Table of Contents

Articles

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  Comparison of Steroid Modulation of Spontaneous Inhibitory Postsynaptic Currents in Cultured Hippocampal Neurons and Steady-State Single-Channel Currents from Heterologously Expressed α1β2γ2L GABA_A Receptors

  Sampurna Chakrabarti, Mingxing Qian, Kathiresan Krishnan, Douglas F. Covey, Steven Mennerick and Gustav Akk

  Molecular Pharmacology April 2016, 89 (4) 399-406; DOI: https://doi.org/10.1124/mol.115.102202
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  Correlation between Activity and Domain Complementation in Adenylyl Cyclase Demonstrated with a Novel Fluorescence Resonance Energy Transfer Sensor

  Michael Ritt and Sivaraj Sivaramakrishnan

  Molecular Pharmacology April 2016, 89 (4) 407-412; DOI: https://doi.org/10.1124/mol.115.101626
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  Binding to and Inhibition of Insulin-Regulated Aminopeptidase by Macrocyclic Disulfides Enhances Spine Density

  Shanti Diwakarla, Erik Nylander, Alfhild Grönbladh, Sudarsana Reddy Vanga, Yasmin Shamsudin Khan, Hugo Gutiérrez-de-Terán, Leelee Ng, Vi Pham, Jonas Sävmarker, Thomas Lundbäck, Annika Jenmalm-Jensen, Hanna Andersson, Karin Engen, Ulrika Rosenström, Mats Larhed, Johan Åqvist, Siew Yeen Chai and Mathias Hallberg

  Molecular Pharmacology April 2016, 89 (4) 413-424; DOI: https://doi.org/10.1124/mol.115.102533
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  Targeting Nonsquamous Nonsmall Cell Lung Cancer via the Proton-Coupled Folate Transporter with 6-Substituted Pyrrolo[2,3-d]Pyrimidine Thienoyl Antifolates

  Mike R. Wilson, Zhanjun Hou, Si Yang, Lisa Polin, Juiwanna Kushner, Kathryn White, Jenny Huang, Manohar Ratnam, Aleem Gangjee and Larry H. Matherly

  Molecular Pharmacology April 2016, 89 (4) 425-434; DOI: https://doi.org/10.1124/mol.115.102798
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  Structure-Function Analysis of Mammalian CYP2B Enzymes Using 7-Substituted Coumarin Derivatives as Probes: Utility of Crystal Structures and Molecular Modeling in Understanding Xenobiotic Metabolism

  Manish B. Shah, Jingbao Liu, Lu Huo, Qinghai Zhang, M. Denise Dearing, P. Ross Wilderman, Grazyna D. Szklarz, C. David Stout and James R. Halpert

  Molecular Pharmacology April 2016, 89 (4) 435-445; DOI: https://doi.org/10.1124/mol.115.102111
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  Dipicrylamine Modulates GABAρ1 Receptors through Interactions with Residues in the TM4 and Cys-Loop Domains

  Agenor Limon, Argel Estrada-Mondragón, Jorge M. Reyes Ruiz and Ricardo Miledi

  Molecular Pharmacology April 2016, 89 (4) 446-456; DOI: https://doi.org/10.1124/mol.116.103432
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  Evidence for Noncanonical Neurotransmitter Activation: Norepinephrine as a Dopamine D₂-Like Receptor Agonist

  Marta Sánchez-Soto, Alessandro Bonifazi, Ning Sheng Cai, Michael P. Ellenberger, Amy Hauck Newman, Sergi Ferré and Hideaki Yano

  Molecular Pharmacology April 2016, 89 (4) 457-466; DOI: https://doi.org/10.1124/mol.115.101808
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  Long Receptor Residence Time of C26 Contributes to Super Agonist Activity at the Human β₂ Adrenoceptor

  Elizabeth M. Rosethorne, Michelle E. Bradley, Karolina Gherbi, David A. Sykes, Afrah Sattikar, John D. Wright, Emilie Renard, Alex Trifilieff, Robin A. Fairhurst and Steven J. Charlton

  Molecular Pharmacology April 2016, 89 (4) 467-475; DOI: https://doi.org/10.1124/mol.115.101253
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  Voltage-Independent Inhibition of the Tetrodotoxin-Sensitive Sodium Currents by Oxotremorine and Angiotensin II in Rat Sympathetic Neurons

  Erika I. Puente, Lizbeth De la Cruz, Isabel Arenas, David Elias-Viñas and David E. Garcia

  Molecular Pharmacology April 2016, 89 (4) 476-483; DOI: https://doi.org/10.1124/mol.115.101931