Index by author
April 01, 2018; Volume 93,Issue 4
A
Abrie, J. Albert
- Open AccessInvestigation into the Mechanism of Homo- and Heterodimerization of Angiotensin-Converting EnzymeJ. Albert Abrie, Wessel J. A. Moolman, Gyles E. Cozier, Sylva L. Schwager, K. Ravi Acharya and Edward D. SturrockMolecular Pharmacology April 2018, 93 (4) 344-354; DOI: https://doi.org/10.1124/mol.117.110866
Acharya, K. Ravi
- Open AccessInvestigation into the Mechanism of Homo- and Heterodimerization of Angiotensin-Converting EnzymeJ. Albert Abrie, Wessel J. A. Moolman, Gyles E. Cozier, Sylva L. Schwager, K. Ravi Acharya and Edward D. SturrockMolecular Pharmacology April 2018, 93 (4) 344-354; DOI: https://doi.org/10.1124/mol.117.110866
Agarwal, Shailesh R.
- You have accesscAMP Signaling Compartmentation: Adenylyl Cyclases as Anchors of Dynamic Signaling ComplexesTimothy B. Johnstone, Shailesh R. Agarwal, Robert D. Harvey and Rennolds S. OstromMolecular Pharmacology April 2018, 93 (4) 270-276; DOI: https://doi.org/10.1124/mol.117.110825
Albert, Christoph M.
- You have accessAssay Conditions Influence Affinities of Rat Organic Cation Transporter 1: Analysis of Mutagenesis in the Modeled Outward-Facing Cleft by Measuring Effects of Substrates and Inhibitors on Initial UptakeValentin Gorboulev, Saba Rehman, Christoph M. Albert, Ursula Roth, Marleen J. Meyer, Mladen V. Tzvetkov, Thomas D. Mueller and Hermann KoepsellMolecular Pharmacology April 2018, 93 (4) 402-415; DOI: https://doi.org/10.1124/mol.117.110767
Åqvist, Johan
- Open AccessElucidation of the Binding Mode of the Carboxyterminal Region of Peptide YY to the Human Y2 ReceptorBo Xu, Silvana Vasile, Søren Østergaard, Johan F. Paulsson, Jasna Pruner, Johan Åqvist, Birgitte S. Wulff, Hugo Gutiérrez-de-Terán and Dan LarhammarMolecular Pharmacology April 2018, 93 (4) 323-334; DOI: https://doi.org/10.1124/mol.117.110627
B
Bao, Mei-Hua
- You have accessLong Noncoding RNA LINC00657 Acting as a miR-590-3p Sponge to Facilitate Low Concentration Oxidized Low-Density Lipoprotein–Induced AngiogenesisMei-Hua Bao, Guang-Yi Li, Xiao-Shan Huang, Liang Tang, Li-Ping Dong and Jian-Ming LiMolecular Pharmacology April 2018, 93 (4) 368-375; DOI: https://doi.org/10.1124/mol.117.110650
Baumeister, Paul
- You have accessMolecular Mechanisms of Biased and Probe-Dependent Signaling at CXC-Motif Chemokine Receptor CXCR3 Induced by Negative Allosteric ModulatorsRegine Brox, Lampros Milanos, Noureldin Saleh, Paul Baumeister, Armin Buschauer, Dagmar Hofmann, Markus R. Heinrich, Timothy Clark and Nuska TschammerMolecular Pharmacology April 2018, 93 (4) 309-322; DOI: https://doi.org/10.1124/mol.117.110296
Beck-Sickinger, Annette G.
- You have accessG Protein Preassembly Rescues Efficacy of W6.48 Toggle Mutations in Neuropeptide Y2 ReceptorAnette Kaiser, Caroline Hempel, Lizzy Wanka, Mario Schubert, Heidi E. Hamm and Annette G. Beck-SickingerMolecular Pharmacology April 2018, 93 (4) 387-401; DOI: https://doi.org/10.1124/mol.117.110544
Berg, Kelly A.
- You have accessAllosterism within δ Opioid–κ Opioid Receptor Heteromers in Peripheral Sensory Neurons: Regulation of κ Opioid Agonist EfficacyBlaine A. Jacobs, Miryam M. Pando, Elaine Jennings, Teresa A. Chavera, William P. Clarke and Kelly A. BergMolecular Pharmacology April 2018, 93 (4) 376-386; DOI: https://doi.org/10.1124/mol.117.109975
Bhattacharya, Supriyo
- You have accessIdentifying Functional Hotspot Residues for Biased Ligand Design in G-Protein-Coupled ReceptorsAnita K. Nivedha, Christofer S. Tautermann, Supriyo Bhattacharya, Sangbae Lee, Paola Casarosa, Ines Kollak, Tobias Kiechle and Nagarajan VaidehiMolecular Pharmacology April 2018, 93 (4) 288-296; DOI: https://doi.org/10.1124/mol.117.110395
Booe, Jason M.
