Index by author
February 01, 2018; Volume 93,Issue 2
A
Akk, Gustav
- You have accessGABA Type A Receptor Activation in the Allosteric Coagonist Model Framework: Relationship between EC50 and Basal ActivityGustav Akk, Daniel J. Shin, Allison L. Germann and Joe Henry SteinbachMolecular Pharmacology February 2018, 93 (2) 90-100; DOI: https://doi.org/10.1124/mol.117.110569
- You have accessPropofol Is an Allosteric Agonist with Multiple Binding Sites on Concatemeric Ternary GABAA ReceptorsDaniel J. Shin, Allison L. Germann, Alexander D. Johnson, Stuart A. Forman, Joe Henry Steinbach and Gustav AkkMolecular Pharmacology February 2018, 93 (2) 178-189; DOI: https://doi.org/10.1124/mol.117.110403
Alt, Andrew
- You have accessPharmacologic Evidence for a Putative Conserved Allosteric Site on Opioid ReceptorsKathryn E. Livingston, M. Alexander Stanczyk, Neil T. Burford, Andrew Alt, Meritxell Canals and John R. TraynorMolecular Pharmacology February 2018, 93 (2) 157-167; DOI: https://doi.org/10.1124/mol.117.109561
B
Bhattacharya, Subhrajit
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
Birker-Robaczewska, Magdalena
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
Bolli, Martin
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
Boucher, Maxime
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
Bouvet, Vincent
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Burford, Neil T.
- You have accessPharmacologic Evidence for a Putative Conserved Allosteric Site on Opioid ReceptorsKathryn E. Livingston, M. Alexander Stanczyk, Neil T. Burford, Andrew Alt, Meritxell Canals and John R. TraynorMolecular Pharmacology February 2018, 93 (2) 157-167; DOI: https://doi.org/10.1124/mol.117.109561
Burger, Pieter B.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
C
Canals, Meritxell
- You have accessPharmacologic Evidence for a Putative Conserved Allosteric Site on Opioid ReceptorsKathryn E. Livingston, M. Alexander Stanczyk, Neil T. Burford, Andrew Alt, Meritxell Canals and John R. TraynorMolecular Pharmacology February 2018, 93 (2) 157-167; DOI: https://doi.org/10.1124/mol.117.109561
Chatzidaki, Anna
- Open AccessDiversity of Nicotinic Acetylcholine Receptor Positive Allosteric Modulators Revealed by Mutagenesis and a Revised Structural ModelJoseph Newcombe, Anna Chatzidaki, Tom D. Sheppard, Maya Topf and Neil S. MillarMolecular Pharmacology February 2018, 93 (2) 128-140; DOI: https://doi.org/10.1124/mol.117.110551
Cheeseman, Chris
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Chen, Taosheng
- You have accessPXR: More Than Just a Master Xenobiotic ReceptorPeter O. Oladimeji and Taosheng ChenMolecular Pharmacology February 2018, 93 (2) 119-127; DOI: https://doi.org/10.1124/mol.117.110155
Cox, Bryan D.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
D
De Iuliis, Geoffry N.
- You have access(Z)-2-(3,4-Dichlorophenyl)-3-(1H-Pyrrol-2-yl)Acrylonitrile Exhibits Selective Antitumor Activity in Breast Cancer Cell Lines via the Aryl Hydrocarbon Receptor PathwayJayne Gilbert, Geoffry N. De Iuliis, Mark Tarleton, Adam McCluskey and Jennette A. SakoffMolecular Pharmacology February 2018, 93 (2) 168-177; DOI: https://doi.org/10.1124/mol.117.109827
de Kanter, Ruben
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
Dhopeshwarkar, Amey S.
- You have accessSlowly Signaling G Protein–Biased CB2 Cannabinoid Receptor Agonist LY2828360 Suppresses Neuropathic Pain with Sustained Efficacy and Attenuates Morphine Tolerance and DependenceXiaoyan Lin, Amey S. Dhopeshwarkar, Megan Huibregtse, Ken Mackie and Andrea G. HohmannMolecular Pharmacology February 2018, 93 (2) 49-62; DOI: https://doi.org/10.1124/mol.117.109355
E
Epplin, Matthew P.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
F
Forman, Stuart A.
