Molecular Pharmacology: 88 (2)

August 01, 2015; Volume 88,Issue 2

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Nucleotides Acting at P2Y Receptors: Connecting Structure and Function
Kenneth A. Jacobson, Silvia Paoletta, Vsevolod Katritch, Beili Wu, Zhan-Guo Gao, Qiang Zhao, Raymond C. Stevens and Evgeny Kiselev

Molecular Pharmacology August 2015, 88 (2) 220-230; DOI: https://doi.org/10.1124/mol.114.095711

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Direct Coupling of a Seven-Transmembrane-Span Receptor to a Gαi G-Protein Regulatory Motif Complex
William G. Robichaux, Sukru S. Oner, Stephen M. Lanier and Joe B. Blumer

Molecular Pharmacology August 2015, 88 (2) 231-237; DOI: https://doi.org/10.1124/mol.115.097741
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Structural Basis of Species-Dependent Differential Affinity of 6-Alkoxy-5-Aryl-3-Pyridinecarboxamide Cannabinoid-1 Receptor Antagonists
Malliga R. Iyer, Resat Cinar, Jie Liu, Grzegorz Godlewski, Gergö Szanda, Henry Puhl, Stephen R. Ikeda, Jeffrey Deschamps, Yong-Sok Lee, Peter J. Steinbach and George Kunos

Molecular Pharmacology August 2015, 88 (2) 238-244; DOI: https://doi.org/10.1124/mol.115.098541

Articles

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Synthesis and Evaluation of a Novel Deguelin Derivative, L80, which Disrupts ATP Binding to the C-terminal Domain of Heat Shock Protein 90
Su-Chan Lee, Hye-Young Min, Hoon Choi, Ho Shin Kim, Kyong-Cheol Kim, So-Jung Park, Myeong A Seong, Ji Hae Seo, Hyun-Ju Park, Young-Ger Suh, Kyu-Won Kim, Hyun-Seok Hong, Hee Kim, Min-Young Lee, Jeewoo Lee and Ho-Young Lee

Molecular Pharmacology August 2015, 88 (2) 245-255; DOI: https://doi.org/10.1124/mol.114.096883
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Menthol Enhances the Desensitization of Human α3β4 Nicotinic Acetylcholine Receptors
Hoai T. Ton, Amanda E. Smart, Brittany L. Aguilar, Thao T. Olson, Kenneth J. Kellar and Gerard P. Ahern

Molecular Pharmacology August 2015, 88 (2) 256-264; DOI: https://doi.org/10.1124/mol.115.098285
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The Lysophosphatidylinositol Receptor GPR55 Modulates Pain Perception in the Periaqueductal Gray
Elena Deliu, Margaret Sperow, Linda Console-Bram, Rhonda L. Carter, Douglas G. Tilley, Daniel J. Kalamarides, Lynn G. Kirby, G. Cristina Brailoiu, Eugen Brailoiu, Khalid Benamar and Mary E. Abood

Molecular Pharmacology August 2015, 88 (2) 265-272; DOI: https://doi.org/10.1124/mol.115.099333
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Rotational Symmetry of Two Pyrethroid Receptor Sites in the Mosquito Sodium Channel
Yuzhe Du, Yoshiko Nomura, Boris S. Zhorov and Ke Dong

Molecular Pharmacology August 2015, 88 (2) 273-280; DOI: https://doi.org/10.1124/mol.115.098707
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Soluble Epoxide Hydrolase Pharmacological Inhibition Ameliorates Experimental Acute Pancreatitis in Mice
Ahmed Bettaieb, Samah Chahed, Santana Bachaalany, Stephen Griffey, Bruce D. Hammock and Fawaz G. Haj

Molecular Pharmacology August 2015, 88 (2) 281-290; DOI: https://doi.org/10.1124/mol.114.097501
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Identification and Characterization of ProTx-III [μ-TRTX-Tp1a], a New Voltage-Gated Sodium Channel Inhibitor from Venom of the Tarantula Thrixopelma pruriens
Fernanda C. Cardoso, Zoltan Dekan, K. Johan Rosengren, Andelain Erickson, Irina Vetter, Jennifer R. Deuis, Volker Herzig, Paul F. Alewood, Glenn F. King and Richard J. Lewis

Molecular Pharmacology August 2015, 88 (2) 291-303; DOI: https://doi.org/10.1124/mol.115.098178
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Dysregulation of Endoplasmic Reticulum Stress and Autophagic Responses by the Antiretroviral Drug Efavirenz
Luc Bertrand and Michal Toborek

Molecular Pharmacology August 2015, 88 (2) 304-315; DOI: https://doi.org/10.1124/mol.115.098590
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Identification of a Dual Inhibitor of SRPK1 and CK2 That Attenuates Pathological Angiogenesis of Macular Degeneration in Mice
Satoshi Morooka, Mitsuteru Hoshina, Isao Kii, Takayoshi Okabe, Hirotatsu Kojima, Naoko Inoue, Yukiko Okuno, Masatsugu Denawa, Suguru Yoshida, Junichi Fukuhara, Kensuke Ninomiya, Teikichi Ikura, Toshio Furuya, Tetsuo Nagano, Kousuke Noda, Susumu Ishida, Takamitsu Hosoya, Nobutoshi Ito, Nagahisa Yoshimura and Masatoshi Hagiwara

