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Index by author

October 01, 2015; Volume 88,Issue 4

A

  1. Abali, Emine Ercikan

    1. Suppression of Cytosolic NADPH Pool by Thionicotinamide Increases Oxidative Stress and Synergizes with Chemotherapy
      Philip M. Tedeschi, HongXia Lin, Murugesan Gounder, John E. Kerrigan, Emine Ercikan Abali, Kathleen Scotto and Joseph R. Bertino
      Molecular Pharmacology October 2015, 88 (4) 720-727; DOI: https://doi.org/10.1124/mol.114.096727

  2. Ahring, Philip K.

    1. Acetylcholine-Binding Protein Engineered to Mimic the α4-α4 Binding Pocket in α4β2 Nicotinic Acetylcholine Receptors Reveals Interface Specific Interactions Important for Binding and Activity
      Azadeh Shahsavar, Philip K. Ahring, Jeppe A. Olsen, Christian Krintel, Jette S. Kastrup, Thomas Balle and Michael Gajhede
      Molecular Pharmacology October 2015, 88 (4) 697-707; DOI: https://doi.org/10.1124/mol.115.098061

  3. Akk, Gustav

    1. Mutational Analysis of the Putative High-Affinity Propofol Binding Site in Human β3 Homomeric GABAA Receptors
      Megan M. Eaton, Lily Q. Cao, Ziwei Chen, Nicholas P. Franks, Alex S. Evers and Gustav Akk
      Molecular Pharmacology October 2015, 88 (4) 736-745; DOI: https://doi.org/10.1124/mol.115.100347

  4. Al-Muhtasib, Nour

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

  5. Amano, Jun

    1. Intracellular Dynamics and Fate of a Humanized Anti–Interleukin-6 Receptor Monoclonal Antibody, Tocilizumab
      Keiko Fujimoto, Hiroaki Ida, Yuko Hirota, Masaki Ishigai, Jun Amano and Yoshitaka Tanaka
      Molecular Pharmacology October 2015, 88 (4) 660-675; DOI: https://doi.org/10.1124/mol.115.099184

  6. Andersen, Jacob

    1. Substrate and Inhibitor–Specific Conformational Changes in the Human Serotonin Transporter Revealed by Voltage-Clamp Fluorometry
      Pella C. Söderhielm, Jacob Andersen, Lachlan Munro, Anne T. Nielsen and Anders S. Kristensen
      Molecular Pharmacology October 2015, 88 (4) 676-688; DOI: https://doi.org/10.1124/mol.115.099911

  7. Anderson, Marc O.

    1. Benzopyrimido-pyrrolo-oxazine-dione (R)-BPO-27 Inhibits CFTR Chloride Channel Gating by Competition with ATP
      Yonjung Kim, Marc O. Anderson, Jinhong Park, Min Goo Lee, Wan Namkung and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 689-696; DOI: https://doi.org/10.1124/mol.115.098368

  8. Aneja, Ritu

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

  9. Arttamangkul, Seksiri

    1. Agonist Binding and Desensitization of the μ-Opioid Receptor Is Modulated by Phosphorylation of the C-Terminal Tail Domain
      William T. Birdsong, Seksiri Arttamangkul, James R. Bunzow and John T. Williams
      Molecular Pharmacology October 2015, 88 (4) 816-824; DOI: https://doi.org/10.1124/mol.114.097527

B

  1. Balle, Thomas

    1. Acetylcholine-Binding Protein Engineered to Mimic the α4-α4 Binding Pocket in α4β2 Nicotinic Acetylcholine Receptors Reveals Interface Specific Interactions Important for Binding and Activity
      Azadeh Shahsavar, Philip K. Ahring, Jeppe A. Olsen, Christian Krintel, Jette S. Kastrup, Thomas Balle and Michael Gajhede
      Molecular Pharmacology October 2015, 88 (4) 697-707; DOI: https://doi.org/10.1124/mol.115.098061

  2. Bertino, Joseph R.

    1. Suppression of Cytosolic NADPH Pool by Thionicotinamide Increases Oxidative Stress and Synergizes with Chemotherapy
      Philip M. Tedeschi, HongXia Lin, Murugesan Gounder, John E. Kerrigan, Emine Ercikan Abali, Kathleen Scotto and Joseph R. Bertino
      Molecular Pharmacology October 2015, 88 (4) 720-727; DOI: https://doi.org/10.1124/mol.114.096727

  3. Birdsong, William T.

    1. Agonist Binding and Desensitization of the μ-Opioid Receptor Is Modulated by Phosphorylation of the C-Terminal Tail Domain
      William T. Birdsong, Seksiri Arttamangkul, James R. Bunzow and John T. Williams
      Molecular Pharmacology October 2015, 88 (4) 816-824; DOI: https://doi.org/10.1124/mol.114.097527

  4. Bogard, Amy S.

    1. Protein Kinase C (PKC)ζ Pseudosubstrate Inhibitor Peptide Promiscuously Binds PKC Family Isoforms and Disrupts Conventional PKC Targeting and Translocation
      Amy S. Bogard and Steven J. Tavalin
      Molecular Pharmacology October 2015, 88 (4) 728-735; DOI: https://doi.org/10.1124/mol.115.099457