- You have accessPropofol Is an Allosteric Agonist with Multiple Binding Sites on Concatemeric Ternary GABAA ReceptorsDaniel J. Shin, Allison L. Germann, Alexander D. Johnson, Stuart A. Forman, Joe Henry Steinbach and Gustav AkkMolecular Pharmacology February 2018, 93 (2) 178-189; DOI: https://doi.org/10.1124/mol.117.110403
G
Germann, Allison L.
- You have accessGABA Type A Receptor Activation in the Allosteric Coagonist Model Framework: Relationship between EC50 and Basal ActivityGustav Akk, Daniel J. Shin, Allison L. Germann and Joe Henry SteinbachMolecular Pharmacology February 2018, 93 (2) 90-100; DOI: https://doi.org/10.1124/mol.117.110569
- You have accessPropofol Is an Allosteric Agonist with Multiple Binding Sites on Concatemeric Ternary GABAA ReceptorsDaniel J. Shin, Allison L. Germann, Alexander D. Johnson, Stuart A. Forman, Joe Henry Steinbach and Gustav AkkMolecular Pharmacology February 2018, 93 (2) 178-189; DOI: https://doi.org/10.1124/mol.117.110403
Gilbert, Jayne
- You have access(Z)-2-(3,4-Dichlorophenyl)-3-(1H-Pyrrol-2-yl)Acrylonitrile Exhibits Selective Antitumor Activity in Breast Cancer Cell Lines via the Aryl Hydrocarbon Receptor PathwayJayne Gilbert, Geoffry N. De Iuliis, Mark Tarleton, Adam McCluskey and Jennette A. SakoffMolecular Pharmacology February 2018, 93 (2) 168-177; DOI: https://doi.org/10.1124/mol.117.109827
Glubrecht, Darryl
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Gong, Zehui
- You have accessABIN-1 Negatively Regulates μ-Opioid Receptor FunctionPeilan Zhou, Jiebing Jiang, Hui Yan, Yulei Li, Junru Zhao, Xiao Wang, Ruibin Su and Zehui GongMolecular Pharmacology February 2018, 93 (2) 36-48; DOI: https://doi.org/10.1124/mol.117.109009
Gorren, Antonius C. F.
- Open AccessIrreversible Activation and Stabilization of Soluble Guanylate Cyclase by the Protoporphyrin IX Mimetic CinaciguatAlexander Kollau, Marissa Opelt, Gerald Wölkart, Antonius C. F. Gorren, Michael Russwurm, Doris Koesling, Bernd Mayer and Astrid SchrammelMolecular Pharmacology February 2018, 93 (2) 73-78; DOI: https://doi.org/10.1124/mol.117.109918
Guo, Fusheng
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
H
Hamann, Ingrit
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Hohmann, Andrea G.
- You have accessSlowly Signaling G Protein–Biased CB2 Cannabinoid Receptor Agonist LY2828360 Suppresses Neuropathic Pain with Sustained Efficacy and Attenuates Morphine Tolerance and DependenceXiaoyan Lin, Amey S. Dhopeshwarkar, Megan Huibregtse, Ken Mackie and Andrea G. HohmannMolecular Pharmacology February 2018, 93 (2) 49-62; DOI: https://doi.org/10.1124/mol.117.109355
Huibregtse, Megan
- You have accessSlowly Signaling G Protein–Biased CB2 Cannabinoid Receptor Agonist LY2828360 Suppresses Neuropathic Pain with Sustained Efficacy and Attenuates Morphine Tolerance and DependenceXiaoyan Lin, Amey S. Dhopeshwarkar, Megan Huibregtse, Ken Mackie and Andrea G. HohmannMolecular Pharmacology February 2018, 93 (2) 49-62; DOI: https://doi.org/10.1124/mol.117.109355
J
Jiang, Jiebing
- You have accessABIN-1 Negatively Regulates μ-Opioid Receptor FunctionPeilan Zhou, Jiebing Jiang, Hui Yan, Yulei Li, Junru Zhao, Xiao Wang, Ruibin Su and Zehui GongMolecular Pharmacology February 2018, 93 (2) 36-48; DOI: https://doi.org/10.1124/mol.117.109009
Jin, Lihua
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
Jin, Shikai
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
Johnson, Alexander D.
