Table of Contents

Articles

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  Effective Attenuation of Adenosine A1R Signaling by Neurabin Requires Oligomerization of Neurabin

  Yunjia Chen, Christopher Booth, Hongxia Wang, Raymond X. Wang, Dimitra Terzi, Venetia Zachariou, Kai Jiao, Jin Zhang and Qin Wang

  Molecular Pharmacology December 2017, 92 (6) 630-639; DOI: https://doi.org/10.1124/mol.117.109462
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  Activation of AMPK/mTORC1-Mediated Autophagy by Metformin Reverses Clk1 Deficiency-Sensitized Dopaminergic Neuronal Death

  Qiuting Yan, Chaojun Han, Guanghui Wang, John L. Waddington, Longtai Zheng and Xuechu Zhen

  Molecular Pharmacology December 2017, 92 (6) 640-652; DOI: https://doi.org/10.1124/mol.117.109512
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  Activation of Human Transient Receptor Potential Melastatin-8 (TRPM8) by Calcium-Rich Particulate Materials and Effects on Human Lung Cells

  John G. Lamb, Erin G. Romero, Zhenyu Lu, Seychelle K. Marcus, Hannah C. Peterson, John M. Veranth, Cassandra E. Deering-Rice and Christopher A. Reilly

  Molecular Pharmacology December 2017, 92 (6) 653-664; DOI: https://doi.org/10.1124/mol.117.109959
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  Diminazene Is a Slow Pore Blocker of Acid-Sensing Ion Channel 1a (ASIC1a)

  Axel Schmidt, Giulia Rossetti, Sylvia Joussen and Stefan Gründer

  Molecular Pharmacology December 2017, 92 (6) 665-675; DOI: https://doi.org/10.1124/mol.117.110064
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  RVX-297, a BET Bromodomain Inhibitor, Has Therapeutic Effects in Preclinical Models of Acute Inflammation and Autoimmune Disease

  Ravi Jahagirdar, Sarah Attwell, Suzana Marusic, Alison Bendele, Narmada Shenoy, Kevin G. McLure, Dean Gilham, Karen Norek, Henrik C. Hansen, Raymond Yu, Jennifer Tobin, Gregory S. Wagner, Peter R. Young, Norman C. W. Wong and Ewelina Kulikowski

  Molecular Pharmacology December 2017, 92 (6) 694-706; DOI: https://doi.org/10.1124/mol.117.110379
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  Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein–Coupled Receptor Kinase 2 Inhibitors

  Renee Bouley, Helen V. Waldschmidt, M. Claire Cato, Alessandro Cannavo, Jianliang Song, Joseph Y. Cheung, Xin-Qiu Yao, Walter J. Koch, Scott D. Larsen and John J. G. Tesmer

  Molecular Pharmacology December 2017, 92 (6) 707-717; DOI: https://doi.org/10.1124/mol.117.110130
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  Hydrogen Sulfide Preserves Endothelial Nitric Oxide Synthase Function by Inhibiting Proline-Rich Kinase 2: Implications for Cardiomyocyte Survival and Cardioprotection

  Sofia-Iris Bibli, Csaba Szabo, Athanasia Chatzianastasiou, Bert Luck, Sven Zukunft, Ingrid Fleming and Andreas Papapetropoulos

  Molecular Pharmacology December 2017, 92 (6) 718-730; DOI: https://doi.org/10.1124/mol.117.109645