  5. Bowman Dalley, Carrie

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

  6. Brand, Cameron S.

    1. Adenylyl Cyclase 5 Regulation by G<em>βγ</em> Involves Isoform-Specific Use of Multiple Interaction Sites
      Adenylyl Cyclase 5 Regulation by Gβγ Involves Isoform-Specific Use of Multiple Interaction Sites
      Cameron S. Brand, Rachna Sadana, Sundeep Malik, Alan V. Smrcka and Carmen W. Dessauer
      Molecular Pharmacology October 2015, 88 (4) 758-767; DOI: https://doi.org/10.1124/mol.115.099556

  7. Bunzow, James R.

    1. Agonist Binding and Desensitization of the μ-Opioid Receptor Is Modulated by Phosphorylation of the C-Terminal Tail Domain
      William T. Birdsong, Seksiri Arttamangkul, James R. Bunzow and John T. Williams
      Molecular Pharmacology October 2015, 88 (4) 816-824; DOI: https://doi.org/10.1124/mol.114.097527

C

  1. Canals, Meritxell

    1. The Complex Roles of μ-Opioid Receptor Phosphorylation: A Key Determinant in Receptor Signaling and Regulation
      Meritxell Canals
      Molecular Pharmacology October 2015, 88 (4) 814-815; DOI: https://doi.org/10.1124/mol.115.100180

  2. Cao, Lily Q.

    1. Mutational Analysis of the Putative High-Affinity Propofol Binding Site in Human β3 Homomeric GABAA Receptors
      Megan M. Eaton, Lily Q. Cao, Ziwei Chen, Nicholas P. Franks, Alex S. Evers and Gustav Akk
      Molecular Pharmacology October 2015, 88 (4) 736-745; DOI: https://doi.org/10.1124/mol.115.100347

  3. Charman, William N.

    1. Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists
      Darren M. Riddy, Celine Valant, Patricia Rueda, William N. Charman, Patrick M. Sexton, Roger J. Summers, Arthur Christopoulos and Christopher J. Langmead
      Molecular Pharmacology October 2015, 88 (4) 779-790; DOI: https://doi.org/10.1124/mol.115.100545

  4. Chen, Ziwei

    1. Mutational Analysis of the Putative High-Affinity Propofol Binding Site in Human β3 Homomeric GABAA Receptors
      Megan M. Eaton, Lily Q. Cao, Ziwei Chen, Nicholas P. Franks, Alex S. Evers and Gustav Akk
      Molecular Pharmacology October 2015, 88 (4) 736-745; DOI: https://doi.org/10.1124/mol.115.100347

  5. Choi, Hyeong Jwa

    1. Aspirin Targets SIRT1 and AMPK to Induce Senescence of Colorectal Carcinoma Cells
      Yu Ri Jung, Eun Ju Kim, Hyeong Jwa Choi, Jung-Jin Park, Hak-Su Kim, Yoon-Jin Lee, Myung-Jin Park and Minyoung Lee
      Molecular Pharmacology October 2015, 88 (4) 708-719; DOI: https://doi.org/10.1124/mol.115.098616

  6. Chopra, Divyan A.

    1. Bidirectional Effect of Pregnenolone Sulfate on GluN1/GluN2A N-Methyl-d-Aspartate Receptor Gating Depending on Extracellular Calcium and Intracellular Milieu
      Divyan A. Chopra, Daniel T. Monaghan and Shashank M. Dravid
      Molecular Pharmacology October 2015, 88 (4) 650-659; DOI: https://doi.org/10.1124/mol.115.100396

  7. Christie, MacDonald J.

    1. Role of Phosphorylation Sites in Desensitization of µ-Opioid Receptor
      Arsalan Yousuf, Elke Miess, Setareh Sianati, Yan-Ping Du, Stefan Schulz and MacDonald J. Christie
      Molecular Pharmacology October 2015, 88 (4) 825-835; DOI: https://doi.org/10.1124/mol.115.098244

  8. Christopoulos, Arthur

    1. Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists
      Darren M. Riddy, Celine Valant, Patricia Rueda, William N. Charman, Patrick M. Sexton, Roger J. Summers, Arthur Christopoulos and Christopher J. Langmead
      Molecular Pharmacology October 2015, 88 (4) 779-790; DOI: https://doi.org/10.1124/mol.115.100545

  9. Chuttani, Krishna

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

D

  1. Dessauer, Carmen W.

    1. Adenylyl Cyclase 5 Regulation by G<em>βγ</em> Involves Isoform-Specific Use of Multiple Interaction Sites
      Adenylyl Cyclase 5 Regulation by Gβγ Involves Isoform-Specific Use of Multiple Interaction Sites
      Cameron S. Brand, Rachna Sadana, Sundeep Malik, Alan V. Smrcka and Carmen W. Dessauer
      Molecular Pharmacology October 2015, 88 (4) 758-767; DOI: https://doi.org/10.1124/mol.115.099556

  2. Dravid, Shashank M.

    1. Bidirectional Effect of Pregnenolone Sulfate on GluN1/GluN2A N-Methyl-d-Aspartate Receptor Gating Depending on Extracellular Calcium and Intracellular Milieu
      Divyan A. Chopra, Daniel T. Monaghan and Shashank M. Dravid
      Molecular Pharmacology October 2015, 88 (4) 650-659; DOI: https://doi.org/10.1124/mol.115.100396

  3. Du, Yan-Ping

    1. Role of Phosphorylation Sites in Desensitization of µ-Opioid Receptor
      Arsalan Yousuf, Elke Miess, Setareh Sianati, Yan-Ping Du, Stefan Schulz and MacDonald J. Christie
      Molecular Pharmacology October 2015, 88 (4) 825-835; DOI: https://doi.org/10.1124/mol.115.098244