- You have accessPropofol Is an Allosteric Agonist with Multiple Binding Sites on Concatemeric Ternary GABAA ReceptorsDaniel J. Shin, Allison L. Germann, Alexander D. Johnson, Stuart A. Forman, Joe Henry Steinbach and Gustav AkkMolecular Pharmacology February 2018, 93 (2) 178-189; DOI: https://doi.org/10.1124/mol.117.110403
K
Kaiser, Thomas M.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
Kell, Steven A.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
Koesling, Doris
- Open AccessIrreversible Activation and Stabilization of Soluble Guanylate Cyclase by the Protoporphyrin IX Mimetic CinaciguatAlexander Kollau, Marissa Opelt, Gerald Wölkart, Antonius C. F. Gorren, Michael Russwurm, Doris Koesling, Bernd Mayer and Astrid SchrammelMolecular Pharmacology February 2018, 93 (2) 73-78; DOI: https://doi.org/10.1124/mol.117.109918
Kohl, Christopher
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
Kollau, Alexander
- Open AccessIrreversible Activation and Stabilization of Soluble Guanylate Cyclase by the Protoporphyrin IX Mimetic CinaciguatAlexander Kollau, Marissa Opelt, Gerald Wölkart, Antonius C. F. Gorren, Michael Russwurm, Doris Koesling, Bernd Mayer and Astrid SchrammelMolecular Pharmacology February 2018, 93 (2) 73-78; DOI: https://doi.org/10.1124/mol.117.109918
Krys, Daniel
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Kusumoto, Hirofumi
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
L
Lam, Morrie
- You have accessDrugs and Scaffold That Inhibit Cytochrome P450 27A1 In Vitro and In VivoMorrie Lam, Natalia Mast and Irina A. PikulevaMolecular Pharmacology February 2018, 93 (2) 101-108; DOI: https://doi.org/10.1124/mol.117.110742
Lescop, Cyrille
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
Li, Yong
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
Li, Yulei
- You have accessABIN-1 Negatively Regulates μ-Opioid Receptor FunctionPeilan Zhou, Jiebing Jiang, Hui Yan, Yulei Li, Junru Zhao, Xiao Wang, Ruibin Su and Zehui GongMolecular Pharmacology February 2018, 93 (2) 36-48; DOI: https://doi.org/10.1124/mol.117.109009
Lin, Shengchen
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
Lin, Xiaoyan
- You have accessSlowly Signaling G Protein–Biased CB2 Cannabinoid Receptor Agonist LY2828360 Suppresses Neuropathic Pain with Sustained Efficacy and Attenuates Morphine Tolerance and DependenceXiaoyan Lin, Amey S. Dhopeshwarkar, Megan Huibregtse, Ken Mackie and Andrea G. HohmannMolecular Pharmacology February 2018, 93 (2) 49-62; DOI: https://doi.org/10.1124/mol.117.109355
Liotta, Dennis C.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
Liu, Xi
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
Livingston, Kathryn E.
- You have accessPharmacologic Evidence for a Putative Conserved Allosteric Site on Opioid ReceptorsKathryn E. Livingston, M. Alexander Stanczyk, Neil T. Burford, Andrew Alt, Meritxell Canals and John R. TraynorMolecular Pharmacology February 2018, 93 (2) 157-167; DOI: https://doi.org/10.1124/mol.117.109561
Lu, Yi
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
M
Mackie, Ken
- You have accessSlowly Signaling G Protein–Biased CB2 Cannabinoid Receptor Agonist LY2828360 Suppresses Neuropathic Pain with Sustained Efficacy and Attenuates Morphine Tolerance and DependenceXiaoyan Lin, Amey S. Dhopeshwarkar, Megan Huibregtse, Ken Mackie and Andrea G. HohmannMolecular Pharmacology February 2018, 93 (2) 49-62; DOI: https://doi.org/10.1124/mol.117.109355
Marshall, Alison
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Mast, Natalia
- You have accessDrugs and Scaffold That Inhibit Cytochrome P450 27A1 In Vitro and In VivoMorrie Lam, Natalia Mast and Irina A. PikulevaMolecular Pharmacology February 2018, 93 (2) 101-108; DOI: https://doi.org/10.1124/mol.117.110742
Mayer, Bernd
- Open AccessIrreversible Activation and Stabilization of Soluble Guanylate Cyclase by the Protoporphyrin IX Mimetic CinaciguatAlexander Kollau, Marissa Opelt, Gerald Wölkart, Antonius C. F. Gorren, Michael Russwurm, Doris Koesling, Bernd Mayer and Astrid SchrammelMolecular Pharmacology February 2018, 93 (2) 73-78; DOI: https://doi.org/10.1124/mol.117.109918
McCluskey, Adam
- You have access(Z)-2-(3,4-Dichlorophenyl)-3-(1H-Pyrrol-2-yl)Acrylonitrile Exhibits Selective Antitumor Activity in Breast Cancer Cell Lines via the Aryl Hydrocarbon Receptor PathwayJayne Gilbert, Geoffry N. De Iuliis, Mark Tarleton, Adam McCluskey and Jennette A. SakoffMolecular Pharmacology February 2018, 93 (2) 168-177; DOI: https://doi.org/10.1124/mol.117.109827
Menaldino, David S.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
Millar, Neil S.
