Table of Contents

Articles

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  Cannabinoid Receptor Interacting Protein 1a Competition with β-Arrestin for CB₁ Receptor Binding Sites

  Lawrence C. Blume, Theresa Patten, Khalil Eldeeb, Sandra Leone-Kabler, Alexander A. Ilyasov, Bradley M. Keegan, Jeremy E. O’Neal, Caroline E. Bass, Roy R. Hantgan, W. Todd Lowther, Dana E. Selley and A­llyn C. Howlett

  Molecular Pharmacology February 2017, 91 (2) 75-86; DOI: https://doi.org/10.1124/mol.116.104638
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  Isoform-Specific Biased Agonism of Histamine H₃ Receptor Agonists

  Darren M. Riddy, Anna E. Cook, Natalie A. Diepenhorst, Sanja Bosnyak, Ryan Brady, Clotilde Mannoury la Cour, Elisabeth Mocaer, Roger J. Summers, William N. Charman, Patrick M. Sexton, Arthur Christopoulos and Christopher J. Langmead

  Molecular Pharmacology February 2017, 91 (2) 87-99; DOI: https://doi.org/10.1124/mol.116.106153
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  The E Loop of the Transmitter Binding Site Is a Key Determinant of the Modulatory Effects of Physostigmine on Neuronal Nicotinic α4β2 Receptors

  Xiaochun Jin, Megan M. McCollum, Allison L. Germann, Gustav Akk and Joe Henry Steinbach

  Molecular Pharmacology February 2017, 91 (2) 100-109; DOI: https://doi.org/10.1124/mol.116.106484
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  Orally Administered Berberine Modulates Hepatic Lipid Metabolism by Altering Microbial Bile Acid Metabolism and the Intestinal FXR Signaling Pathway

  Runbin Sun, Na Yang, Bo Kong, Bei Cao, Dong Feng, Xiaoyi Yu, Chun Ge, Jingqiu Huang, Jianliang Shen, Pei Wang, Siqi Feng, Fei Fei, Jiahua Guo, Jun He, Nan Aa, Qiang Chen, Yang Pan, Justin D. Schumacher, Chung S. Yang, Grace L. Guo, Jiye Aa and Guangji Wang

  Molecular Pharmacology February 2017, 91 (2) 110-122; DOI: https://doi.org/10.1124/mol.116.106617
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  Homobivalent Conjugation Increases the Allosteric Effect of 9-aminoacridine at the α₁-Adrenergic Receptors

  Adrian P. Campbell, Laurence P. G. Wakelin, William A. Denny and Angela M. Finch

  Molecular Pharmacology February 2017, 91 (2) 135-144; DOI: https://doi.org/10.1124/mol.116.105874
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  G Protein–Coupled Receptor Endocytosis Confers Uniformity in Responses to Chemically Distinct Ligands

  Nikoleta G. Tsvetanova, Michelle Trester-Zedlitz, Billy W. Newton, Daniel P. Riordan, Aparna B. Sundaram, Jeffrey R. Johnson, Nevan J. Krogan and Mark von Zastrow

  Molecular Pharmacology February 2017, 91 (2) 145-156; DOI: https://doi.org/10.1124/mol.116.106369