Table of Contents

Articles

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  GluN2D-Containing N-methyl-d-Aspartate Receptors Mediate Synaptic Transmission in Hippocampal Interneurons and Regulate Interneuron Activity

  Riley E. Perszyk, John O. DiRaddo, Katie L. Strong, Chian-Ming Low, Kevin K. Ogden, Alpa Khatri, Geoffrey A. Vargish, Kenneth A. Pelkey, Ludovic Tricoire, Dennis C. Liotta, Yoland Smith, Chris J. McBain and Stephen F. Traynelis

  Molecular Pharmacology December 2016, 90 (6) 689-702; DOI: https://doi.org/10.1124/mol.116.105130
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  Extracellular Loop 2 of the Adenosine A₁ Receptor Has a Key Role in Orthosteric Ligand Affinity and Agonist Efficacy

  Anh T.N. Nguyen, Jo-Anne Baltos, Trayder Thomas, Toan D. Nguyen, Laura López Muñoz, Karen J. Gregory, Paul J. White, Patrick M. Sexton, Arthur Christopoulos and Lauren T. May

  Molecular Pharmacology December 2016, 90 (6) 703-714; DOI: https://doi.org/10.1124/mol.116.105007
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  Role of the Second Extracellular Loop of the Adenosine A₁ Receptor on Allosteric Modulator Binding, Signaling, and Cooperativity

  Anh T. N. Nguyen, Elizabeth A. Vecchio, Trayder Thomas, Toan D. Nguyen, Luigi Aurelio, Peter J. Scammells, Paul J. White, Patrick M. Sexton, Karen J. Gregory, Lauren T. May and Arthur Christopoulos

  Molecular Pharmacology December 2016, 90 (6) 715-725; DOI: https://doi.org/10.1124/mol.116.105015
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  Discovery and Characterization of Novel GPR39 Agonists Allosterically Modulated by Zinc

  Seiji Sato, Xi-Ping Huang, Wesley K. Kroeze and Bryan L. Roth

  Molecular Pharmacology December 2016, 90 (6) 726-737; DOI: https://doi.org/10.1124/mol.116.106112
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  Molecular Basis for Inhibition of the Na⁺/Citrate Transporter NaCT (SLC13A5) by Dicarboxylate Inhibitors

  Ana M. Pajor, Cesar A. de Oliveira, Kun Song, Kim Huard, Veerabahu Shanmugasundaram and Derek M. Erion

  Molecular Pharmacology December 2016, 90 (6) 755-765; DOI: https://doi.org/10.1124/mol.116.105049
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  State-Dependent Allosteric Inhibition of the Human SLC13A5 Citrate Transporter by Hydroxysuccinic Acids, PF-06649298 and PF-06761281

  Marie-Laure Rives, Morena Shaw, Bin Zhu, Simon A. Hinke and Alan D. Wickenden

  Molecular Pharmacology December 2016, 90 (6) 766-774; DOI: https://doi.org/10.1124/mol.116.106575