  4. Dunn, Henry A.

    1. PDZ Protein Regulation of G Protein–Coupled Receptor Trafficking and Signaling Pathways
      Henry A. Dunn and Stephen S. G. Ferguson
      Molecular Pharmacology October 2015, 88 (4) 624-639; DOI: https://doi.org/10.1124/mol.115.098509

E

  1. Eaton, Megan M.

    1. Mutational Analysis of the Putative High-Affinity Propofol Binding Site in Human β3 Homomeric GABAA Receptors
      Megan M. Eaton, Lily Q. Cao, Ziwei Chen, Nicholas P. Franks, Alex S. Evers and Gustav Akk
      Molecular Pharmacology October 2015, 88 (4) 736-745; DOI: https://doi.org/10.1124/mol.115.100347

  2. Evers, Alex S.

    1. Mutational Analysis of the Putative High-Affinity Propofol Binding Site in Human β3 Homomeric GABAA Receptors
      Megan M. Eaton, Lily Q. Cao, Ziwei Chen, Nicholas P. Franks, Alex S. Evers and Gustav Akk
      Molecular Pharmacology October 2015, 88 (4) 736-745; DOI: https://doi.org/10.1124/mol.115.100347

F

  1. Ferguson, Stephen S. G.

    1. PDZ Protein Regulation of G Protein–Coupled Receptor Trafficking and Signaling Pathways
      Henry A. Dunn and Stephen S. G. Ferguson
      Molecular Pharmacology October 2015, 88 (4) 624-639; DOI: https://doi.org/10.1124/mol.115.098509

  2. Finkbeiner, Walter E.

    1. Potentiators of Defective ΔF508–CFTR Gating that Do Not Interfere with Corrector Action
      Puay-Wah Phuan, Guido Veit, Joseph A. Tan, Walter E. Finkbeiner, Gergely L. Lukacs and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 791-799; DOI: https://doi.org/10.1124/mol.115.099689

  3. Franks, Nicholas P.

    1. Mutational Analysis of the Putative High-Affinity Propofol Binding Site in Human β3 Homomeric GABAA Receptors
      Megan M. Eaton, Lily Q. Cao, Ziwei Chen, Nicholas P. Franks, Alex S. Evers and Gustav Akk
      Molecular Pharmacology October 2015, 88 (4) 736-745; DOI: https://doi.org/10.1124/mol.115.100347

  4. Fujimoto, Keiko

    1. Intracellular Dynamics and Fate of a Humanized Anti–Interleukin-6 Receptor Monoclonal Antibody, Tocilizumab
      Keiko Fujimoto, Hiroaki Ida, Yuko Hirota, Masaki Ishigai, Jun Amano and Yoshitaka Tanaka
      Molecular Pharmacology October 2015, 88 (4) 660-675; DOI: https://doi.org/10.1124/mol.115.099184

G

  1. Gajhede, Michael

    1. Acetylcholine-Binding Protein Engineered to Mimic the α4-α4 Binding Pocket in α4β2 Nicotinic Acetylcholine Receptors Reveals Interface Specific Interactions Important for Binding and Activity
      Azadeh Shahsavar, Philip K. Ahring, Jeppe A. Olsen, Christian Krintel, Jette S. Kastrup, Thomas Balle and Michael Gajhede
      Molecular Pharmacology October 2015, 88 (4) 697-707; DOI: https://doi.org/10.1124/mol.115.098061

  2. Gao, Yongiun

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

  3. Gounder, Murugesan

    1. Suppression of Cytosolic NADPH Pool by Thionicotinamide Increases Oxidative Stress and Synergizes with Chemotherapy
      Philip M. Tedeschi, HongXia Lin, Murugesan Gounder, John E. Kerrigan, Emine Ercikan Abali, Kathleen Scotto and Joseph R. Bertino
      Molecular Pharmacology October 2015, 88 (4) 720-727; DOI: https://doi.org/10.1124/mol.114.096727

  4. Gundala, Sushma R.

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

H

  1. Hazari, Puja P.

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

  2. Hirota, Yuko

    1. Intracellular Dynamics and Fate of a Humanized Anti–Interleukin-6 Receptor Monoclonal Antibody, Tocilizumab
      Keiko Fujimoto, Hiroaki Ida, Yuko Hirota, Masaki Ishigai, Jun Amano and Yoshitaka Tanaka
      Molecular Pharmacology October 2015, 88 (4) 660-675; DOI: https://doi.org/10.1124/mol.115.099184

  3. Horti, Andrew G.

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

I

  1. Ida, Hiroaki

    1. Intracellular Dynamics and Fate of a Humanized Anti–Interleukin-6 Receptor Monoclonal Antibody, Tocilizumab
      Keiko Fujimoto, Hiroaki Ida, Yuko Hirota, Masaki Ishigai, Jun Amano and Yoshitaka Tanaka
      Molecular Pharmacology October 2015, 88 (4) 660-675; DOI: https://doi.org/10.1124/mol.115.099184

  2. Ishigai, Masaki

    1. Intracellular Dynamics and Fate of a Humanized Anti–Interleukin-6 Receptor Monoclonal Antibody, Tocilizumab
      Keiko Fujimoto, Hiroaki Ida, Yuko Hirota, Masaki Ishigai, Jun Amano and Yoshitaka Tanaka
      Molecular Pharmacology October 2015, 88 (4) 660-675; DOI: https://doi.org/10.1124/mol.115.099184

