, Heidi Figler, Melissa A. Marshall, Mahendra Chordia, Robert Figler, Joel Linden, Ruben Abagyan and Mark Yeager

  Molecular Pharmacology February 2014, 85 (2) 301-309; DOI: https://doi.org/10.1124/mol.113.088682
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  Enhanced Receptor-Mediated Endocytosis and Cytotoxicity of a Folic Acid-Desacetylvinblastine Monohydrazide Conjugate in a Pemetrexed-Resistant Cell Line Lacking Folate-Specific Facilitative Carriers but with Increased Folate Receptor Expression

  Rongbao Zhao, Ndeye Diop-Bove and I. David Goldman

  Molecular Pharmacology February 2014, 85 (2) 310-321; DOI: https://doi.org/10.1124/mol.113.089110
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  Glutamate, Substance P, and Calcitonin Gene-Related Peptide Cooperate in Inflammation-Induced Heat Hyperalgesia

  Katarzyna Rogoz, Helena Haddadi Andersen, Klas Kullander and Malin C. Lagerström

  Molecular Pharmacology February 2014, 85 (2) 322-334; DOI: https://doi.org/10.1124/mol.113.089532
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  Modulation of Transient Receptor Vanilloid 1 Activity by Transient Receptor Potential Ankyrin 1

  Viola Spahn, Christoph Stein and Christian Zöllner

  Molecular Pharmacology February 2014, 85 (2) 335-344; DOI: https://doi.org/10.1124/mol.113.088997
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  Interactions between the Regulatory Subunit of Type I Protein Kinase A and p90 Ribosomal S6 Kinase1 Regulate Cardiomyocyte Apoptosis

  Xianlong Gao, Brian Lin, Sakthivel Sadayappan and Tarun B. Patel

  Molecular Pharmacology February 2014, 85 (2) 357-367; DOI: https://doi.org/10.1124/mol.113.090613
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  Morphine Regulates Expression of μ-Opioid Receptor MOR-1A, an Intron-Retention Carboxyl Terminal Splice Variant of the μ-Opioid Receptor (OPRM1) Gene via miR-103/miR-107

  Zhigang Lu, Jin Xu, Mingming Xu, Gavril W. Pasternak and Ying-Xian Pan

  Molecular Pharmacology February 2014, 85 (2) 368-380; DOI: https://doi.org/10.1124/mol.113.089292