Research ArticleArticle
Fluoxetine Blocks Nav1.5 Channels via a Mechanism Similar to That of Class 1 Antiarrhythmics
Hugo Poulin, Iva Bruhova, Quadiri Timour, Olivier Theriault, Jean-Martin Beaulieu, Dominique Frassati and Mohamed Chahine
Molecular Pharmacology October 2014, 86 (4) 378-389; DOI: https://doi.org/10.1124/mol.114.093104
Hugo Poulin
Centre de recherche, Institut universitaire en santé mentale de Québec, Quebec City, Quebec, Canada (H.P., O.T., J.-M.B., M.C.); State University of New York at Buffalo, Buffalo, New York (I.B.); Laboratoire de Pharmacologie Médicale, EA 4612 Neurocardiologie, Université Lyon 1, Lyon, France (Q.T.); Department of Psychiatry and Neuroscience, Université Laval, Quebec City, Quebec, Canada (J.-M.B.); Pôle Dapela, Département de l’autisme et des psychoses d’évolution lente de l’adulte, Centre Hospitalier Le Vinatier, Bron, France (D.F.); and Department of Medicine, Université Laval, Quebec City, Quebec, Canada (M.C.)
Iva Bruhova
Centre de recherche, Institut universitaire en santé mentale de Québec, Quebec City, Quebec, Canada (H.P., O.T., J.-M.B., M.C.); State University of New York at Buffalo, Buffalo, New York (I.B.); Laboratoire de Pharmacologie Médicale, EA 4612 Neurocardiologie, Université Lyon 1, Lyon, France (Q.T.); Department of Psychiatry and Neuroscience, Université Laval, Quebec City, Quebec, Canada (J.-M.B.); Pôle Dapela, Département de l’autisme et des psychoses d’évolution lente de l’adulte, Centre Hospitalier Le Vinatier, Bron, France (D.F.); and Department of Medicine, Université Laval, Quebec City, Quebec, Canada (M.C.)
Quadiri Timour
Centre de recherche, Institut universitaire en santé mentale de Québec, Quebec City, Quebec, Canada (H.P., O.T., J.-M.B., M.C.); State University of New York at Buffalo, Buffalo, New York (I.B.); Laboratoire de Pharmacologie Médicale, EA 4612 Neurocardiologie, Université Lyon 1, Lyon, France (Q.T.); Department of Psychiatry and Neuroscience, Université Laval, Quebec City, Quebec, Canada (J.-M.B.); Pôle Dapela, Département de l’autisme et des psychoses d’évolution lente de l’adulte, Centre Hospitalier Le Vinatier, Bron, France (D.F.); and Department of Medicine, Université Laval, Quebec City, Quebec, Canada (M.C.)
Olivier Theriault
Centre de recherche, Institut universitaire en santé mentale de Québec, Quebec City, Quebec, Canada (H.P., O.T., J.-M.B., M.C.); State University of New York at Buffalo, Buffalo, New York (I.B.); Laboratoire de Pharmacologie Médicale, EA 4612 Neurocardiologie, Université Lyon 1, Lyon, France (Q.T.); Department of Psychiatry and Neuroscience, Université Laval, Quebec City, Quebec, Canada (J.-M.B.); Pôle Dapela, Département de l’autisme et des psychoses d’évolution lente de l’adulte, Centre Hospitalier Le Vinatier, Bron, France (D.F.); and Department of Medicine, Université Laval, Quebec City, Quebec, Canada (M.C.)
Jean-Martin Beaulieu
Centre de recherche, Institut universitaire en santé mentale de Québec, Quebec City, Quebec, Canada (H.P., O.T., J.-M.B., M.C.); State University of New York at Buffalo, Buffalo, New York (I.B.); Laboratoire de Pharmacologie Médicale, EA 4612 Neurocardiologie, Université Lyon 1, Lyon, France (Q.T.); Department of Psychiatry and Neuroscience, Université Laval, Quebec City, Quebec, Canada (J.-M.B.); Pôle Dapela, Département de l’autisme et des psychoses d’évolution lente de l’adulte, Centre Hospitalier Le Vinatier, Bron, France (D.F.); and Department of Medicine, Université Laval, Quebec City, Quebec, Canada (M.C.)
Dominique Frassati
Centre de recherche, Institut universitaire en santé mentale de Québec, Quebec City, Quebec, Canada (H.P., O.T., J.-M.B., M.C.); State University of New York at Buffalo, Buffalo, New York (I.B.); Laboratoire de Pharmacologie Médicale, EA 4612 Neurocardiologie, Université Lyon 1, Lyon, France (Q.T.); Department of Psychiatry and Neuroscience, Université Laval, Quebec City, Quebec, Canada (J.-M.B.); Pôle Dapela, Département de l’autisme et des psychoses d’évolution lente de l’adulte, Centre Hospitalier Le Vinatier, Bron, France (D.F.); and Department of Medicine, Université Laval, Quebec City, Quebec, Canada (M.C.)
Mohamed Chahine
Centre de recherche, Institut universitaire en santé mentale de Québec, Quebec City, Quebec, Canada (H.P., O.T., J.-M.B., M.C.); State University of New York at Buffalo, Buffalo, New York (I.B.); Laboratoire de Pharmacologie Médicale, EA 4612 Neurocardiologie, Université Lyon 1, Lyon, France (Q.T.); Department of Psychiatry and Neuroscience, Université Laval, Quebec City, Quebec, Canada (J.-M.B.); Pôle Dapela, Département de l’autisme et des psychoses d’évolution lente de l’adulte, Centre Hospitalier Le Vinatier, Bron, France (D.F.); and Department of Medicine, Université Laval, Quebec City, Quebec, Canada (M.C.)
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Research ArticleArticle
Fluoxetine Blocks Nav1.5 Channels
Hugo Poulin, Iva Bruhova, Quadiri Timour, Olivier Theriault, Jean-Martin Beaulieu, Dominique Frassati and Mohamed Chahine
Molecular Pharmacology October 1, 2014, 86 (4) 378-389; DOI: https://doi.org/10.1124/mol.114.093104
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