  3. Ishii, Yuji

    1. Suppression of Cytochrome P450 3A4 Function by UDP-Glucuronosyltransferase 2B7 through a Protein-Protein Interaction: Cooperative Roles of the Cytosolic Carboxyl-Terminal Domain and the Luminal Anchoring Region
      Yuu Miyauchi, Kiyoshi Nagata, Yasushi Yamazoe, Peter I. Mackenzie, Hideyuki Yamada and Yuji Ishii
      Molecular Pharmacology October 2015, 88 (4) 800-812; DOI: https://doi.org/10.1124/mol.115.098582

J

  1. Jung, Yu Ri

    1. Aspirin Targets SIRT1 and AMPK to Induce Senescence of Colorectal Carcinoma Cells
      Yu Ri Jung, Eun Ju Kim, Hyeong Jwa Choi, Jung-Jin Park, Hak-Su Kim, Yoon-Jin Lee, Myung-Jin Park and Minyoung Lee
      Molecular Pharmacology October 2015, 88 (4) 708-719; DOI: https://doi.org/10.1124/mol.115.098616

K

  1. Kastrup, Jette S.

    1. Acetylcholine-Binding Protein Engineered to Mimic the α4-α4 Binding Pocket in α4β2 Nicotinic Acetylcholine Receptors Reveals Interface Specific Interactions Important for Binding and Activity
      Azadeh Shahsavar, Philip K. Ahring, Jeppe A. Olsen, Christian Krintel, Jette S. Kastrup, Thomas Balle and Michael Gajhede
      Molecular Pharmacology October 2015, 88 (4) 697-707; DOI: https://doi.org/10.1124/mol.115.098061

  2. Katyal, Anju

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

  3. Kellar, Kenneth J.

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

  4. Kerrigan, John E.

    1. Suppression of Cytosolic NADPH Pool by Thionicotinamide Increases Oxidative Stress and Synergizes with Chemotherapy
      Philip M. Tedeschi, HongXia Lin, Murugesan Gounder, John E. Kerrigan, Emine Ercikan Abali, Kathleen Scotto and Joseph R. Bertino
      Molecular Pharmacology October 2015, 88 (4) 720-727; DOI: https://doi.org/10.1124/mol.114.096727

  5. Kim, Eun Ju

    1. Aspirin Targets SIRT1 and AMPK to Induce Senescence of Colorectal Carcinoma Cells
      Yu Ri Jung, Eun Ju Kim, Hyeong Jwa Choi, Jung-Jin Park, Hak-Su Kim, Yoon-Jin Lee, Myung-Jin Park and Minyoung Lee
      Molecular Pharmacology October 2015, 88 (4) 708-719; DOI: https://doi.org/10.1124/mol.115.098616

  6. Kim, Hak-Su

    1. Aspirin Targets SIRT1 and AMPK to Induce Senescence of Colorectal Carcinoma Cells
      Yu Ri Jung, Eun Ju Kim, Hyeong Jwa Choi, Jung-Jin Park, Hak-Su Kim, Yoon-Jin Lee, Myung-Jin Park and Minyoung Lee
      Molecular Pharmacology October 2015, 88 (4) 708-719; DOI: https://doi.org/10.1124/mol.115.098616

  7. Kim, Yonjung

    1. Benzopyrimido-pyrrolo-oxazine-dione (R)-BPO-27 Inhibits CFTR Chloride Channel Gating by Competition with ATP
      Yonjung Kim, Marc O. Anderson, Jinhong Park, Min Goo Lee, Wan Namkung and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 689-696; DOI: https://doi.org/10.1124/mol.115.098368

  8. Kodama, Susumu

    1. Pregnane X Receptor Represses HNF4α Gene to Induce Insulin-Like Growth Factor–Binding Protein IGFBP1 that Alters Morphology of and Migrates HepG2 Cells
      Susumu Kodama, Yuichi Yamazaki and Masahiko Negishi
      Molecular Pharmacology October 2015, 88 (4) 746-757; DOI: https://doi.org/10.1124/mol.115.099341

  9. Krintel, Christian

    1. Acetylcholine-Binding Protein Engineered to Mimic the α4-α4 Binding Pocket in α4β2 Nicotinic Acetylcholine Receptors Reveals Interface Specific Interactions Important for Binding and Activity
      Azadeh Shahsavar, Philip K. Ahring, Jeppe A. Olsen, Christian Krintel, Jette S. Kastrup, Thomas Balle and Michael Gajhede
      Molecular Pharmacology October 2015, 88 (4) 697-707; DOI: https://doi.org/10.1124/mol.115.098061

  10. Kristensen, Anders S.

    1. Substrate and Inhibitor–Specific Conformational Changes in the Human Serotonin Transporter Revealed by Voltage-Clamp Fluorometry
      Pella C. Söderhielm, Jacob Andersen, Lachlan Munro, Anne T. Nielsen and Anders S. Kristensen
      Molecular Pharmacology October 2015, 88 (4) 676-688; DOI: https://doi.org/10.1124/mol.115.099911

L

  1. Lal, Jawahar

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

  2. Langmead, Christopher J.

    1. Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists
      Darren M. Riddy, Celine Valant, Patricia Rueda, William N. Charman, Patrick M. Sexton, Roger J. Summers, Arthur Christopoulos and Christopher J. Langmead
      Molecular Pharmacology October 2015, 88 (4) 779-790; DOI: https://doi.org/10.1124/mol.115.100545

