Table of Contents

Articles

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  Targeted Degradation of Proteins Localized in Subcellular Compartments by Hybrid Small Molecules

  Keiichiro Okuhira, Takuji Shoda, Risa Omura, Nobumichi Ohoka, Takayuki Hattori, Norihito Shibata, Yosuke Demizu, Ryo Sugihara, Asato Ichino, Haruka Kawahara, Yukihiro Itoh, Minoru Ishikawa, Yuichi Hashimoto, Masaaki Kurihara, Susumu Itoh, Hiroyuki Saito and Mikihiko Naito

  Molecular Pharmacology March 2017, 91 (3) 159-166; DOI: https://doi.org/10.1124/mol.116.105569
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  Cross-Talk between Alternatively Spliced UGT1A Isoforms and Colon Cancer Cell Metabolism

  Yannick Audet-Delage, Michèle Rouleau, Mélanie Rouleau, Joannie Roberge, Stéphanie Miard, Frédéric Picard, Bernard Têtu and Chantal Guillemette

  Molecular Pharmacology March 2017, 91 (3) 167-177; DOI: https://doi.org/10.1124/mol.116.106161
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  Circadian Regulation of Benzo[a]Pyrene Metabolism and DNA Adduct Formation in Breast Cells and the Mouse Mammary Gland

  Emily E. Schmitt, Rola Barhoumi, Richard P. Metz and Weston W. Porter

  Molecular Pharmacology March 2017, 91 (3) 178-188; DOI: https://doi.org/10.1124/mol.116.106740
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  Pyruvate Dehydrogenase Kinase 4 Deficiency Results in Expedited Cellular Proliferation through E2F1-Mediated Increase of Cyclins

  Jonathan Choiniere, Jianguo Wu and Li Wang

  Molecular Pharmacology March 2017, 91 (3) 189-196; DOI: https://doi.org/10.1124/mol.116.106757
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  Regulator of G Protein Signaling 10 (Rgs10) Expression Is Transcriptionally Silenced in Activated Microglia by Histone Deacetylase Activity

  Mohammed Alqinyah, Nagini Maganti, Mourad W. Ali, Ruchi Yadav, Mei Gao, Ercan Cacan, Han-Rong Weng, Susanna F. Greer and Shelley B. Hooks

  Molecular Pharmacology March 2017, 91 (3) 197-207; DOI: https://doi.org/10.1124/mol.116.106963
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  Ability of Bruton’s Tyrosine Kinase Inhibitors to Sequester Y551 and Prevent Phosphorylation Determines Potency for Inhibition of Fc Receptor but not B-Cell Receptor Signaling

  Andrew T. Bender, Anna Gardberg, Albertina Pereira, Theresa Johnson, Yin Wu, Roland Grenningloh, Jared Head, Federica Morandi, Philipp Haselmayer and Lesley Liu-Bujalski

  Molecular Pharmacology March 2017, 91 (3) 208-219; DOI: https://doi.org/10.1124/mol.116.107037
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  Olefin Isomers of a Triazole Bisphosphonate Synergistically Inhibit Geranylgeranyl Diphosphate Synthase

  Cheryl Allen, Sandhya Kortagere, Huaxiang Tong, Robert A. Matthiesen, Joseph I. Metzger, David F. Wiemer and Sarah A. Holstein

  Molecular Pharmacology March 2017, 91 (3) 229-236; DOI: https://doi.org/10.1124/mol.116.107326
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  Buprenorphine, Norbuprenorphine, R-Methadone, and S-Methadone Upregulate BCRP/ABCG2 Expression by Activating Aryl Hydrocarbon Receptor in Human Placental Trophoblasts

  Naveen K. Neradugomma, Michael Z. Liao and Qingcheng Mao

  Molecular Pharmacology March 2017, 91 (3) 237-249; DOI: https://doi.org/10.1124/mol.116.107367
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  Differential Contribution of Subunit Interfaces to α9α10 Nicotinic Acetylcholine Receptor Function

  Juan Carlos Boffi, Irina Marcovich, JasKiran K. Gill-Thind, Jeremías Corradi, Toby Collins, María Marcela Lipovsek, Marcelo Moglie, Paola V. Plazas, Patricio O. Craig, Neil S. Millar, Cecilia Bouzat and Ana Belén Elgoyhen

  Molecular Pharmacology March 2017, 91 (3) 250-262; DOI: https://doi.org/10.1124/mol.116.107482