Research ArticleArticle
Quantification of Ligand Bias for Clinically Relevant β2-Adrenergic Receptor Ligands: Implications for Drug Taxonomy
Emma T. van der Westhuizen, Billy Breton, Arthur Christopoulos and Michel Bouvier
Molecular Pharmacology March 2014, 85 (3) 492-509; DOI: https://doi.org/10.1124/mol.113.088880
Emma T. van der Westhuizen
Department of Biochemistry and Institute for Research in Immunology and Cancer, University of Montreal, Montreal, Quebec, Canada (E.T.v.d.W., B.B., M.B.); and Drug Discovery Biology and Department of Pharmacology, Monash Institute for Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (E.T.v.d.W., A.C.)
Billy Breton
Department of Biochemistry and Institute for Research in Immunology and Cancer, University of Montreal, Montreal, Quebec, Canada (E.T.v.d.W., B.B., M.B.); and Drug Discovery Biology and Department of Pharmacology, Monash Institute for Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (E.T.v.d.W., A.C.)
Arthur Christopoulos
Department of Biochemistry and Institute for Research in Immunology and Cancer, University of Montreal, Montreal, Quebec, Canada (E.T.v.d.W., B.B., M.B.); and Drug Discovery Biology and Department of Pharmacology, Monash Institute for Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (E.T.v.d.W., A.C.)
Michel Bouvier
Department of Biochemistry and Institute for Research in Immunology and Cancer, University of Montreal, Montreal, Quebec, Canada (E.T.v.d.W., B.B., M.B.); and Drug Discovery Biology and Department of Pharmacology, Monash Institute for Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (E.T.v.d.W., A.C.)
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β2AR Ligands Are Biased toward ERK1/2 Signaling
Emma T. van der Westhuizen, Billy Breton, Arthur Christopoulos and Michel Bouvier
Molecular Pharmacology March 1, 2014, 85 (3) 492-509; DOI: https://doi.org/10.1124/mol.113.088880
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