Molecular Pharmacology August 2015, 88 (2) 316-325; DOI: https://doi.org/10.1124/mol.114.097345
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Neuritogenic Activity of Tetradecyl 2,3-Dihydroxybenzoate Is Mediated through the Insulin-Like Growth Factor 1 Receptor/Phosphatidylinositol 3 Kinase/Mitogen-Activated Protein Kinase Signaling Pathway
Ruiqi Tang, Lijuan Gao, Makoto Kawatani, Jianzhong Chen, Xueli Cao, Hiroyuki Osada, Lan Xiang and Jianhua Qi

Molecular Pharmacology August 2015, 88 (2) 326-334; DOI: https://doi.org/10.1124/mol.115.097758
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Biased Agonism of Endogenous Opioid Peptides at the μ-Opioid Receptor
Georgina L. Thompson, J. Robert Lane, Thomas Coudrat, Patrick M. Sexton, Arthur Christopoulos and Meritxell Canals

Molecular Pharmacology August 2015, 88 (2) 335-346; DOI: https://doi.org/10.1124/mol.115.098848
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Role of G Protein–Coupled Receptor Kinases 2 and 3 in μ-Opioid Receptor Desensitization and Internalization
Janet D. Lowe, Helen S. Sanderson, Alexandra E. Cooke, Mehrnoosh Ostovar, Elena Tsisanova, Sarah L. Withey, Charles Chavkin, Stephen M. Husbands, Eamonn Kelly, Graeme Henderson and Chris P. Bailey

Molecular Pharmacology August 2015, 88 (2) 347-356; DOI: https://doi.org/10.1124/mol.115.098293
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Discovery and Characterization of Nonpeptidyl Agonists of the Tissue-Protective Erythropoietin Receptor
James L. Miller, Timothy J. Church, Dmitri Leonoudakis, Karen Lariosa-Willingham, Normand L. Frigon, Connie S. Tettenborn, Jeffrey R. Spencer and Juha Punnonen

Molecular Pharmacology August 2015, 88 (2) 357-367; DOI: https://doi.org/10.1124/mol.115.098400
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Biased Agonism and Biased Allosteric Modulation at the CB₁ Cannabinoid Receptor
Elham Khajehali, Daniel T. Malone, Michelle Glass, Patrick M. Sexton, Arthur Christopoulos and Katie Leach

Molecular Pharmacology August 2015, 88 (2) 368-379; DOI: https://doi.org/10.1124/mol.115.099192
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Pharmacologic Inhibition of MNKs in Acute Myeloid Leukemia
Theodosia Teo, Frankie Lam, Mingfeng Yu, Yuchao Yang, Sunita K. C. Basnet, Hugo Albrecht, Matthew J. Sykes and Shudong Wang

Molecular Pharmacology August 2015, 88 (2) 380-389; DOI: https://doi.org/10.1124/mol.115.098012
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Biphasic Effects of Ingenol 3,20-Dibenzoate on the Erythropoietin Receptor: Synergism at Low Doses and Antagonism at High Doses
Jin-Gyo Oh, Young-Won Chin, Sung-Jo Kim, Jong Min Choi, Sang Kyum Kim, Hee Eun Kang and Tae-Hwe Heo

Molecular Pharmacology August 2015, 88 (2) 392-400; DOI: https://doi.org/10.1124/mol.114.097436
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A Multifaceted GABA_A Receptor Modulator: Functional Properties and Mechanism of Action of the Sedative-Hypnotic and Recreational Drug Methaqualone (Quaalude)
Harriet Hammer, Benjamin M. Bader, Corina Ehnert, Christoffer Bundgaard, Lennart Bunch, Kirsten Hoestgaard-Jensen, Olaf H.-U. Schroeder, Jesper F. Bastlund, Alexandra Gramowski-Voß and Anders A. Jensen

Molecular Pharmacology August 2015, 88 (2) 401-420; DOI: https://doi.org/10.1124/mol.115.099291

Notices of Retraction

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Re: Ling Y-H, Li T, Yuan Z, Haigentz M, Jr., Weber TK, and Perez-Soler R (2007) Erlotinib, an Effective Epidermal Growth Factor Receptor Tyrosine Kinase Inhibitor, Induces p27^KIP1 Up-Regulation and Nuclear Translocation in Association with Cell Growth Inhibition and G₁/S Phase Arrest in Human Non-Small-Cell Lung Cancer Cell Lines. Mol Pharmacol 72:248–258; doi:10.1124/mol.107.034827
Molecular Pharmacology August 2015, 88 (2) 390; DOI: https://doi.org/10.1124/mol.115.08er15a
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Re: Ling Y-H, Lin R, and Perez-Soler R (2008) Erlotinib Induces Mitochondrial-Mediated Apoptosis in Human H3255 Non-Small-Cell Lung Cancer Cells with Epidermal Growth Factor Receptor^L858R Mutation through Mitochondrial Oxidative Phosphorylation-Dependent Activation of BAX and BAK Mol Pharmacol 74:793–806; doi:10.1124/mol.107.044396
Molecular Pharmacology August 2015, 88 (2) 391; DOI: https://doi.org/10.1124/mol.115.08er15b

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