- You have accessProbing the Mechanism of Receptor Activity–Modifying Protein Modulation of GPCR Ligand Selectivity through Rational Design of Potent Adrenomedullin and Calcitonin Gene-Related Peptide AntagonistsJason M. Booe, Margaret L. Warner, Amanda M. Roehrkasse, Debbie L. Hay and Augen A. PioszakMolecular Pharmacology April 2018, 93 (4) 355-367; DOI: https://doi.org/10.1124/mol.117.110916
Brox, Regine
- You have accessMolecular Mechanisms of Biased and Probe-Dependent Signaling at CXC-Motif Chemokine Receptor CXCR3 Induced by Negative Allosteric ModulatorsRegine Brox, Lampros Milanos, Noureldin Saleh, Paul Baumeister, Armin Buschauer, Dagmar Hofmann, Markus R. Heinrich, Timothy Clark and Nuska TschammerMolecular Pharmacology April 2018, 93 (4) 309-322; DOI: https://doi.org/10.1124/mol.117.110296
Buschauer, Armin
- You have accessMolecular Mechanisms of Biased and Probe-Dependent Signaling at CXC-Motif Chemokine Receptor CXCR3 Induced by Negative Allosteric ModulatorsRegine Brox, Lampros Milanos, Noureldin Saleh, Paul Baumeister, Armin Buschauer, Dagmar Hofmann, Markus R. Heinrich, Timothy Clark and Nuska TschammerMolecular Pharmacology April 2018, 93 (4) 309-322; DOI: https://doi.org/10.1124/mol.117.110296
C
Casarosa, Paola
- You have accessIdentifying Functional Hotspot Residues for Biased Ligand Design in G-Protein-Coupled ReceptorsAnita K. Nivedha, Christofer S. Tautermann, Supriyo Bhattacharya, Sangbae Lee, Paola Casarosa, Ines Kollak, Tobias Kiechle and Nagarajan VaidehiMolecular Pharmacology April 2018, 93 (4) 288-296; DOI: https://doi.org/10.1124/mol.117.110395
Charlton, Steven J.
- You have accessBiased Agonism in Drug Discovery—Is It Too Soon to Choose a Path?Martin C. Michel and Steven J. CharltonMolecular Pharmacology April 2018, 93 (4) 259-265; DOI: https://doi.org/10.1124/mol.117.110890
Chavera, Teresa A.
- You have accessAllosterism within δ Opioid–κ Opioid Receptor Heteromers in Peripheral Sensory Neurons: Regulation of κ Opioid Agonist EfficacyBlaine A. Jacobs, Miryam M. Pando, Elaine Jennings, Teresa A. Chavera, William P. Clarke and Kelly A. BergMolecular Pharmacology April 2018, 93 (4) 376-386; DOI: https://doi.org/10.1124/mol.117.109975
Clark, Timothy
- You have accessMolecular Mechanisms of Biased and Probe-Dependent Signaling at CXC-Motif Chemokine Receptor CXCR3 Induced by Negative Allosteric ModulatorsRegine Brox, Lampros Milanos, Noureldin Saleh, Paul Baumeister, Armin Buschauer, Dagmar Hofmann, Markus R. Heinrich, Timothy Clark and Nuska TschammerMolecular Pharmacology April 2018, 93 (4) 309-322; DOI: https://doi.org/10.1124/mol.117.110296
Clarke, William P.
- You have accessAllosterism within δ Opioid–κ Opioid Receptor Heteromers in Peripheral Sensory Neurons: Regulation of κ Opioid Agonist EfficacyBlaine A. Jacobs, Miryam M. Pando, Elaine Jennings, Teresa A. Chavera, William P. Clarke and Kelly A. BergMolecular Pharmacology April 2018, 93 (4) 376-386; DOI: https://doi.org/10.1124/mol.117.109975
Cozier, Gyles E.
- Open AccessInvestigation into the Mechanism of Homo- and Heterodimerization of Angiotensin-Converting EnzymeJ. Albert Abrie, Wessel J. A. Moolman, Gyles E. Cozier, Sylva L. Schwager, K. Ravi Acharya and Edward D. SturrockMolecular Pharmacology April 2018, 93 (4) 344-354; DOI: https://doi.org/10.1124/mol.117.110866
D
Dong, Li-Ping
- You have accessLong Noncoding RNA LINC00657 Acting as a miR-590-3p Sponge to Facilitate Low Concentration Oxidized Low-Density Lipoprotein–Induced AngiogenesisMei-Hua Bao, Guang-Yi Li, Xiao-Shan Huang, Liang Tang, Li-Ping Dong and Jian-Ming LiMolecular Pharmacology April 2018, 93 (4) 368-375; DOI: https://doi.org/10.1124/mol.117.110650
E
Eroglu, Emrah
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
F
Fassett, John T.
