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Molecular Pharmacology

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Table of Contents

October 01, 2017; Volume 92,Issue 4

Minireview

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    A Scale of Agonism and Allosteric Modulation for Assessment of Selectivity, Bias, and Receptor Mutation
    Terry Kenakin
    Molecular Pharmacology October 2017, 92 (4) 414-424; DOI: https://doi.org/10.1124/mol.117.108787

Articles

  • Open Access
    NO-Sensitive Guanylate Cyclase Isoforms NO-GC1 and NO-GC2 Contribute to Noise-Induced Inner Hair Cell Synaptopathy
    Dorit Möhrle, Katrin Reimann, Steffen Wolter, Markus Wolters, Ksenya Varakina, Evanthia Mergia, Nicole Eichert, Hyun-Soon Geisler, Peter Sandner, Peter Ruth, Andreas Friebe, Robert Feil, Ulrike Zimmermann, Doris Koesling, Marlies Knipper and Lukas Rüttiger
    Molecular Pharmacology October 2017, 92 (4) 375-388; DOI: https://doi.org/10.1124/mol.117.108548
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    A Novel Selective Inverse Agonist of the CB2 Receptor as a Radiolabeled Tool Compound for Kinetic Binding Studies
    Andrea Martella, Huub Sijben, Arne C. Rufer, Uwe Grether, Juergen Fingerle, Christoph Ullmer, Thomas Hartung, Adriaan P. IJzerman, Mario van der Stelt and Laura H. Heitman
    Molecular Pharmacology October 2017, 92 (4) 389-400; DOI: https://doi.org/10.1124/mol.117.108605
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    Molecular Mechanism of Taurocholate Transport by the Bile Salt Export Pump, an ABC Transporter Associated with Intrahepatic Cholestasis
    Muhammad Imran Sohail, Diethart Schmid, Katrin Wlcek, Matthias Spork, Gergely Szakács, Michael Trauner, Thomas Stockner and Peter Chiba
    Molecular Pharmacology October 2017, 92 (4) 401-413; DOI: https://doi.org/10.1124/mol.117.108688
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    Altenusin, a Nonsteroidal Microbial Metabolite, Attenuates Nonalcoholic Fatty Liver Disease by Activating the Farnesoid X Receptor
    Zhihui Zheng, Zanmei Zhao, Shuqiang Li, Xinhua Lu, Mengxi Jiang, Jie Lin, Yunqi An, Yang Xie, Meishu Xu, Wenbin Shen, Grace L. Guo, Yixian Huang, Song Li, Xuexia Zhang and Wen Xie
    Molecular Pharmacology October 2017, 92 (4) 425-436; DOI: https://doi.org/10.1124/mol.117.108829
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    Molecular Basis of Altered hERG1 Channel Gating Induced by Ginsenoside Rg3
    Alison Gardner, Wei Wu, Steven Thomson, Eva-Maria Zangerl-Plessl, Anna Stary-Weinzinger and Michael C. Sanguinetti
    Molecular Pharmacology October 2017, 92 (4) 437-450; DOI: https://doi.org/10.1124/mol.117.108886
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    Human Missense Mutations in Regulator of G Protein Signaling 2 Affect the Protein Function Through Multiple Mechanisms
    Hoa T.N. Phan, Benita Sjögren and Richard R. Neubig
    Molecular Pharmacology October 2017, 92 (4) 451-458; DOI: https://doi.org/10.1124/mol.117.109215
  • Open Access
    Suramin Inhibits Osteoarthritic Cartilage Degradation by Increasing Extracellular Levels of Chondroprotective Tissue Inhibitor of Metalloproteinases 3
    Anastasios Chanalaris, Christine Doherty, Brian D. Marsden, Gabriel Bambridge, Stephen P. Wren, Hideaki Nagase and Linda Troeberg
    Molecular Pharmacology October 2017, 92 (4) 459-468; DOI: https://doi.org/10.1124/mol.117.109397
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    Structural Determinants for the Selectivity of the Positive KCa3.1 Gating Modulator 5-Methylnaphtho[2,1-d]oxazol-2-amine (SKA-121)
    Brandon M. Brown, Heesung Shim, Miao Zhang, Vladimir Yarov-Yarovoy and Heike Wulff
    Molecular Pharmacology October 2017, 92 (4) 469-480; DOI: https://doi.org/10.1124/mol.117.109421
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    Nitro-Oleic Acid Regulates Endothelin Signaling in Human Endothelial Cells
    Emilia Kansanen, Suvi M. Kuosmanen, Anna-Kaisa Ruotsalainen, Heidi Hynynen and Anna-Liisa Levonen
    Molecular Pharmacology October 2017, 92 (4) 481-490; DOI: https://doi.org/10.1124/mol.117.109751
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    Splice Variants of pH-Sensitive Chloride Channel Identify a Key Determinant of Ivermectin Sensitivity in the Larvae of the Silkworm Bombyx mori
    Daiki Okuhara, Shogo Furutani, Katsuhiko Ito, Makoto Ihara and Kazuhiko Matsuda
    Molecular Pharmacology October 2017, 92 (4) 491-499; DOI: https://doi.org/10.1124/mol.117.109199

Erratum

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    Correction to “6-Mercaptopurine Decreases the Bcl-2/Bax Ratio and Induces Apoptosis in Activated Splenic B Lymphocytes”
    Molecular Pharmacology October 2017, 92 (4) 500; DOI: https://doi.org/10.1124/mol.111.513err
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In this issue

Molecular Pharmacology: 92 (4)
Molecular Pharmacology
Vol. 92, Issue 4
1 Oct 2017
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  • SB-431542 Is a Potent and Specific Inhibitor of Transforming Growth Factor-β Superfamily Type I Activin Receptor-Like Kinase (ALK) Receptors ALK4, ALK5, and ALK7
  • The G-Protein-Coupled Receptors in the Human Genome Form Five Main Families. Phylogenetic Analysis, Paralogon Groups, and Fingerprints
  • Pharmacological Properties of Y-27632, a Specific Inhibitor of Rho-Associated Kinases
  • Pharmacological characterization of five cloned voltage-gated K+ channels, types Kv1.1, 1.2, 1.3, 1.5, and 3.1, stably expressed in mammalian cell lines.
  • The Orphan Human Pregnane X Receptor Mediates the Transcriptional Activation of CYP3A4 by Rifampicin through a Distal Enhancer Module
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