Research ArticleArticle
Biased Agonism of Endogenous Opioid Peptides at the μ-Opioid Receptor
Georgina L. Thompson, J. Robert Lane, Thomas Coudrat, Patrick M. Sexton, Arthur Christopoulos and Meritxell Canals
Molecular Pharmacology August 2015, 88 (2) 335-346; DOI: https://doi.org/10.1124/mol.115.098848
Georgina L. Thompson
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (G.L.T., J.R.L., T.C., P.M.S., A.C., M.C.); and Defence Science and Technology Organisation, Department of Defence, Fishermans Bend, Victoria, Australia (G.L.T.)
J. Robert Lane
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (G.L.T., J.R.L., T.C., P.M.S., A.C., M.C.); and Defence Science and Technology Organisation, Department of Defence, Fishermans Bend, Victoria, Australia (G.L.T.)
Thomas Coudrat
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (G.L.T., J.R.L., T.C., P.M.S., A.C., M.C.); and Defence Science and Technology Organisation, Department of Defence, Fishermans Bend, Victoria, Australia (G.L.T.)
Patrick M. Sexton
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (G.L.T., J.R.L., T.C., P.M.S., A.C., M.C.); and Defence Science and Technology Organisation, Department of Defence, Fishermans Bend, Victoria, Australia (G.L.T.)
Arthur Christopoulos
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (G.L.T., J.R.L., T.C., P.M.S., A.C., M.C.); and Defence Science and Technology Organisation, Department of Defence, Fishermans Bend, Victoria, Australia (G.L.T.)
Meritxell Canals
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia (G.L.T., J.R.L., T.C., P.M.S., A.C., M.C.); and Defence Science and Technology Organisation, Department of Defence, Fishermans Bend, Victoria, Australia (G.L.T.)
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Research ArticleArticle
Endogenous Biased Agonism at the μ-Opioid Receptor
Georgina L. Thompson, J. Robert Lane, Thomas Coudrat, Patrick M. Sexton, Arthur Christopoulos and Meritxell Canals
Molecular Pharmacology August 1, 2015, 88 (2) 335-346; DOI: https://doi.org/10.1124/mol.115.098848
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