Table of Contents

Articles

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  The Physical Association of the P2Y12 Receptor with PAR4 Regulates Arrestin-Mediated Akt Activation

  Aasma Khan, Dongjun Li, Salam Ibrahim, Emer Smyth and Donna S. Woulfe

  Molecular Pharmacology July 2014, 86 (1) 1-11; DOI: https://doi.org/10.1124/mol.114.091595
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  Antileukemic Activity and Mechanism of Drug Resistance to the Marine Salinispora tropica Proteasome Inhibitor Salinosporamide A (Marizomib)

  Denise Niewerth, Gerrit Jansen, Lesley F. V. Riethoff, Johan van Meerloo, Andrew J. Kale, Bradley S. Moore, Yehuda G. Assaraf, Janet L. Anderl, Sonja Zweegman, Gertjan J. L. Kaspers and Jacqueline Cloos

  Molecular Pharmacology July 2014, 86 (1) 12-19; DOI: https://doi.org/10.1124/mol.114.092114
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  Mutations in the Main Cytoplasmic Loop of the GABA_A Receptor α₄ and δ Subunits Have Opposite Effects on Surface Expression

  John R. Bracamontes, Ping Li, Gustav Akk and Joe Henry Steinbach

  Molecular Pharmacology July 2014, 86 (1) 20-27; DOI: https://doi.org/10.1124/mol.114.092791
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  Structure, Molecular Modeling, and Function of the Novel Potassium Channel Blocker Urotoxin Isolated from the Venom of the Australian Scorpion Urodacus yaschenkoi

  Karen Luna-Ramírez, Adam Bartok, Rita Restano-Cassulini, Veronica Quintero-Hernández, Fredy I. V. Coronas, Janni Christensen, Christine E. Wright, Gyorgy Panyi and Lourival D. Possani

  Molecular Pharmacology July 2014, 86 (1) 28-41; DOI: https://doi.org/10.1124/mol.113.090183
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  Synergy-Based Small-Molecule Screen Using a Human Lung Epithelial Cell Line Yields ΔF508-CFTR Correctors That Augment VX-809 Maximal Efficacy

  Puay-Wah Phuan, Guido Veit, Joseph Tan, Ariel Roldan, Walter E. Finkbeiner, Gergely L. Lukacs and A. S. Verkman

  Molecular Pharmacology July 2014, 86 (1) 42-51; DOI: https://doi.org/10.1124/mol.114.092478
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  Desensitization of Functional µ-Opioid Receptors Increases Agonist Off-Rate

  John T. Williams

  Molecular Pharmacology July 2014, 86 (1) 52-61; DOI: https://doi.org/10.1124/mol.114.092098
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  Characterization of the Zebrafish Ugt Repertoire Reveals a New Class of Drug-Metabolizing UDP Glucuronosyltransferases

  Yuanming Wang, Haiyan Huang and Qiang Wu

  Molecular Pharmacology July 2014, 86 (1) 62-75; DOI: https://doi.org/10.1124/mol.113.091462
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  An N-Terminal Threonine Mutation Produces an Efflux-Favorable, Sodium-Primed Conformation of the Human Dopamine Transporter

  Rheaclare Fraser, Yongyue Chen, Bipasha Guptaroy, Kathryn D. Luderman, Stephanie L. Stokes, Asim Beg, Louis J. DeFelice and Margaret E. Gnegy

  Molecular Pharmacology July 2014, 86 (1) 76-85; DOI: https://doi.org/10.1124/mol.114.091926
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  A Plasma Concentration of α-Ketoglutarate Influences the Kinetic Interaction of Ligands with Organic Anion Transporter 1

  Leslie Ingraham, Mansong Li, J. Larry Renfro, Sonda Parker, Arpine Vapurcuyan, Imad Hanna and Ryan M. Pelis

  Molecular Pharmacology July 2014, 86 (1) 86-95; DOI: https://doi.org/10.1124/mol.114.091777
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  Characterization of the Novel Positive Allosteric Modulator, LY2119620, at the Muscarinic M₂ and M₄ Receptors

  Carrie H. Croy, Douglas A. Schober, Hongling Xiao, Anne Quets, Arthur Christopoulos and Christian C. Felder

  Molecular Pharmacology July 2014, 86 (1) 106-115; DOI: https://doi.org/10.1124/mol.114.091751
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  Development of a Radioligand, [³H]LY2119620, to Probe the Human M₂ and M₄ Muscarinic Receptor Allosteric Binding Sites

  Douglas A. Schober, Carrie H. Croy, Hongling Xiao, Arthur Christopoulos and Christian C. Felder

  Molecular Pharmacology July 2014, 86 (1) 116-123; DOI: https://doi.org/10.1124/mol.114.091785