  3. Lee, Min Goo

    1. Benzopyrimido-pyrrolo-oxazine-dione (R)-BPO-27 Inhibits CFTR Chloride Channel Gating by Competition with ATP
      Yonjung Kim, Marc O. Anderson, Jinhong Park, Min Goo Lee, Wan Namkung and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 689-696; DOI: https://doi.org/10.1124/mol.115.098368

  4. Lee, Minyoung

    1. Aspirin Targets SIRT1 and AMPK to Induce Senescence of Colorectal Carcinoma Cells
      Yu Ri Jung, Eun Ju Kim, Hyeong Jwa Choi, Jung-Jin Park, Hak-Su Kim, Yoon-Jin Lee, Myung-Jin Park and Minyoung Lee
      Molecular Pharmacology October 2015, 88 (4) 708-719; DOI: https://doi.org/10.1124/mol.115.098616

  5. Lee, Yoon-Jin

    1. Aspirin Targets SIRT1 and AMPK to Induce Senescence of Colorectal Carcinoma Cells
      Yu Ri Jung, Eun Ju Kim, Hyeong Jwa Choi, Jung-Jin Park, Hak-Su Kim, Yoon-Jin Lee, Myung-Jin Park and Minyoung Lee
      Molecular Pharmacology October 2015, 88 (4) 708-719; DOI: https://doi.org/10.1124/mol.115.098616

  6. Lewin, Amanda E.

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

  7. Lin, HongXia

    1. Suppression of Cytosolic NADPH Pool by Thionicotinamide Increases Oxidative Stress and Synergizes with Chemotherapy
      Philip M. Tedeschi, HongXia Lin, Murugesan Gounder, John E. Kerrigan, Emine Ercikan Abali, Kathleen Scotto and Joseph R. Bertino
      Molecular Pharmacology October 2015, 88 (4) 720-727; DOI: https://doi.org/10.1124/mol.114.096727

  8. Lukacs, Gergely L.

    1. Potentiators of Defective ΔF508–CFTR Gating that Do Not Interfere with Corrector Action
      Puay-Wah Phuan, Guido Veit, Joseph A. Tan, Walter E. Finkbeiner, Gergely L. Lukacs and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 791-799; DOI: https://doi.org/10.1124/mol.115.099689

M

  1. Mackenzie, Peter I.

    1. Suppression of Cytochrome P450 3A4 Function by UDP-Glucuronosyltransferase 2B7 through a Protein-Protein Interaction: Cooperative Roles of the Cytosolic Carboxyl-Terminal Domain and the Luminal Anchoring Region
      Yuu Miyauchi, Kiyoshi Nagata, Yasushi Yamazoe, Peter I. Mackenzie, Hideyuki Yamada and Yuji Ishii
      Molecular Pharmacology October 2015, 88 (4) 800-812; DOI: https://doi.org/10.1124/mol.115.098582

  2. Malik, Sundeep

    1. Adenylyl Cyclase 5 Regulation by G<em>βγ</em> Involves Isoform-Specific Use of Multiple Interaction Sites
      Adenylyl Cyclase 5 Regulation by Gβγ Involves Isoform-Specific Use of Multiple Interaction Sites
      Cameron S. Brand, Rachna Sadana, Sundeep Malik, Alan V. Smrcka and Carmen W. Dessauer
      Molecular Pharmacology October 2015, 88 (4) 758-767; DOI: https://doi.org/10.1124/mol.115.099556

  3. Miess, Elke

    1. Role of Phosphorylation Sites in Desensitization of µ-Opioid Receptor
      Arsalan Yousuf, Elke Miess, Setareh Sianati, Yan-Ping Du, Stefan Schulz and MacDonald J. Christie
      Molecular Pharmacology October 2015, 88 (4) 825-835; DOI: https://doi.org/10.1124/mol.115.098244

  4. Mishra, Anil K.

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

  5. Miyauchi, Yuu

    1. Suppression of Cytochrome P450 3A4 Function by UDP-Glucuronosyltransferase 2B7 through a Protein-Protein Interaction: Cooperative Roles of the Cytosolic Carboxyl-Terminal Domain and the Luminal Anchoring Region
      Yuu Miyauchi, Kiyoshi Nagata, Yasushi Yamazoe, Peter I. Mackenzie, Hideyuki Yamada and Yuji Ishii
      Molecular Pharmacology October 2015, 88 (4) 800-812; DOI: https://doi.org/10.1124/mol.115.098582

  6. Monaghan, Daniel T.

    1. Bidirectional Effect of Pregnenolone Sulfate on GluN1/GluN2A N-Methyl-d-Aspartate Receptor Gating Depending on Extracellular Calcium and Intracellular Milieu
      Divyan A. Chopra, Daniel T. Monaghan and Shashank M. Dravid
      Molecular Pharmacology October 2015, 88 (4) 650-659; DOI: https://doi.org/10.1124/mol.115.100396

  7. Munro, Lachlan

    1. Substrate and Inhibitor–Specific Conformational Changes in the Human Serotonin Transporter Revealed by Voltage-Clamp Fluorometry
      Pella C. Söderhielm, Jacob Andersen, Lachlan Munro, Anne T. Nielsen and Anders S. Kristensen
      Molecular Pharmacology October 2015, 88 (4) 676-688; DOI: https://doi.org/10.1124/mol.115.099911

