Research ArticleArticle
“Selective” Class C G Protein-Coupled Receptor Modulators Are Neutral or Biased mGlu5 Allosteric Ligands
Shane D. Hellyer, Sabine Albold, Taide Wang, Amy N. Y. Chen, Lauren T. May, Katie Leach and Karen J. Gregory
Molecular Pharmacology May 2018, 93 (5) 504-514; DOI: https://doi.org/10.1124/mol.117.111518
Shane D. Hellyer
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
Sabine Albold
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
Taide Wang
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
Amy N. Y. Chen
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
Lauren T. May
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
Katie Leach
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
Karen J. Gregory
Drug Discovery Biology, Monash Institute of Pharmaceutical Sciences and Department of Pharmacology, Monash University, Parkville, Victoria, Australia
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Cooperativity Drives Modulator Selectivity for Class C GPCRs
Shane D. Hellyer, Sabine Albold, Taide Wang, Amy N. Y. Chen, Lauren T. May, Katie Leach and Karen J. Gregory
Molecular Pharmacology May 1, 2018, 93 (5) 504-514; DOI: https://doi.org/10.1124/mol.117.111518
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