- Open AccessDiversity of Nicotinic Acetylcholine Receptor Positive Allosteric Modulators Revealed by Mutagenesis and a Revised Structural ModelJoseph Newcombe, Anna Chatzidaki, Tom D. Sheppard, Maya Topf and Neil S. MillarMolecular Pharmacology February 2018, 93 (2) 128-140; DOI: https://doi.org/10.1124/mol.117.110551
Miller, Eric J.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
N
Nayler, Oliver
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
Newcombe, Joseph
- Open AccessDiversity of Nicotinic Acetylcholine Receptor Positive Allosteric Modulators Revealed by Mutagenesis and a Revised Structural ModelJoseph Newcombe, Anna Chatzidaki, Tom D. Sheppard, Maya Topf and Neil S. MillarMolecular Pharmacology February 2018, 93 (2) 128-140; DOI: https://doi.org/10.1124/mol.117.110551
O
Oladimeji, Peter O.
- You have accessPXR: More Than Just a Master Xenobiotic ReceptorPeter O. Oladimeji and Taosheng ChenMolecular Pharmacology February 2018, 93 (2) 119-127; DOI: https://doi.org/10.1124/mol.117.110155
Opelt, Marissa
- Open AccessIrreversible Activation and Stabilization of Soluble Guanylate Cyclase by the Protoporphyrin IX Mimetic CinaciguatAlexander Kollau, Marissa Opelt, Gerald Wölkart, Antonius C. F. Gorren, Michael Russwurm, Doris Koesling, Bernd Mayer and Astrid SchrammelMolecular Pharmacology February 2018, 93 (2) 73-78; DOI: https://doi.org/10.1124/mol.117.109918
P
Pikuleva, Irina A.
- You have accessDrugs and Scaffold That Inhibit Cytochrome P450 27A1 In Vitro and In VivoMorrie Lam, Natalia Mast and Irina A. PikulevaMolecular Pharmacology February 2018, 93 (2) 101-108; DOI: https://doi.org/10.1124/mol.117.110742
Poirey, Sylvie
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
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Rey, Markus
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
Russwurm, Michael
- Open AccessIrreversible Activation and Stabilization of Soluble Guanylate Cyclase by the Protoporphyrin IX Mimetic CinaciguatAlexander Kollau, Marissa Opelt, Gerald Wölkart, Antonius C. F. Gorren, Michael Russwurm, Doris Koesling, Bernd Mayer and Astrid SchrammelMolecular Pharmacology February 2018, 93 (2) 73-78; DOI: https://doi.org/10.1124/mol.117.109918
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Sakoff, Jennette A.
- You have access(Z)-2-(3,4-Dichlorophenyl)-3-(1H-Pyrrol-2-yl)Acrylonitrile Exhibits Selective Antitumor Activity in Breast Cancer Cell Lines via the Aryl Hydrocarbon Receptor PathwayJayne Gilbert, Geoffry N. De Iuliis, Mark Tarleton, Adam McCluskey and Jennette A. SakoffMolecular Pharmacology February 2018, 93 (2) 168-177; DOI: https://doi.org/10.1124/mol.117.109827
Schrammel, Astrid
- Open AccessIrreversible Activation and Stabilization of Soluble Guanylate Cyclase by the Protoporphyrin IX Mimetic CinaciguatAlexander Kollau, Marissa Opelt, Gerald Wölkart, Antonius C. F. Gorren, Michael Russwurm, Doris Koesling, Bernd Mayer and Astrid SchrammelMolecular Pharmacology February 2018, 93 (2) 73-78; DOI: https://doi.org/10.1124/mol.117.109918
Shaulsky, Gil
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
Sheppard, Tom D.