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
Fathima, Samreen
- Open AccessPharmacogenomics of Chemically Distinct Classes of Keap1-Nrf2 Activators Identify Common and Unique Gene, Protein, and Pathway Responses In VivoRyan S. Wible, Quynh T. Tran, Samreen Fathima, Carrie H. Sutter, Thomas W. Kensler and Thomas R. SutterMolecular Pharmacology April 2018, 93 (4) 297-308; DOI: https://doi.org/10.1124/mol.117.110262
G
Gorboulev, Valentin
- You have accessAssay Conditions Influence Affinities of Rat Organic Cation Transporter 1: Analysis of Mutagenesis in the Modeled Outward-Facing Cleft by Measuring Effects of Substrates and Inhibitors on Initial UptakeValentin Gorboulev, Saba Rehman, Christoph M. Albert, Ursula Roth, Marleen J. Meyer, Mladen V. Tzvetkov, Thomas D. Mueller and Hermann KoepsellMolecular Pharmacology April 2018, 93 (4) 402-415; DOI: https://doi.org/10.1124/mol.117.110767
Gorren, Antonius C. F.
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
Graier, Wolfgang F.
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
Gutiérrez-de-Terán, Hugo
- Open AccessElucidation of the Binding Mode of the Carboxyterminal Region of Peptide YY to the Human Y2 ReceptorBo Xu, Silvana Vasile, Søren Østergaard, Johan F. Paulsson, Jasna Pruner, Johan Åqvist, Birgitte S. Wulff, Hugo Gutiérrez-de-Terán and Dan LarhammarMolecular Pharmacology April 2018, 93 (4) 323-334; DOI: https://doi.org/10.1124/mol.117.110627
H
Hamm, Heidi E.
- You have accessG Protein Preassembly Rescues Efficacy of W6.48 Toggle Mutations in Neuropeptide Y2 ReceptorAnette Kaiser, Caroline Hempel, Lizzy Wanka, Mario Schubert, Heidi E. Hamm and Annette G. Beck-SickingerMolecular Pharmacology April 2018, 93 (4) 387-401; DOI: https://doi.org/10.1124/mol.117.110544
Harvey, Robert D.
- You have accesscAMP Signaling Compartmentation: Adenylyl Cyclases as Anchors of Dynamic Signaling ComplexesTimothy B. Johnstone, Shailesh R. Agarwal, Robert D. Harvey and Rennolds S. OstromMolecular Pharmacology April 2018, 93 (4) 270-276; DOI: https://doi.org/10.1124/mol.117.110825
Hay, Debbie L.
- You have accessProbing the Mechanism of Receptor Activity–Modifying Protein Modulation of GPCR Ligand Selectivity through Rational Design of Potent Adrenomedullin and Calcitonin Gene-Related Peptide AntagonistsJason M. Booe, Margaret L. Warner, Amanda M. Roehrkasse, Debbie L. Hay and Augen A. PioszakMolecular Pharmacology April 2018, 93 (4) 355-367; DOI: https://doi.org/10.1124/mol.117.110916
Head, Brian P.
- You have accessCaveolins as Regulators of Stress AdaptationJan M. Schilling, Brian P. Head and Hemal H. PatelMolecular Pharmacology April 2018, 93 (4) 277-285; DOI: https://doi.org/10.1124/mol.117.111237
Heinrich, Markus R.
- You have accessMolecular Mechanisms of Biased and Probe-Dependent Signaling at CXC-Motif Chemokine Receptor CXCR3 Induced by Negative Allosteric ModulatorsRegine Brox, Lampros Milanos, Noureldin Saleh, Paul Baumeister, Armin Buschauer, Dagmar Hofmann, Markus R. Heinrich, Timothy Clark and Nuska TschammerMolecular Pharmacology April 2018, 93 (4) 309-322; DOI: https://doi.org/10.1124/mol.117.110296
Hempel, Caroline
- You have accessG Protein Preassembly Rescues Efficacy of W6.48 Toggle Mutations in Neuropeptide Y2 ReceptorAnette Kaiser, Caroline Hempel, Lizzy Wanka, Mario Schubert, Heidi E. Hamm and Annette G. Beck-SickingerMolecular Pharmacology April 2018, 93 (4) 387-401; DOI: https://doi.org/10.1124/mol.117.110544
Hofmann, Dagmar
- You have accessMolecular Mechanisms of Biased and Probe-Dependent Signaling at CXC-Motif Chemokine Receptor CXCR3 Induced by Negative Allosteric ModulatorsRegine Brox, Lampros Milanos, Noureldin Saleh, Paul Baumeister, Armin Buschauer, Dagmar Hofmann, Markus R. Heinrich, Timothy Clark and Nuska TschammerMolecular Pharmacology April 2018, 93 (4) 309-322; DOI: https://doi.org/10.1124/mol.117.110296
Huang, Xiao-Shan
- You have accessLong Noncoding RNA LINC00657 Acting as a miR-590-3p Sponge to Facilitate Low Concentration Oxidized Low-Density Lipoprotein–Induced AngiogenesisMei-Hua Bao, Guang-Yi Li, Xiao-Shan Huang, Liang Tang, Li-Ping Dong and Jian-Ming LiMolecular Pharmacology April 2018, 93 (4) 368-375; DOI: https://doi.org/10.1124/mol.117.110650
I
Insel, Paul A.
