Research ArticleArticle
Development of a Radioligand, [3H]LY2119620, to Probe the Human M2 and M4 Muscarinic Receptor Allosteric Binding Sites
Douglas A. Schober, Carrie H. Croy, Hongling Xiao, Arthur Christopoulos and Christian C. Felder
Molecular Pharmacology July 2014, 86 (1) 116-123; DOI: https://doi.org/10.1124/mol.114.091785
Douglas A. Schober
Lilly Neuroscience, Lilly Research Laboratories, Eli Lilly and Co., Lilly Corporate Center, Indianapolis, Indiana (D.A.S., C.H.C., H.X., C.C.F.); and Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Parkville, Victoria, Australia (A.C.)
Carrie H. Croy
Lilly Neuroscience, Lilly Research Laboratories, Eli Lilly and Co., Lilly Corporate Center, Indianapolis, Indiana (D.A.S., C.H.C., H.X., C.C.F.); and Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Parkville, Victoria, Australia (A.C.)
Hongling Xiao
Lilly Neuroscience, Lilly Research Laboratories, Eli Lilly and Co., Lilly Corporate Center, Indianapolis, Indiana (D.A.S., C.H.C., H.X., C.C.F.); and Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Parkville, Victoria, Australia (A.C.)
Arthur Christopoulos
Lilly Neuroscience, Lilly Research Laboratories, Eli Lilly and Co., Lilly Corporate Center, Indianapolis, Indiana (D.A.S., C.H.C., H.X., C.C.F.); and Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Parkville, Victoria, Australia (A.C.)
Christian C. Felder
Lilly Neuroscience, Lilly Research Laboratories, Eli Lilly and Co., Lilly Corporate Center, Indianapolis, Indiana (D.A.S., C.H.C., H.X., C.C.F.); and Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Parkville, Victoria, Australia (A.C.)

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[3H]LY2119620, a Novel M2 and M4 mAChR Allosteric Probe
Douglas A. Schober, Carrie H. Croy, Hongling Xiao, Arthur Christopoulos and Christian C. Felder
Molecular Pharmacology July 1, 2014, 86 (1) 116-123; DOI: https://doi.org/10.1124/mol.114.091785
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