Table of Contents

Articles

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  Desformylflustrabromine (dFBr) and [³H]dFBr-Labeled Binding Sites in a Nicotinic Acetylcholine Receptor

  Ayman K. Hamouda, Ze-Jun Wang, Deirdre S. Stewart, Atul D. Jain, Richard A. Glennon and Jonathan B. Cohen

  Molecular Pharmacology July 2015, 88 (1) 1-11; DOI: https://doi.org/10.1124/mol.115.098913
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  Ligand Selectivity among the Dopamine and Serotonin Transporters Specified by the Forward Binding Reaction

  Peter S. Hasenhuetl, Klaus Schicker, Xaver Koenig, Yang Li, Subhodeep Sarker, Thomas Stockner, Sonja Sucic, Harald H. Sitte, Michael Freissmuth and Walter Sandtner

  Molecular Pharmacology July 2015, 88 (1) 12-18; DOI: https://doi.org/10.1124/mol.115.099036
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  C-Linker Accounts for Differential Sensitivity of ERG1 and ERG2 K⁺ Channels to RPR260243-Induced Slow Deactivation

  Alison Gardner and Michael C. Sanguinetti

  Molecular Pharmacology July 2015, 88 (1) 19-28; DOI: https://doi.org/10.1124/mol.115.098384
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  Circadian Modulation in the Intestinal Absorption of P-Glycoprotein Substrates in Monkeys

  Masaru Iwasaki, Satoru Koyanagi, Norio Suzuki, Chiharu Katamune, Naoya Matsunaga, Nobuaki Watanabe, Masayuki Takahashi, Takashi Izumi and Shigehiro Ohdo

  Molecular Pharmacology July 2015, 88 (1) 29-37; DOI: https://doi.org/10.1124/mol.114.096735
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  A Sexual Dimorphism Influences Bicyclol-Induced Hepatic Heat Shock Factor 1 Activation and Hepatoprotection

  Xiaosong Chen, Jianjian Zhang, Conghui Han, Huijuan Dai, Xianming Kong, Longmei Xu, Qiang Xia, Ming Zhang and Jianjun Zhang

  Molecular Pharmacology July 2015, 88 (1) 38-47; DOI: https://doi.org/10.1124/mol.114.097584
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  Antiobesity Effect of a Small Molecule Repressor of RORγ

  Mi Ra Chang, Yuanjun He, Tanya M. Khan, Dana S. Kuruvilla, Ruben Garcia-Ordonez, Cesar A. Corzo, Thaddeus J. Unger, David W. White, Susan Khan, Li Lin, Michael D. Cameron, Theodore M. Kamenecka and Patrick R. Griffin

  Molecular Pharmacology July 2015, 88 (1) 48-56; DOI: https://doi.org/10.1124/mol.114.097485
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  Essential Role of Calmodulin in RyR Inhibition by Dantrolene

  Ye Win Oo, Nieves Gomez-Hurtado, Kafa Walweel, Dirk F. van Helden, Mohammad S. Imtiaz, Bjorn C. Knollmann and Derek R. Laver

  Molecular Pharmacology July 2015, 88 (1) 57-63; DOI: https://doi.org/10.1124/mol.115.097691
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  CB₁ Knockout Mice Unveil Sustained CB₂-Mediated Antiallodynic Effects of the Mixed CB₁/CB₂ Agonist CP55,940 in a Mouse Model of Paclitaxel-Induced Neuropathic Pain

  Liting Deng, Benjamin L. Cornett, Ken Mackie and Andrea G. Hohmann

  Molecular Pharmacology July 2015, 88 (1) 64-74; DOI: https://doi.org/10.1124/mol.115.098483
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  Targeted Disruption of Organic Cation Transporter 3 Attenuates the Pharmacologic Response to Metformin

  Eugene C. Chen, Xiaomin Liang, Sook Wah Yee, Ethan G. Geier, Sophie L. Stocker, Ligong Chen and Kathleen M. Giacomini

  Molecular Pharmacology July 2015, 88 (1) 75-83; DOI: https://doi.org/10.1124/mol.114.096776
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  ATP–Binding Cassette Transporter Structure Changes Detected by Intramolecular Fluorescence Energy Transfer for High-Throughput Screening

  Surtaj H. Iram, Simon J. Gruber, Olga N. Raguimova, David D. Thomas and Seth L. Robia

  Molecular Pharmacology July 2015, 88 (1) 84-94; DOI: https://doi.org/10.1124/mol.114.096792
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  Characterization of Thrombin-Bound Dabigatran Effects on Protease-Activated Receptor-1 Expression and Signaling In Vitro

  Buxin Chen, Antonio G. Soto, Luisa J. Coronel, Ashley Goss, Joanne van Ryn and JoAnn Trejo

  Molecular Pharmacology July 2015, 88 (1) 95-105; DOI: https://doi.org/10.1124/mol.114.096446
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  Estrogen-Induced Cholestasis Leads to Repressed CYP2D6 Expression in CYP2D6-Humanized Mice

  Xian Pan and Hyunyoung Jeong

  Molecular Pharmacology July 2015, 88 (1) 106-112; DOI: https://doi.org/10.1124/mol.115.098822
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  The ClC-7 Chloride Channel Is Downregulated by Hypoosmotic Stress in Human Chondrocytes

  Takashi Kurita, Hisao Yamamura, Yoshiaki Suzuki, Wayne R. Giles and Yuji Imaizumi

  Molecular Pharmacology July 2015, 88 (1) 113-120; DOI: https://doi.org/10.1124/mol.115.098160
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  KU675, a Concomitant Heat-Shock Protein Inhibitor of Hsp90 and Hsc70 that Manifests Isoform Selectivity for Hsp90α in Prostate Cancer Cells

  Weiya Liu, George A. Vielhauer, Jeffrey M. Holzbeierlein, Huiping Zhao, Suman Ghosh, Douglas Brown, Eugene Lee and Brian S. J. Blagg

  Molecular Pharmacology July 2015, 88 (1) 121-130; DOI: https://doi.org/10.1124/mol.114.097303
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  The Pore Loop Domain of TRPV1 Is Required for Its Activation by the Volatile Anesthetics Chloroform and Isoflurane

  Corinna Kimball, Jialie Luo, Shijin Yin, Hongzhen Hu and Ajay Dhaka

  Molecular Pharmacology July 2015, 88 (1) 131-138; DOI: https://doi.org/10.1124/mol.115.098277