- You have accessG Protein-Coupled Receptors as Targets for Approved Drugs: How Many Targets and How Many Drugs?Krishna Sriram and Paul A. InselMolecular Pharmacology April 2018, 93 (4) 251-258; DOI: https://doi.org/10.1124/mol.117.111062
J
Jacobs, Blaine A.
- You have accessAllosterism within δ Opioid–κ Opioid Receptor Heteromers in Peripheral Sensory Neurons: Regulation of κ Opioid Agonist EfficacyBlaine A. Jacobs, Miryam M. Pando, Elaine Jennings, Teresa A. Chavera, William P. Clarke and Kelly A. BergMolecular Pharmacology April 2018, 93 (4) 376-386; DOI: https://doi.org/10.1124/mol.117.109975
Jennings, Elaine
- You have accessAllosterism within δ Opioid–κ Opioid Receptor Heteromers in Peripheral Sensory Neurons: Regulation of κ Opioid Agonist EfficacyBlaine A. Jacobs, Miryam M. Pando, Elaine Jennings, Teresa A. Chavera, William P. Clarke and Kelly A. BergMolecular Pharmacology April 2018, 93 (4) 376-386; DOI: https://doi.org/10.1124/mol.117.109975
Johnstone, Timothy B.
- You have accesscAMP Signaling Compartmentation: Adenylyl Cyclases as Anchors of Dynamic Signaling ComplexesTimothy B. Johnstone, Shailesh R. Agarwal, Robert D. Harvey and Rennolds S. OstromMolecular Pharmacology April 2018, 93 (4) 270-276; DOI: https://doi.org/10.1124/mol.117.110825
K
Kaiser, Anette
- You have accessG Protein Preassembly Rescues Efficacy of W6.48 Toggle Mutations in Neuropeptide Y2 ReceptorAnette Kaiser, Caroline Hempel, Lizzy Wanka, Mario Schubert, Heidi E. Hamm and Annette G. Beck-SickingerMolecular Pharmacology April 2018, 93 (4) 387-401; DOI: https://doi.org/10.1124/mol.117.110544
Kenakin, Terry
- You have accessIs the Quest for Signaling Bias Worth the Effort?Terry KenakinMolecular Pharmacology April 2018, 93 (4) 266-269; DOI: https://doi.org/10.1124/mol.117.111187
Kensler, Thomas W.
- Open AccessPharmacogenomics of Chemically Distinct Classes of Keap1-Nrf2 Activators Identify Common and Unique Gene, Protein, and Pathway Responses In VivoRyan S. Wible, Quynh T. Tran, Samreen Fathima, Carrie H. Sutter, Thomas W. Kensler and Thomas R. SutterMolecular Pharmacology April 2018, 93 (4) 297-308; DOI: https://doi.org/10.1124/mol.117.110262
Kiechle, Tobias
- You have accessIdentifying Functional Hotspot Residues for Biased Ligand Design in G-Protein-Coupled ReceptorsAnita K. Nivedha, Christofer S. Tautermann, Supriyo Bhattacharya, Sangbae Lee, Paola Casarosa, Ines Kollak, Tobias Kiechle and Nagarajan VaidehiMolecular Pharmacology April 2018, 93 (4) 288-296; DOI: https://doi.org/10.1124/mol.117.110395
Koepsell, Hermann
- You have accessAssay Conditions Influence Affinities of Rat Organic Cation Transporter 1: Analysis of Mutagenesis in the Modeled Outward-Facing Cleft by Measuring Effects of Substrates and Inhibitors on Initial UptakeValentin Gorboulev, Saba Rehman, Christoph M. Albert, Ursula Roth, Marleen J. Meyer, Mladen V. Tzvetkov, Thomas D. Mueller and Hermann KoepsellMolecular Pharmacology April 2018, 93 (4) 402-415; DOI: https://doi.org/10.1124/mol.117.110767
Kollak, Ines
- You have accessIdentifying Functional Hotspot Residues for Biased Ligand Design in G-Protein-Coupled ReceptorsAnita K. Nivedha, Christofer S. Tautermann, Supriyo Bhattacharya, Sangbae Lee, Paola Casarosa, Ines Kollak, Tobias Kiechle and Nagarajan VaidehiMolecular Pharmacology April 2018, 93 (4) 288-296; DOI: https://doi.org/10.1124/mol.117.110395
Kollau, Alexander
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
L
Larhammar, Dan
- Open AccessElucidation of the Binding Mode of the Carboxyterminal Region of Peptide YY to the Human Y2 ReceptorBo Xu, Silvana Vasile, Søren Østergaard, Johan F. Paulsson, Jasna Pruner, Johan Åqvist, Birgitte S. Wulff, Hugo Gutiérrez-de-Terán and Dan LarhammarMolecular Pharmacology April 2018, 93 (4) 323-334; DOI: https://doi.org/10.1124/mol.117.110627
Lee, Sangbae