- Open AccessDiversity of Nicotinic Acetylcholine Receptor Positive Allosteric Modulators Revealed by Mutagenesis and a Revised Structural ModelJoseph Newcombe, Anna Chatzidaki, Tom D. Sheppard, Maya Topf and Neil S. MillarMolecular Pharmacology February 2018, 93 (2) 128-140; DOI: https://doi.org/10.1124/mol.117.110551
Shin, Daniel J.
- You have accessGABA Type A Receptor Activation in the Allosteric Coagonist Model Framework: Relationship between EC50 and Basal ActivityGustav Akk, Daniel J. Shin, Allison L. Germann and Joe Henry SteinbachMolecular Pharmacology February 2018, 93 (2) 90-100; DOI: https://doi.org/10.1124/mol.117.110569
- You have accessPropofol Is an Allosteric Agonist with Multiple Binding Sites on Concatemeric Ternary GABAA ReceptorsDaniel J. Shin, Allison L. Germann, Alexander D. Johnson, Stuart A. Forman, Joe Henry Steinbach and Gustav AkkMolecular Pharmacology February 2018, 93 (2) 178-189; DOI: https://doi.org/10.1124/mol.117.110403
Soueidan, Olivier-Mohamad
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Stanczyk, M. Alexander
- You have accessPharmacologic Evidence for a Putative Conserved Allosteric Site on Opioid ReceptorsKathryn E. Livingston, M. Alexander Stanczyk, Neil T. Burford, Andrew Alt, Meritxell Canals and John R. TraynorMolecular Pharmacology February 2018, 93 (2) 157-167; DOI: https://doi.org/10.1124/mol.117.109561
Steinbach, Joe Henry
- You have accessGABA Type A Receptor Activation in the Allosteric Coagonist Model Framework: Relationship between EC50 and Basal ActivityGustav Akk, Daniel J. Shin, Allison L. Germann and Joe Henry SteinbachMolecular Pharmacology February 2018, 93 (2) 90-100; DOI: https://doi.org/10.1124/mol.117.110569
- You have accessPropofol Is an Allosteric Agonist with Multiple Binding Sites on Concatemeric Ternary GABAA ReceptorsDaniel J. Shin, Allison L. Germann, Alexander D. Johnson, Stuart A. Forman, Joe Henry Steinbach and Gustav AkkMolecular Pharmacology February 2018, 93 (2) 178-189; DOI: https://doi.org/10.1124/mol.117.110403
Steiner, Beat
- Open AccessS1P1 Modulator-Induced Gαi Signaling and β-Arrestin Recruitment Are Both Necessary to Induce Rapid and Efficient Reduction of Blood Lymphocyte Count In VivoMagdalena Birker-Robaczewska, Martin Bolli, Markus Rey, Ruben de Kanter, Christopher Kohl, Cyrille Lescop, Maxime Boucher, Sylvie Poirey, Beat Steiner and Oliver NaylerMolecular Pharmacology February 2018, 93 (2) 109-118; DOI: https://doi.org/10.1124/mol.117.109140
Strong, Katie L.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
Su, Ruibin
- You have accessABIN-1 Negatively Regulates μ-Opioid Receptor FunctionPeilan Zhou, Jiebing Jiang, Hui Yan, Yulei Li, Junru Zhao, Xiao Wang, Ruibin Su and Zehui GongMolecular Pharmacology February 2018, 93 (2) 36-48; DOI: https://doi.org/10.1124/mol.117.109009
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Tarleton, Mark
- You have access(Z)-2-(3,4-Dichlorophenyl)-3-(1H-Pyrrol-2-yl)Acrylonitrile Exhibits Selective Antitumor Activity in Breast Cancer Cell Lines via the Aryl Hydrocarbon Receptor PathwayJayne Gilbert, Geoffry N. De Iuliis, Mark Tarleton, Adam McCluskey and Jennette A. SakoffMolecular Pharmacology February 2018, 93 (2) 168-177; DOI: https://doi.org/10.1124/mol.117.109827
Topf, Maya
- Open AccessDiversity of Nicotinic Acetylcholine Receptor Positive Allosteric Modulators Revealed by Mutagenesis and a Revised Structural ModelJoseph Newcombe, Anna Chatzidaki, Tom D. Sheppard, Maya Topf and Neil S. MillarMolecular Pharmacology February 2018, 93 (2) 128-140; DOI: https://doi.org/10.1124/mol.117.110551
Traynelis, Stephen F.