N

  1. Nagata, Kiyoshi

    1. Suppression of Cytochrome P450 3A4 Function by UDP-Glucuronosyltransferase 2B7 through a Protein-Protein Interaction: Cooperative Roles of the Cytosolic Carboxyl-Terminal Domain and the Luminal Anchoring Region
      Yuu Miyauchi, Kiyoshi Nagata, Yasushi Yamazoe, Peter I. Mackenzie, Hideyuki Yamada and Yuji Ishii
      Molecular Pharmacology October 2015, 88 (4) 800-812; DOI: https://doi.org/10.1124/mol.115.098582

  2. Namkung, Wan

    1. Benzopyrimido-pyrrolo-oxazine-dione (R)-BPO-27 Inhibits CFTR Chloride Channel Gating by Competition with ATP
      Yonjung Kim, Marc O. Anderson, Jinhong Park, Min Goo Lee, Wan Namkung and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 689-696; DOI: https://doi.org/10.1124/mol.115.098368

  3. Negishi, Masahiko

    1. Pregnane X Receptor Represses HNF4α Gene to Induce Insulin-Like Growth Factor–Binding Protein IGFBP1 that Alters Morphology of and Migrates HepG2 Cells
      Susumu Kodama, Yuichi Yamazaki and Masahiko Negishi
      Molecular Pharmacology October 2015, 88 (4) 746-757; DOI: https://doi.org/10.1124/mol.115.099341

  4. Nielsen, Anne T.

    1. Substrate and Inhibitor–Specific Conformational Changes in the Human Serotonin Transporter Revealed by Voltage-Clamp Fluorometry
      Pella C. Söderhielm, Jacob Andersen, Lachlan Munro, Anne T. Nielsen and Anders S. Kristensen
      Molecular Pharmacology October 2015, 88 (4) 676-688; DOI: https://doi.org/10.1124/mol.115.099911

  5. Nimesh, Hemlata

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

O

  1. Olsen, Jeppe A.

    1. Acetylcholine-Binding Protein Engineered to Mimic the α4-α4 Binding Pocket in α4β2 Nicotinic Acetylcholine Receptors Reveals Interface Specific Interactions Important for Binding and Activity
      Azadeh Shahsavar, Philip K. Ahring, Jeppe A. Olsen, Christian Krintel, Jette S. Kastrup, Thomas Balle and Michael Gajhede
      Molecular Pharmacology October 2015, 88 (4) 697-707; DOI: https://doi.org/10.1124/mol.115.098061

  2. Olson, Thao T.

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

P

  1. Park, Jinhong

    1. Benzopyrimido-pyrrolo-oxazine-dione (R)-BPO-27 Inhibits CFTR Chloride Channel Gating by Competition with ATP
      Yonjung Kim, Marc O. Anderson, Jinhong Park, Min Goo Lee, Wan Namkung and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 689-696; DOI: https://doi.org/10.1124/mol.115.098368

  2. Park, Jung-Jin

    1. Aspirin Targets SIRT1 and AMPK to Induce Senescence of Colorectal Carcinoma Cells
      Yu Ri Jung, Eun Ju Kim, Hyeong Jwa Choi, Jung-Jin Park, Hak-Su Kim, Yoon-Jin Lee, Myung-Jin Park and Minyoung Lee
      Molecular Pharmacology October 2015, 88 (4) 708-719; DOI: https://doi.org/10.1124/mol.115.098616

  3. Park, Myung-Jin

    1. Aspirin Targets SIRT1 and AMPK to Induce Senescence of Colorectal Carcinoma Cells
      Yu Ri Jung, Eun Ju Kim, Hyeong Jwa Choi, Jung-Jin Park, Hak-Su Kim, Yoon-Jin Lee, Myung-Jin Park and Minyoung Lee
      Molecular Pharmacology October 2015, 88 (4) 708-719; DOI: https://doi.org/10.1124/mol.115.098616

  4. Phuan, Puay-Wah

    1. Potentiators of Defective ΔF508–CFTR Gating that Do Not Interfere with Corrector Action
      Puay-Wah Phuan, Guido Veit, Joseph A. Tan, Walter E. Finkbeiner, Gergely L. Lukacs and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 791-799; DOI: https://doi.org/10.1124/mol.115.099689

R

  1. Riddy, Darren M.

    1. Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists
      Darren M. Riddy, Celine Valant, Patricia Rueda, William N. Charman, Patrick M. Sexton, Roger J. Summers, Arthur Christopoulos and Christopher J. Langmead
      Molecular Pharmacology October 2015, 88 (4) 779-790; DOI: https://doi.org/10.1124/mol.115.100545

  2. Rueda, Patricia

    1. Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists
      Darren M. Riddy, Celine Valant, Patricia Rueda, William N. Charman, Patrick M. Sexton, Roger J. Summers, Arthur Christopoulos and Christopher J. Langmead
      Molecular Pharmacology October 2015, 88 (4) 779-790; DOI: https://doi.org/10.1124/mol.115.100545

S

  1. Sadana, Rachna

    1. Adenylyl Cyclase 5 Regulation by G<em>βγ</em> Involves Isoform-Specific Use of Multiple Interaction Sites
      Adenylyl Cyclase 5 Regulation by Gβγ Involves Isoform-Specific Use of Multiple Interaction Sites
      Cameron S. Brand, Rachna Sadana, Sundeep Malik, Alan V. Smrcka and Carmen W. Dessauer
      Molecular Pharmacology October 2015, 88 (4) 758-767; DOI: https://doi.org/10.1124/mol.115.099556