- You have accessIdentifying Functional Hotspot Residues for Biased Ligand Design in G-Protein-Coupled ReceptorsAnita K. Nivedha, Christofer S. Tautermann, Supriyo Bhattacharya, Sangbae Lee, Paola Casarosa, Ines Kollak, Tobias Kiechle and Nagarajan VaidehiMolecular Pharmacology April 2018, 93 (4) 288-296; DOI: https://doi.org/10.1124/mol.117.110395
Li, Guang-Yi
- You have accessLong Noncoding RNA LINC00657 Acting as a miR-590-3p Sponge to Facilitate Low Concentration Oxidized Low-Density Lipoprotein–Induced AngiogenesisMei-Hua Bao, Guang-Yi Li, Xiao-Shan Huang, Liang Tang, Li-Ping Dong and Jian-Ming LiMolecular Pharmacology April 2018, 93 (4) 368-375; DOI: https://doi.org/10.1124/mol.117.110650
Li, Jian-Ming
- You have accessLong Noncoding RNA LINC00657 Acting as a miR-590-3p Sponge to Facilitate Low Concentration Oxidized Low-Density Lipoprotein–Induced AngiogenesisMei-Hua Bao, Guang-Yi Li, Xiao-Shan Huang, Liang Tang, Li-Ping Dong and Jian-Ming LiMolecular Pharmacology April 2018, 93 (4) 368-375; DOI: https://doi.org/10.1124/mol.117.110650
M
Malli, Roland
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
Mayer, Bernd
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
Meyer, Marleen J.
- You have accessAssay Conditions Influence Affinities of Rat Organic Cation Transporter 1: Analysis of Mutagenesis in the Modeled Outward-Facing Cleft by Measuring Effects of Substrates and Inhibitors on Initial UptakeValentin Gorboulev, Saba Rehman, Christoph M. Albert, Ursula Roth, Marleen J. Meyer, Mladen V. Tzvetkov, Thomas D. Mueller and Hermann KoepsellMolecular Pharmacology April 2018, 93 (4) 402-415; DOI: https://doi.org/10.1124/mol.117.110767
Michel, Martin C.
- You have accessBiased Agonism in Drug Discovery—Is It Too Soon to Choose a Path?Martin C. Michel and Steven J. CharltonMolecular Pharmacology April 2018, 93 (4) 259-265; DOI: https://doi.org/10.1124/mol.117.110890
Milanos, Lampros
- You have accessMolecular Mechanisms of Biased and Probe-Dependent Signaling at CXC-Motif Chemokine Receptor CXCR3 Induced by Negative Allosteric ModulatorsRegine Brox, Lampros Milanos, Noureldin Saleh, Paul Baumeister, Armin Buschauer, Dagmar Hofmann, Markus R. Heinrich, Timothy Clark and Nuska TschammerMolecular Pharmacology April 2018, 93 (4) 309-322; DOI: https://doi.org/10.1124/mol.117.110296
Moolman, Wessel J. A.
- Open AccessInvestigation into the Mechanism of Homo- and Heterodimerization of Angiotensin-Converting EnzymeJ. Albert Abrie, Wessel J. A. Moolman, Gyles E. Cozier, Sylva L. Schwager, K. Ravi Acharya and Edward D. SturrockMolecular Pharmacology April 2018, 93 (4) 344-354; DOI: https://doi.org/10.1124/mol.117.110866
Mueller, Thomas D.
- You have accessAssay Conditions Influence Affinities of Rat Organic Cation Transporter 1: Analysis of Mutagenesis in the Modeled Outward-Facing Cleft by Measuring Effects of Substrates and Inhibitors on Initial UptakeValentin Gorboulev, Saba Rehman, Christoph M. Albert, Ursula Roth, Marleen J. Meyer, Mladen V. Tzvetkov, Thomas D. Mueller and Hermann KoepsellMolecular Pharmacology April 2018, 93 (4) 402-415; DOI: https://doi.org/10.1124/mol.117.110767
N
Nivedha, Anita K.
- You have accessIdentifying Functional Hotspot Residues for Biased Ligand Design in G-Protein-Coupled ReceptorsAnita K. Nivedha, Christofer S. Tautermann, Supriyo Bhattacharya, Sangbae Lee, Paola Casarosa, Ines Kollak, Tobias Kiechle and Nagarajan VaidehiMolecular Pharmacology April 2018, 93 (4) 288-296; DOI: https://doi.org/10.1124/mol.117.110395
O
Opelt, Marissa
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
Østergaard, Søren
- Open AccessElucidation of the Binding Mode of the Carboxyterminal Region of Peptide YY to the Human Y2 ReceptorBo Xu, Silvana Vasile, Søren Østergaard, Johan F. Paulsson, Jasna Pruner, Johan Åqvist, Birgitte S. Wulff, Hugo Gutiérrez-de-Terán and Dan LarhammarMolecular Pharmacology April 2018, 93 (4) 323-334; DOI: https://doi.org/10.1124/mol.117.110627
Ostrom, Rennolds S.