- You have accessThe Bioactive Protein-Ligand Conformation of GluN2C-Selective Positive Allosteric Modulators Bound to the NMDA ReceptorThomas M. Kaiser, Steven A. Kell, Hirofumi Kusumoto, Gil Shaulsky, Subhrajit Bhattacharya, Matthew P. Epplin, Katie L. Strong, Eric J. Miller, Bryan D. Cox, David S. Menaldino, Dennis C. Liotta, Stephen F. Traynelis and Pieter B. BurgerMolecular Pharmacology February 2018, 93 (2) 141-156; DOI: https://doi.org/10.1124/mol.117.110940
Trayner, Brendan
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Traynor, John R.
- You have accessPharmacologic Evidence for a Putative Conserved Allosteric Site on Opioid ReceptorsKathryn E. Livingston, M. Alexander Stanczyk, Neil T. Burford, Andrew Alt, Meritxell Canals and John R. TraynorMolecular Pharmacology February 2018, 93 (2) 157-167; DOI: https://doi.org/10.1124/mol.117.109561
W
Wagner, Michael
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Wang, Xiao
- You have accessABIN-1 Negatively Regulates μ-Opioid Receptor FunctionPeilan Zhou, Jiebing Jiang, Hui Yan, Yulei Li, Junru Zhao, Xiao Wang, Ruibin Su and Zehui GongMolecular Pharmacology February 2018, 93 (2) 36-48; DOI: https://doi.org/10.1124/mol.117.109009
Wei, Yijuan
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
West, Frederick
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Wölkart, Gerald
- Open AccessIrreversible Activation and Stabilization of Soluble Guanylate Cyclase by the Protoporphyrin IX Mimetic CinaciguatAlexander Kollau, Marissa Opelt, Gerald Wölkart, Antonius C. F. Gorren, Michael Russwurm, Doris Koesling, Bernd Mayer and Astrid SchrammelMolecular Pharmacology February 2018, 93 (2) 73-78; DOI: https://doi.org/10.1124/mol.117.109918
Wuest, Frank
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Wuest, Melinda
- You have accessMolecular Imaging of GLUT1 and GLUT5 in Breast Cancer: A Multitracer Positron Emission Tomography Imaging Study in MiceMelinda Wuest, Ingrit Hamann, Vincent Bouvet, Darryl Glubrecht, Alison Marshall, Brendan Trayner, Olivier-Mohamad Soueidan, Daniel Krys, Michael Wagner, Chris Cheeseman, Frederick West and Frank WuestMolecular Pharmacology February 2018, 93 (2) 79-89; DOI: https://doi.org/10.1124/mol.117.110007
Y
Yan, Hui
- You have accessABIN-1 Negatively Regulates μ-Opioid Receptor FunctionPeilan Zhou, Jiebing Jiang, Hui Yan, Yulei Li, Junru Zhao, Xiao Wang, Ruibin Su and Zehui GongMolecular Pharmacology February 2018, 93 (2) 36-48; DOI: https://doi.org/10.1124/mol.117.109009
Z
Zhao, Junru
- You have accessABIN-1 Negatively Regulates μ-Opioid Receptor FunctionPeilan Zhou, Jiebing Jiang, Hui Yan, Yulei Li, Junru Zhao, Xiao Wang, Ruibin Su and Zehui GongMolecular Pharmacology February 2018, 93 (2) 36-48; DOI: https://doi.org/10.1124/mol.117.109009
Zheng, Weili
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
Zhou, Peilan
- You have accessABIN-1 Negatively Regulates μ-Opioid Receptor FunctionPeilan Zhou, Jiebing Jiang, Hui Yan, Yulei Li, Junru Zhao, Xiao Wang, Ruibin Su and Zehui GongMolecular Pharmacology February 2018, 93 (2) 36-48; DOI: https://doi.org/10.1124/mol.117.109009
Zhu, Yanlin
- You have accessIdentification of an Oleanane-Type Triterpene Hedragonic Acid as a Novel Farnesoid X Receptor Ligand with Liver Protective Effects and Anti-inflammatory ActivityYi Lu, Weili Zheng, Shengchen Lin, Fusheng Guo, Yanlin Zhu, Yijuan Wei, Xi Liu, Shikai Jin, Lihua Jin and Yong LiMolecular Pharmacology February 2018, 93 (2) 63-72; DOI: https://doi.org/10.1124/mol.117.109900
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