  2. Sahibzada, Niaz

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

  3. Schulz, Stefan

    1. Role of Phosphorylation Sites in Desensitization of µ-Opioid Receptor
      Arsalan Yousuf, Elke Miess, Setareh Sianati, Yan-Ping Du, Stefan Schulz and MacDonald J. Christie
      Molecular Pharmacology October 2015, 88 (4) 825-835; DOI: https://doi.org/10.1124/mol.115.098244

  4. Scotto, Kathleen

    1. Suppression of Cytosolic NADPH Pool by Thionicotinamide Increases Oxidative Stress and Synergizes with Chemotherapy
      Philip M. Tedeschi, HongXia Lin, Murugesan Gounder, John E. Kerrigan, Emine Ercikan Abali, Kathleen Scotto and Joseph R. Bertino
      Molecular Pharmacology October 2015, 88 (4) 720-727; DOI: https://doi.org/10.1124/mol.114.096727

  5. Sexton, Patrick M.

    1. Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists
      Darren M. Riddy, Celine Valant, Patricia Rueda, William N. Charman, Patrick M. Sexton, Roger J. Summers, Arthur Christopoulos and Christopher J. Langmead
      Molecular Pharmacology October 2015, 88 (4) 779-790; DOI: https://doi.org/10.1124/mol.115.100545

  6. Shahsavar, Azadeh

    1. Acetylcholine-Binding Protein Engineered to Mimic the α4-α4 Binding Pocket in α4β2 Nicotinic Acetylcholine Receptors Reveals Interface Specific Interactions Important for Binding and Activity
      Azadeh Shahsavar, Philip K. Ahring, Jeppe A. Olsen, Christian Krintel, Jette S. Kastrup, Thomas Balle and Michael Gajhede
      Molecular Pharmacology October 2015, 88 (4) 697-707; DOI: https://doi.org/10.1124/mol.115.098061

  7. Sharma, Abhisheak

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

  8. Sianati, Setareh

    1. Role of Phosphorylation Sites in Desensitization of µ-Opioid Receptor
      Arsalan Yousuf, Elke Miess, Setareh Sianati, Yan-Ping Du, Stefan Schulz and MacDonald J. Christie
      Molecular Pharmacology October 2015, 88 (4) 825-835; DOI: https://doi.org/10.1124/mol.115.098244

  9. Smrcka, Alan V.

    1. Adenylyl Cyclase 5 Regulation by G<em>βγ</em> Involves Isoform-Specific Use of Multiple Interaction Sites
      Adenylyl Cyclase 5 Regulation by Gβγ Involves Isoform-Specific Use of Multiple Interaction Sites
      Cameron S. Brand, Rachna Sadana, Sundeep Malik, Alan V. Smrcka and Carmen W. Dessauer
      Molecular Pharmacology October 2015, 88 (4) 758-767; DOI: https://doi.org/10.1124/mol.115.099556

  10. Söderhielm, Pella C.

    1. Substrate and Inhibitor–Specific Conformational Changes in the Human Serotonin Transporter Revealed by Voltage-Clamp Fluorometry
      Pella C. Söderhielm, Jacob Andersen, Lachlan Munro, Anne T. Nielsen and Anders S. Kristensen
      Molecular Pharmacology October 2015, 88 (4) 676-688; DOI: https://doi.org/10.1124/mol.115.099911

  11. Stockmeier, Craig A.

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

  12. Summers, Roger J.

    1. Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists
      Darren M. Riddy, Celine Valant, Patricia Rueda, William N. Charman, Patrick M. Sexton, Roger J. Summers, Arthur Christopoulos and Christopher J. Langmead
      Molecular Pharmacology October 2015, 88 (4) 779-790; DOI: https://doi.org/10.1124/mol.115.100545

T

  1. Tan, Joseph A.

    1. Potentiators of Defective ΔF508–CFTR Gating that Do Not Interfere with Corrector Action
      Puay-Wah Phuan, Guido Veit, Joseph A. Tan, Walter E. Finkbeiner, Gergely L. Lukacs and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 791-799; DOI: https://doi.org/10.1124/mol.115.099689

  2. Tanaka, Yoshitaka

    1. Intracellular Dynamics and Fate of a Humanized Anti–Interleukin-6 Receptor Monoclonal Antibody, Tocilizumab
      Keiko Fujimoto, Hiroaki Ida, Yuko Hirota, Masaki Ishigai, Jun Amano and Yoshitaka Tanaka
      Molecular Pharmacology October 2015, 88 (4) 660-675; DOI: https://doi.org/10.1124/mol.115.099184

  3. Tandon, Vibha

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

  4. Tavalin, Steven J.

    1. Protein Kinase C (PKC)ζ Pseudosubstrate Inhibitor Peptide Promiscuously Binds PKC Family Isoforms and Disrupts Conventional PKC Targeting and Translocation
      Amy S. Bogard and Steven J. Tavalin
      Molecular Pharmacology October 2015, 88 (4) 728-735; DOI: https://doi.org/10.1124/mol.115.099457

  5. Tedeschi, Philip M.

    1. Suppression of Cytosolic NADPH Pool by Thionicotinamide Increases Oxidative Stress and Synergizes with Chemotherapy
      Philip M. Tedeschi, HongXia Lin, Murugesan Gounder, John E. Kerrigan, Emine Ercikan Abali, Kathleen Scotto and Joseph R. Bertino
      Molecular Pharmacology October 2015, 88 (4) 720-727; DOI: https://doi.org/10.1124/mol.114.096727