- You have accesscAMP Signaling Compartmentation: Adenylyl Cyclases as Anchors of Dynamic Signaling ComplexesTimothy B. Johnstone, Shailesh R. Agarwal, Robert D. Harvey and Rennolds S. OstromMolecular Pharmacology April 2018, 93 (4) 270-276; DOI: https://doi.org/10.1124/mol.117.110825
P
Pando, Miryam M.
- You have accessAllosterism within δ Opioid–κ Opioid Receptor Heteromers in Peripheral Sensory Neurons: Regulation of κ Opioid Agonist EfficacyBlaine A. Jacobs, Miryam M. Pando, Elaine Jennings, Teresa A. Chavera, William P. Clarke and Kelly A. BergMolecular Pharmacology April 2018, 93 (4) 376-386; DOI: https://doi.org/10.1124/mol.117.109975
Patel, Hemal H.
- You have accessCaveolins as Regulators of Stress AdaptationJan M. Schilling, Brian P. Head and Hemal H. PatelMolecular Pharmacology April 2018, 93 (4) 277-285; DOI: https://doi.org/10.1124/mol.117.111237
Paulsson, Johan F.
- Open AccessElucidation of the Binding Mode of the Carboxyterminal Region of Peptide YY to the Human Y2 ReceptorBo Xu, Silvana Vasile, Søren Østergaard, Johan F. Paulsson, Jasna Pruner, Johan Åqvist, Birgitte S. Wulff, Hugo Gutiérrez-de-Terán and Dan LarhammarMolecular Pharmacology April 2018, 93 (4) 323-334; DOI: https://doi.org/10.1124/mol.117.110627
Pioszak, Augen A.
- You have accessProbing the Mechanism of Receptor Activity–Modifying Protein Modulation of GPCR Ligand Selectivity through Rational Design of Potent Adrenomedullin and Calcitonin Gene-Related Peptide AntagonistsJason M. Booe, Margaret L. Warner, Amanda M. Roehrkasse, Debbie L. Hay and Augen A. PioszakMolecular Pharmacology April 2018, 93 (4) 355-367; DOI: https://doi.org/10.1124/mol.117.110916
Pruner, Jasna
- Open AccessElucidation of the Binding Mode of the Carboxyterminal Region of Peptide YY to the Human Y2 ReceptorBo Xu, Silvana Vasile, Søren Østergaard, Johan F. Paulsson, Jasna Pruner, Johan Åqvist, Birgitte S. Wulff, Hugo Gutiérrez-de-Terán and Dan LarhammarMolecular Pharmacology April 2018, 93 (4) 323-334; DOI: https://doi.org/10.1124/mol.117.110627
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Rehman, Saba
- You have accessAssay Conditions Influence Affinities of Rat Organic Cation Transporter 1: Analysis of Mutagenesis in the Modeled Outward-Facing Cleft by Measuring Effects of Substrates and Inhibitors on Initial UptakeValentin Gorboulev, Saba Rehman, Christoph M. Albert, Ursula Roth, Marleen J. Meyer, Mladen V. Tzvetkov, Thomas D. Mueller and Hermann KoepsellMolecular Pharmacology April 2018, 93 (4) 402-415; DOI: https://doi.org/10.1124/mol.117.110767
Roehrkasse, Amanda M.
- You have accessProbing the Mechanism of Receptor Activity–Modifying Protein Modulation of GPCR Ligand Selectivity through Rational Design of Potent Adrenomedullin and Calcitonin Gene-Related Peptide AntagonistsJason M. Booe, Margaret L. Warner, Amanda M. Roehrkasse, Debbie L. Hay and Augen A. PioszakMolecular Pharmacology April 2018, 93 (4) 355-367; DOI: https://doi.org/10.1124/mol.117.110916
Roth, Ursula
- You have accessAssay Conditions Influence Affinities of Rat Organic Cation Transporter 1: Analysis of Mutagenesis in the Modeled Outward-Facing Cleft by Measuring Effects of Substrates and Inhibitors on Initial UptakeValentin Gorboulev, Saba Rehman, Christoph M. Albert, Ursula Roth, Marleen J. Meyer, Mladen V. Tzvetkov, Thomas D. Mueller and Hermann KoepsellMolecular Pharmacology April 2018, 93 (4) 402-415; DOI: https://doi.org/10.1124/mol.117.110767
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Saleh, Noureldin
- You have accessMolecular Mechanisms of Biased and Probe-Dependent Signaling at CXC-Motif Chemokine Receptor CXCR3 Induced by Negative Allosteric ModulatorsRegine Brox, Lampros Milanos, Noureldin Saleh, Paul Baumeister, Armin Buschauer, Dagmar Hofmann, Markus R. Heinrich, Timothy Clark and Nuska TschammerMolecular Pharmacology April 2018, 93 (4) 309-322; DOI: https://doi.org/10.1124/mol.117.110296
Schilling, Jan M.
