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Molecular Pharmacology

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Table of Contents

October 01, 2015; Volume 88,Issue 4

Special Section on the Many Facets of Opioid Receptor Phosphorylation

  • You have access
    The Complex Roles of μ-Opioid Receptor Phosphorylation: A Key Determinant in Receptor Signaling and Regulation
    Meritxell Canals
    Molecular Pharmacology October 2015, 88 (4) 814-815; DOI: https://doi.org/10.1124/mol.115.100180
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    Agonist Binding and Desensitization of the μ-Opioid Receptor Is Modulated by Phosphorylation of the C-Terminal Tail Domain
    William T. Birdsong, Seksiri Arttamangkul, James R. Bunzow and John T. Williams
    Molecular Pharmacology October 2015, 88 (4) 816-824; DOI: https://doi.org/10.1124/mol.114.097527
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    Role of Phosphorylation Sites in Desensitization of µ-Opioid Receptor
    Arsalan Yousuf, Elke Miess, Setareh Sianati, Yan-Ping Du, Stefan Schulz and MacDonald J. Christie
    Molecular Pharmacology October 2015, 88 (4) 825-835; DOI: https://doi.org/10.1124/mol.115.098244

Minireview

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    PDZ Protein Regulation of G Protein–Coupled Receptor Trafficking and Signaling Pathways
    Henry A. Dunn and Stephen S. G. Ferguson
    Molecular Pharmacology October 2015, 88 (4) 624-639; DOI: https://doi.org/10.1124/mol.115.098509