  6. Tiwari, Vinod

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

  7. Tuan, Edward W.

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

V

  1. Valant, Celine

    1. Label-Free Kinetics: Exploiting Functional Hemi-Equilibrium to Derive Rate Constants for Muscarinic Receptor Antagonists
      Darren M. Riddy, Celine Valant, Patricia Rueda, William N. Charman, Patrick M. Sexton, Roger J. Summers, Arthur Christopoulos and Christopher J. Langmead
      Molecular Pharmacology October 2015, 88 (4) 779-790; DOI: https://doi.org/10.1124/mol.115.100545

  2. Veit, Guido

    1. Potentiators of Defective ΔF508–CFTR Gating that Do Not Interfere with Corrector Action
      Puay-Wah Phuan, Guido Veit, Joseph A. Tan, Walter E. Finkbeiner, Gergely L. Lukacs and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 791-799; DOI: https://doi.org/10.1124/mol.115.099689

  3. Verkman, A. S.

    1. Benzopyrimido-pyrrolo-oxazine-dione (R)-BPO-27 Inhibits CFTR Chloride Channel Gating by Competition with ATP
      Yonjung Kim, Marc O. Anderson, Jinhong Park, Min Goo Lee, Wan Namkung and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 689-696; DOI: https://doi.org/10.1124/mol.115.098368
    2. Potentiators of Defective ΔF508–CFTR Gating that Do Not Interfere with Corrector Action
      Puay-Wah Phuan, Guido Veit, Joseph A. Tan, Walter E. Finkbeiner, Gergely L. Lukacs and A. S. Verkman
      Molecular Pharmacology October 2015, 88 (4) 791-799; DOI: https://doi.org/10.1124/mol.115.099689

W

  1. Williams, John T.

    1. Agonist Binding and Desensitization of the μ-Opioid Receptor Is Modulated by Phosphorylation of the C-Terminal Tail Domain
      William T. Birdsong, Seksiri Arttamangkul, James R. Bunzow and John T. Williams
      Molecular Pharmacology October 2015, 88 (4) 816-824; DOI: https://doi.org/10.1124/mol.114.097527

  2. Wolfe, Barry B.

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

X

  1. Xiao, Yingxian

    1. AT-1001 Is a Partial Agonist with High Affinity and Selectivity at Human and Rat α3β4 Nicotinic Cholinergic Receptors
      Edward W. Tuan, Andrew G. Horti, Thao T. Olson, Yongiun Gao, Craig A. Stockmeier, Nour Al-Muhtasib, Carrie Bowman Dalley, Amanda E. Lewin, Barry B. Wolfe, Niaz Sahibzada, Yingxian Xiao and Kenneth J. Kellar
      Molecular Pharmacology October 2015, 88 (4) 640-649; DOI: https://doi.org/10.1124/mol.115.099978

Y

  1. Yamada, Hideyuki

    1. Suppression of Cytochrome P450 3A4 Function by UDP-Glucuronosyltransferase 2B7 through a Protein-Protein Interaction: Cooperative Roles of the Cytosolic Carboxyl-Terminal Domain and the Luminal Anchoring Region
      Yuu Miyauchi, Kiyoshi Nagata, Yasushi Yamazoe, Peter I. Mackenzie, Hideyuki Yamada and Yuji Ishii
      Molecular Pharmacology October 2015, 88 (4) 800-812; DOI: https://doi.org/10.1124/mol.115.098582

  2. Yamazaki, Yuichi

    1. Pregnane X Receptor Represses HNF4α Gene to Induce Insulin-Like Growth Factor–Binding Protein IGFBP1 that Alters Morphology of and Migrates HepG2 Cells
      Susumu Kodama, Yuichi Yamazaki and Masahiko Negishi
      Molecular Pharmacology October 2015, 88 (4) 746-757; DOI: https://doi.org/10.1124/mol.115.099341

  3. Yamazoe, Yasushi

    1. Suppression of Cytochrome P450 3A4 Function by UDP-Glucuronosyltransferase 2B7 through a Protein-Protein Interaction: Cooperative Roles of the Cytosolic Carboxyl-Terminal Domain and the Luminal Anchoring Region
      Yuu Miyauchi, Kiyoshi Nagata, Yasushi Yamazoe, Peter I. Mackenzie, Hideyuki Yamada and Yuji Ishii
      Molecular Pharmacology October 2015, 88 (4) 800-812; DOI: https://doi.org/10.1124/mol.115.098582

  4. Yang, Chunhua

    1. Preclinical Evaluation of DMA, a Bisbenzimidazole, as Radioprotector: Toxicity, Pharmacokinetics, and Biodistribution Studies in Balb/c Mice
      Hemlata Nimesh, Vinod Tiwari, Chunhua Yang, Sushma R. Gundala, Krishna Chuttani, Puja P. Hazari, Anil K. Mishra, Abhisheak Sharma, Jawahar Lal, Anju Katyal, Ritu Aneja and Vibha Tandon
      Molecular Pharmacology October 2015, 88 (4) 768-778; DOI: https://doi.org/10.1124/mol.115.098376

  5. Yousuf, Arsalan

    1. Role of Phosphorylation Sites in Desensitization of µ-Opioid Receptor
      Arsalan Yousuf, Elke Miess, Setareh Sianati, Yan-Ping Du, Stefan Schulz and MacDonald J. Christie
      Molecular Pharmacology October 2015, 88 (4) 825-835; DOI: https://doi.org/10.1124/mol.115.098244
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