- You have accessCaveolins as Regulators of Stress AdaptationJan M. Schilling, Brian P. Head and Hemal H. PatelMolecular Pharmacology April 2018, 93 (4) 277-285; DOI: https://doi.org/10.1124/mol.117.111237
Schrammel, Astrid
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
Schubert, Mario
- You have accessG Protein Preassembly Rescues Efficacy of W6.48 Toggle Mutations in Neuropeptide Y2 ReceptorAnette Kaiser, Caroline Hempel, Lizzy Wanka, Mario Schubert, Heidi E. Hamm and Annette G. Beck-SickingerMolecular Pharmacology April 2018, 93 (4) 387-401; DOI: https://doi.org/10.1124/mol.117.110544
Schwager, Sylva L.
- Open AccessInvestigation into the Mechanism of Homo- and Heterodimerization of Angiotensin-Converting EnzymeJ. Albert Abrie, Wessel J. A. Moolman, Gyles E. Cozier, Sylva L. Schwager, K. Ravi Acharya and Edward D. SturrockMolecular Pharmacology April 2018, 93 (4) 344-354; DOI: https://doi.org/10.1124/mol.117.110866
Sriram, Krishna
- You have accessG Protein-Coupled Receptors as Targets for Approved Drugs: How Many Targets and How Many Drugs?Krishna Sriram and Paul A. InselMolecular Pharmacology April 2018, 93 (4) 251-258; DOI: https://doi.org/10.1124/mol.117.111062
Sturrock, Edward D.
- Open AccessInvestigation into the Mechanism of Homo- and Heterodimerization of Angiotensin-Converting EnzymeJ. Albert Abrie, Wessel J. A. Moolman, Gyles E. Cozier, Sylva L. Schwager, K. Ravi Acharya and Edward D. SturrockMolecular Pharmacology April 2018, 93 (4) 344-354; DOI: https://doi.org/10.1124/mol.117.110866
Sutter, Carrie H.
- Open AccessPharmacogenomics of Chemically Distinct Classes of Keap1-Nrf2 Activators Identify Common and Unique Gene, Protein, and Pathway Responses In VivoRyan S. Wible, Quynh T. Tran, Samreen Fathima, Carrie H. Sutter, Thomas W. Kensler and Thomas R. SutterMolecular Pharmacology April 2018, 93 (4) 297-308; DOI: https://doi.org/10.1124/mol.117.110262
Sutter, Thomas R.
- Open AccessPharmacogenomics of Chemically Distinct Classes of Keap1-Nrf2 Activators Identify Common and Unique Gene, Protein, and Pathway Responses In VivoRyan S. Wible, Quynh T. Tran, Samreen Fathima, Carrie H. Sutter, Thomas W. Kensler and Thomas R. SutterMolecular Pharmacology April 2018, 93 (4) 297-308; DOI: https://doi.org/10.1124/mol.117.110262
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Tang, Liang
- You have accessLong Noncoding RNA LINC00657 Acting as a miR-590-3p Sponge to Facilitate Low Concentration Oxidized Low-Density Lipoprotein–Induced AngiogenesisMei-Hua Bao, Guang-Yi Li, Xiao-Shan Huang, Liang Tang, Li-Ping Dong and Jian-Ming LiMolecular Pharmacology April 2018, 93 (4) 368-375; DOI: https://doi.org/10.1124/mol.117.110650
Tautermann, Christofer S.
- You have accessIdentifying Functional Hotspot Residues for Biased Ligand Design in G-Protein-Coupled ReceptorsAnita K. Nivedha, Christofer S. Tautermann, Supriyo Bhattacharya, Sangbae Lee, Paola Casarosa, Ines Kollak, Tobias Kiechle and Nagarajan VaidehiMolecular Pharmacology April 2018, 93 (4) 288-296; DOI: https://doi.org/10.1124/mol.117.110395
Tran, Quynh T.
- Open AccessPharmacogenomics of Chemically Distinct Classes of Keap1-Nrf2 Activators Identify Common and Unique Gene, Protein, and Pathway Responses In VivoRyan S. Wible, Quynh T. Tran, Samreen Fathima, Carrie H. Sutter, Thomas W. Kensler and Thomas R. SutterMolecular Pharmacology April 2018, 93 (4) 297-308; DOI: https://doi.org/10.1124/mol.117.110262
Tschammer, Nuska
- You have accessMolecular Mechanisms of Biased and Probe-Dependent Signaling at CXC-Motif Chemokine Receptor CXCR3 Induced by Negative Allosteric ModulatorsRegine Brox, Lampros Milanos, Noureldin Saleh, Paul Baumeister, Armin Buschauer, Dagmar Hofmann, Markus R. Heinrich, Timothy Clark and Nuska TschammerMolecular Pharmacology April 2018, 93 (4) 309-322; DOI: https://doi.org/10.1124/mol.117.110296
Tzvetkov, Mladen V.
