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Rapid CommunicationMinireview—Special Section on Highlights from IUPHAR

Advances in G Protein-Coupled Receptor Allostery: From Function to Structure

Arthur Christopoulos
Molecular Pharmacology November 2014, 86 (5) 463-478; DOI: https://doi.org/10.1124/mol.114.094342
Arthur Christopoulos
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
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Article Information

vol. 86 no. 5 463-478
DOI 
https://doi.org/10.1124/mol.114.094342
PubMed 
25061106

Published By 
American Society for Pharmacology and Experimental Therapeutics
Print ISSN 
0026-895X
Online ISSN 
1521-0111
History 
  • Received June 21, 2014
  • Accepted July 24, 2014
  • Published online September 25, 2014.

Article Versions

  • Earlier version (July 24, 2014 - 06:20).
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Copyright & Usage 
Copyright © 2014 by The American Society for Pharmacology and Experimental Therapeutics

Author Information

  1. Arthur Christopoulos
  1. Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
  1. Address correspondence to:
    Arthur Christopoulos, Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, 399 Royal Parade, Parkville, Victoria 3052, Australia. E-mail: arthur.christopoulos{at}monash.edu
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Molecular Pharmacology: 86 (5)
Molecular Pharmacology
Vol. 86, Issue 5
1 Nov 2014
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Rapid CommunicationMinireview—Special Section on Highlights from IUPHAR

Advances in GPCR Allostery

Arthur Christopoulos
Molecular Pharmacology November 1, 2014, 86 (5) 463-478; DOI: https://doi.org/10.1124/mol.114.094342

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Rapid CommunicationMinireview—Special Section on Highlights from IUPHAR

Advances in GPCR Allostery

Arthur Christopoulos
Molecular Pharmacology November 1, 2014, 86 (5) 463-478; DOI: https://doi.org/10.1124/mol.114.094342
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  • Article
    • Abstract
    • Introduction
    • Classification of Allosteric Modulators
    • Pharmacologic Characteristics of GPCR Allostery
    • Enriching Structure-Activity Studies of GPCR Allostery and Bias
    • Bitopic GPCR Ligands
    • Endogenous Allosteric Modulators
    • Understanding the Structural Basis of GPCR Allostery
    • Concluding Remarks
    • Acknowledgments
    • Footnotes
    • Abbreviations
    • References
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