Articles

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    AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
    Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
    Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978
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    Bidirectional Effect of Pregnenolone Sulfate on GluN1/GluN2A N-Methyl-d-Aspartate Receptor Gating Depending on Extracellular Calcium and Intracellular Milieu
    Divyan A. Chopra, Daniel T. Monaghan and Shashank M. Dravid
    Molecular Pharmacology October 2015, 88 (4) 650-659; DOI: https://doi.org/10.1124/mol.115.100396
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    Intracellular Dynamics and Fate of a Humanized Anti–Interleukin-6 Receptor Monoclonal Antibody, Tocilizumab
    Keiko Fujimoto, Hiroaki Ida, Yuko Hirota, Masaki Ishigai, Jun Amano and Yoshitaka Tanaka
    Molecular Pharmacology October 2015, 88 (4) 660-675; DOI: https://doi.org/10.1124/mol.115.099184
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    Substrate and Inhibitor–Specific Conformational Changes in the Human Serotonin Transporter Revealed by Voltage-Clamp Fluorometry
    Pella C. Söderhielm, Jacob Andersen, Lachlan Munro, Anne T. Nielsen and Anders S. Kristensen
    Molecular Pharmacology October 2015, 88 (4) 676-688; DOI: https://doi.org/10.1124/mol.115.099911
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    Benzopyrimido-pyrrolo-oxazine-dione (R)-BPO-27 Inhibits CFTR Chloride Channel Gating by Competition with ATP
    Yonjung Kim, Marc O. Anderson, Jinhong Park, Min Goo Lee, Wan Namkung and A. S. Verkman
    Molecular Pharmacology October 2015, 88 (4) 689-696; DOI: https://doi.org/10.1124/mol.115.098368
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    Acetylcholine-Binding Protein Engineered to Mimic the α4-α4 Binding Pocket in α4β2 Nicotinic Acetylcholine Receptors Reveals Interface Specific Interactions Important for Binding and Activity
    Azadeh Shahsavar, Philip K. Ahring, Jeppe A. Olsen, Christian Krintel, Jette S. Kastrup, Thomas Balle and Michael Gajhede
    Molecular Pharmacology October 2015, 88 (4) 697-707; DOI: https://doi.org/10.1124/mol.115.098061
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    Aspirin Targets SIRT1 and AMPK to Induce Senescence of Colorectal Carcinoma Cells
    Yu Ri Jung, Eun Ju Kim, Hyeong Jwa Choi, Jung-Jin Park, Hak-Su Kim, Yoon-Jin Lee, Myung-Jin Park and Minyoung Lee
    Molecular Pharmacology October 2015, 88 (4) 708-719; DOI: https://doi.org/10.1124/mol.115.098616
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    Suppression of Cytosolic NADPH Pool by Thionicotinamide Increases Oxidative Stress and Synergizes with Chemotherapy
    Philip M. Tedeschi, HongXia Lin, Murugesan Gounder, John E. Kerrigan, Emine Ercikan Abali, Kathleen Scotto and Joseph R. Bertino
    Molecular Pharmacology October 2015, 88 (4) 720-727; DOI: https://doi.org/10.1124/mol.114.096727
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    Protein Kinase C (PKC)ζ Pseudosubstrate Inhibitor Peptide Promiscuously Binds PKC Family Isoforms and Disrupts Conventional PKC Targeting and Translocation
    Amy S. Bogard and Steven J. Tavalin
    Molecular Pharmacology October 2015, 88 (4) 728-735; DOI: https://doi.org/10.1124/mol.115.099457
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    Mutational Analysis of the Putative High-Affinity Propofol Binding Site in Human β3 Homomeric GABAA Receptors
    Megan M. Eaton, Lily Q. Cao, Ziwei Chen, Nicholas P. Franks, Alex S. Evers and Gustav Akk
    Molecular Pharmacology October 2015, 88 (4) 736-745; DOI: https://doi.org/10.1124/mol.115.100347
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    Pregnane X Receptor Represses HNF4α Gene to Induce Insulin-Like Growth Factor–Binding Protein IGFBP1 that Alters Morphology of and Migrates HepG2 Cells
    Susumu Kodama, Yuichi Yamazaki and Masahiko Negishi
    Molecular Pharmacology October 2015, 88 (4) 746-757; DOI: https://doi.org/10.1124/mol.115.099341
  • Adenylyl Cyclase 5 Regulation by G<em>βγ</em> Involves Isoform-Specific Use of Multiple Interaction Sites
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    Adenylyl Cyclase 5 Regulation by Gβγ Involves Isoform-Specific Use of Multiple Interaction Sites
    Cameron S. Brand, Rachna Sadana, Sundeep Malik, Alan V. Smrcka and Carmen W. Dessauer
    Molecular Pharmacology October 2015, 88 (4) 758-767; DOI: https://doi.org/10.1124/mol.115.099556
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    Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
    Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
    Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376
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    Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists
    Darren M. Riddy, Celine Valant, Patricia Rueda, William N. Charman, Patrick M. Sexton, Roger J. Summers, Arthur Christopoulos and Christopher J. Langmead
    Molecular Pharmacology October 2015, 88 (4) 779-790; DOI: https://doi.org/10.1124/mol.115.100545
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    Potentiators of Defective ΔF508–CFTR Gating that Do Not Interfere with Corrector Action
    Puay-Wah Phuan, Guido Veit, Joseph A. Tan, Walter E. Finkbeiner, Gergely L. Lukacs and A. S. Verkman
    Molecular Pharmacology October 2015, 88 (4) 791-799; DOI: https://doi.org/10.1124/mol.115.099689
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    Suppression of Cytochrome P450 3A4 Function by UDP-Glucuronosyltransferase 2B7 through a Protein-Protein Interaction: Cooperative Roles of the Cytosolic Carboxyl-Terminal Domain and the Luminal Anchoring Region
    Yuu Miyauchi, Kiyoshi Nagata, Yasushi Yamazoe, Peter I. Mackenzie, Hideyuki Yamada and Yuji Ishii
    Molecular Pharmacology October 2015, 88 (4) 800-812; DOI: https://doi.org/10.1124/mol.115.098582

Erratum

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    Correction to: “Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice”
    Molecular Pharmacology October 2015, 88 (4) 813; DOI: https://doi.org/10.1124/mol.115.098376err
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In this issue

Molecular Pharmacology: 88 (4)
Molecular Pharmacology
Vol. 88, Issue 4
1 Oct 2015
  • Table of Contents
  • Table of Contents (PDF)
  • About the Cover
  • Index by author
  • Editorial Board (PDF)
  • Front Matter (PDF)
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  • Special Section on the Many Facets of Opioid Receptor Phosphorylation
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  • SB-431542 Is a Potent and Specific Inhibitor of Transforming Growth Factor-β Superfamily Type I Activin Receptor-Like Kinase (ALK) Receptors ALK4, ALK5, and ALK7
  • The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints
  • Pharmacological Properties of Y-27632, a Specific Inhibitor of Rho-Associated Kinases
  • Pharmacological characterization of five cloned voltage-gated K+ channels, types Kv1.1, 1.2, 1.3, 1.5, and 3.1, stably expressed in mammalian cell lines.
  • The Orphan Human Pregnane X Receptor Mediates the Transcriptional Activation of CYP3A4 by Rifampicin through a Distal Enhancer Module
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