- You have accessAssay Conditions Influence Affinities of Rat Organic Cation Transporter 1: Analysis of Mutagenesis in the Modeled Outward-Facing Cleft by Measuring Effects of Substrates and Inhibitors on Initial UptakeValentin Gorboulev, Saba Rehman, Christoph M. Albert, Ursula Roth, Marleen J. Meyer, Mladen V. Tzvetkov, Thomas D. Mueller and Hermann KoepsellMolecular Pharmacology April 2018, 93 (4) 402-415; DOI: https://doi.org/10.1124/mol.117.110767
V
Vaidehi, Nagarajan
- You have accessIdentifying Functional Hotspot Residues for Biased Ligand Design in G-Protein-Coupled ReceptorsAnita K. Nivedha, Christofer S. Tautermann, Supriyo Bhattacharya, Sangbae Lee, Paola Casarosa, Ines Kollak, Tobias Kiechle and Nagarajan VaidehiMolecular Pharmacology April 2018, 93 (4) 288-296; DOI: https://doi.org/10.1124/mol.117.110395
Vasile, Silvana
- Open AccessElucidation of the Binding Mode of the Carboxyterminal Region of Peptide YY to the Human Y2 ReceptorBo Xu, Silvana Vasile, Søren Østergaard, Johan F. Paulsson, Jasna Pruner, Johan Åqvist, Birgitte S. Wulff, Hugo Gutiérrez-de-Terán and Dan LarhammarMolecular Pharmacology April 2018, 93 (4) 323-334; DOI: https://doi.org/10.1124/mol.117.110627
Vore, Mary
- You have accessPublishing in an ASPET Journal – What’s in It for You?Mary VoreMolecular Pharmacology April 2018, 93 (4) 286-287; DOI: https://doi.org/10.1124/mol.117.112193
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Waldeck-Weiermair, Markus
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
Wanka, Lizzy
- You have accessG Protein Preassembly Rescues Efficacy of W6.48 Toggle Mutations in Neuropeptide Y2 ReceptorAnette Kaiser, Caroline Hempel, Lizzy Wanka, Mario Schubert, Heidi E. Hamm and Annette G. Beck-SickingerMolecular Pharmacology April 2018, 93 (4) 387-401; DOI: https://doi.org/10.1124/mol.117.110544
Warner, Margaret L.
- You have accessProbing the Mechanism of Receptor Activity–Modifying Protein Modulation of GPCR Ligand Selectivity through Rational Design of Potent Adrenomedullin and Calcitonin Gene-Related Peptide AntagonistsJason M. Booe, Margaret L. Warner, Amanda M. Roehrkasse, Debbie L. Hay and Augen A. PioszakMolecular Pharmacology April 2018, 93 (4) 355-367; DOI: https://doi.org/10.1124/mol.117.110916
Wible, Ryan S.
- Open AccessPharmacogenomics of Chemically Distinct Classes of Keap1-Nrf2 Activators Identify Common and Unique Gene, Protein, and Pathway Responses In VivoRyan S. Wible, Quynh T. Tran, Samreen Fathima, Carrie H. Sutter, Thomas W. Kensler and Thomas R. SutterMolecular Pharmacology April 2018, 93 (4) 297-308; DOI: https://doi.org/10.1124/mol.117.110262
Wölkart, Gerald
- Open AccessSustained Formation of Nitroglycerin-Derived Nitric Oxide by Aldehyde Dehydrogenase-2 in Vascular Smooth Muscle without Added Reductants: Implications for the Development of Nitrate ToleranceMarissa Opelt, Gerald Wölkart, Emrah Eroglu, Markus Waldeck-Weiermair, Roland Malli, Wolfgang F. Graier, Alexander Kollau, John T. Fassett, Astrid Schrammel, Bernd Mayer and Antonius C. F. GorrenMolecular Pharmacology April 2018, 93 (4) 335-343; DOI: https://doi.org/10.1124/mol.117.110783
Wulff, Birgitte S.
- Open AccessElucidation of the Binding Mode of the Carboxyterminal Region of Peptide YY to the Human Y2 ReceptorBo Xu, Silvana Vasile, Søren Østergaard, Johan F. Paulsson, Jasna Pruner, Johan Åqvist, Birgitte S. Wulff, Hugo Gutiérrez-de-Terán and Dan LarhammarMolecular Pharmacology April 2018, 93 (4) 323-334; DOI: https://doi.org/10.1124/mol.117.110627
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Xu, Bo
- Open AccessElucidation of the Binding Mode of the Carboxyterminal Region of Peptide YY to the Human Y2 ReceptorBo Xu, Silvana Vasile, Søren Østergaard, Johan F. Paulsson, Jasna Pruner, Johan Åqvist, Birgitte S. Wulff, Hugo Gutiérrez-de-Terán and Dan LarhammarMolecular Pharmacology April 2018, 93 (4) 323-334; DOI: https://doi.org/10.1124/mol.117.110627
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