Table of Contents

Articles

• You have access

  Insulin Receptor Plasma Membrane Levels Increased by the Progesterone Receptor Membrane Component 1

  Kaia K. Hampton, Katie Anderson, Hilaree Frazier, Olivier Thibault and Rolf J. Craven

  Molecular Pharmacology July 2018, 94 (1) 665-673; DOI: https://doi.org/10.1124/mol.117.110510
• You have access

  Ligand-Specific Signaling Profiles and Resensitization Mechanisms of the Neuromedin U2 Receptor

  Khaled Alhosaini, Omar Bahattab, Heider Qassam, R. A. John Challiss and Gary B. Willars

  Molecular Pharmacology July 2018, 94 (1) 674-688; DOI: https://doi.org/10.1124/mol.117.111070
• You have access

  Molecular Mechanisms for Species Differences in Organic Anion Transporter 1, OAT1: Implications for Renal Drug Toxicity

  Ling Zou, Adrian Stecula, Anshul Gupta, Bhagwat Prasad, Huan-Chieh Chien, Sook Wah Yee, Li Wang, Jashvant D. Unadkat, Simone H. Stahl, Katherine S. Fenner and Kathleen M. Giacomini

  Molecular Pharmacology July 2018, 94 (1) 689-699; DOI: https://doi.org/10.1124/mol.117.111153
• You have access

  Thyroid Hormones Are Transport Substrates and Transcriptional Regulators of Organic Anion Transporting Polypeptide 2B1

  Henriette E. Meyer zu Schwabedissen, Celio Ferreira, Anima M. Schaefer, Mouhssin Oufir, Isabell Seibert, Matthias Hamburger and Rommel G. Tirona

  Molecular Pharmacology July 2018, 94 (1) 700-712; DOI: https://doi.org/10.1124/mol.117.111161
• Open Access

  Cysteine Scanning Mutagenesis of TM4b-4c Loop of Glutamate Transporter EAAT1 Reveals Three Conformationally Sensitive Residues

  Wenlong Zhang, Xiuping Zhang and Shaogang Qu

  Molecular Pharmacology July 2018, 94 (1) 713-721; DOI: https://doi.org/10.1124/mol.117.111245
• 

  You have access

  Efficient High-Throughput Screening by Endoplasmic Reticulum Ca²⁺ Measurement to Identify Inhibitors of Ryanodine Receptor Ca²⁺-Release Channels

  Takashi Murayama, Nagomi Kurebayashi, Mari Ishigami-Yuasa, Shuichi Mori, Yukina Suzuki, Ryunosuke Akima, Haruo Ogawa, Junji Suzuki, Kazunori Kanemaru, Hideto Oyamada, Yuji Kiuchi, Masamitsu Iino, Hiroyuki Kagechika and Takashi Sakurai

  Molecular Pharmacology July 2018, 94 (1) 722-730; DOI: https://doi.org/10.1124/mol.117.111468
• You have access

  Restoration of Physiological Expression of 5-HT₆ Receptor into the Primary Cilia of Null Mutant Neurons Lengthens Both Primary Cilia and Dendrites

  Atom J. Lesiak, Matthew Brodsky, Nathalie Cohenca, Alexandra G. Croicu and John F. Neumaier

  Molecular Pharmacology July 2018, 94 (1) 731-742; DOI: https://doi.org/10.1124/mol.117.111583
• You have access

  Cannabidiol Inhibits Endocannabinoid Signaling in Autaptic Hippocampal Neurons

  Alex Straiker, Michaela Dvorakova, Anaelle Zimmowitch and Ken Mackie

  Molecular Pharmacology July 2018, 94 (1) 743-748; DOI: https://doi.org/10.1124/mol.118.111864
• You have access

  A Transcriptional Regulatory Network Containing Nuclear Receptors and Long Noncoding RNAs Controls Basal and Drug-Induced Expression of Cytochrome P450s in HepaRG Cells

  Liming Chen, Yifan Bao, Stephanie C. Piekos, Kexin Zhu, Lirong Zhang and Xiao-bo Zhong

  Molecular Pharmacology July 2018, 94 (1) 749-759; DOI: https://doi.org/10.1124/mol.118.112235
• You have access

  The Temperature Dependence of Kinetics Associated with Drug Block of hERG Channels Is Compound-Specific and an Important Factor for Proarrhythmic Risk Prediction

  Monique J. Windley, William Lee, Jamie I. Vandenberg and Adam P. Hill

  Molecular Pharmacology July 2018, 94 (1) 760-769; DOI: https://doi.org/10.1124/mol.117.111534
• You have access

  Assessment of the Molecular Mechanisms of Action of Novel 4-Phenylpyridine-2-One and 6-Phenylpyrimidin-4-One Allosteric Modulators at the M₁ Muscarinic Acetylcholine Receptors

  Emma T. van der Westhuizen, Arthur Spathis, Elham Khajehali, Manuela Jörg, Shailesh N. Mistry, Ben Capuano, Andrew B. Tobin, Patrick M. Sexton, Peter J. Scammells, Celine Valant and Arthur Christopoulos

  Molecular Pharmacology July 2018, 94 (1) 770-783; DOI: https://doi.org/10.1124/mol.118.111633