Table of Contents

Articles

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  The Mitochondrial Complex V–Associated Large-Conductance Inner Membrane Current Is Regulated by Cyclosporine and Dexpramipexole

  Kambiz N. Alavian, Steven I. Dworetzky, Laura Bonanni, Ping Zhang, Silvio Sacchetti, Hongmei Li, Armando P. Signore, Peter J. S. Smith, Valentin K. Gribkoff and Elizabeth A. Jonas

  Molecular Pharmacology January 2015, 87 (1) 1-8; DOI: https://doi.org/10.1124/mol.114.095661
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  Influence of Gα_q on the Dynamics of M₃-Acetylcholine Receptor–G-Protein–Coupled Receptor Kinase 2 Interaction

  Valerie Wolters, Cornelius Krasel, Jörg Brockmann and Moritz Bünemann

  Molecular Pharmacology January 2015, 87 (1) 9-17; DOI: https://doi.org/10.1124/mol.114.094722
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  In Vitro Antitumor Mechanism of (E)-N-(2-methoxy-5-(((2,4,6-trimethoxystyryl)sulfonyl)methyl)pyridin-3-yl)methanesulfonamide

  Tiangong Lu, Charles A. Laughton, Shudong Wang and Tracey D. Bradshaw

  Molecular Pharmacology January 2015, 87 (1) 18-30; DOI: https://doi.org/10.1124/mol.114.093245
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  P-Retigabine: An N-Propargyled Retigabine with Improved Brain Distribution and Enhanced Antiepileptic Activity

  Pingzheng Zhou, Yangming Zhang, Haiyan Xu, Fei Chen, Xueqin Chen, Xiaoying Li, Xiaoping Pi, Lipeng Wang, Li Zhan, Fajun Nan and Zhaobing Gao

  Molecular Pharmacology January 2015, 87 (1) 31-38; DOI: https://doi.org/10.1124/mol.114.095190
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  Chaperoning of the A₁-Adenosine Receptor by Endogenous Adenosine—An Extension of the Retaliatory Metabolite Concept

  Justyna Kusek, Qiong Yang, Martin Witek, Christian W. Gruber, Christian Nanoff and Michael Freissmuth

  Molecular Pharmacology January 2015, 87 (1) 39-51; DOI: https://doi.org/10.1124/mol.114.094045
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  Superiority of Combined Phosphodiesterase PDE3/PDE4 Inhibition over PDE4 Inhibition Alone on Glucocorticoid- and Long-Acting β₂-Adrenoceptor Agonist–Induced Gene Expression in Human Airway Epithelial Cells

  Hawazen BinMahfouz, Bibhusana Borthakur, Dong Yan, Tresa George, Mark A. Giembycz and Robert Newton

  Molecular Pharmacology January 2015, 87 (1) 64-76; DOI: https://doi.org/10.1124/mol.114.093393
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  S-Adenosylmethionine and Methylthioadenosine Inhibit β-Catenin Signaling by Multiple Mechanisms in Liver and Colon Cancer

  Tony W. H. Li, Hui Peng, Heping Yang, Steven Kurniawidjaja, Parizad Panthaki, Yuhua Zheng, José M. Mato and Shelly C. Lu

  Molecular Pharmacology January 2015, 87 (1) 77-86; DOI: https://doi.org/10.1124/mol.114.095679
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  Activation of Human 5-Hydroxytryptamine Type 3 Receptors via an Allosteric Transmembrane Site

  Stuart J. Lansdell, Chaitra Sathyaprakash, Anne Doward and Neil S. Millar

  Molecular Pharmacology January 2015, 87 (1) 87-95; DOI: https://doi.org/10.1124/mol.114.094540
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  Monepantel Irreversibly Binds to and Opens Haemonchus contortus MPTL-1 and Caenorhabditis elegans ACR-20 Receptors

  Roland Baur, Robin Beech, Erwin Sigel and Lucien Rufener

  Molecular Pharmacology January 2015, 87 (1) 96-102; DOI: https://doi.org/10.1124/mol.114.095653
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  Salmeterol’s Extreme β2 Selectivity Is Due to Residues in Both Extracellular Loops and Transmembrane Domains

  Jillian G. Baker, Richard G. W. Proudman and Stephen J. Hill

  Molecular Pharmacology January 2015, 87 (1) 103-120; DOI: https://doi.org/10.1124/mol.114.095364
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  Extracellular Surface Residues of the α_1B-Adrenoceptor Critical for G Protein–Coupled Receptor Function

  Lotten Ragnarsson, Åsa Andersson, Walter G. Thomas and Richard J. Lewis

  Molecular Pharmacology January 2015, 87 (1) 121-129; DOI: https://doi.org/10.1124/mol.114.094557
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  Development of a Highly Selective Allosteric Antagonist Radioligand for the Type 1 Cholecystokinin Receptor and Elucidation of Its Molecular Basis of Binding

  Maoqing Dong, Ashton M. Vattelana, Polo C.-H. Lam, Andrew J. Orry, Ruben Abagyan, Arthur Christopoulos, Patrick M. Sexton, David R. Haines and Laurence J. Miller

  Molecular Pharmacology January 2015, 87 (1) 130-140; DOI: https://doi.org/10.1124/mol.114.095430