Research ArticleArticle
Assessment of Substrate-Dependent Ligand Interactions at the Organic Cation Transporter OCT2 Using Six Model Substrates
Philip J. Sandoval, Kimberley M. Zorn, Alex M. Clark, Sean Ekins and Stephen H. Wright
Molecular Pharmacology September 2018, 94 (3) 1057-1068; DOI: https://doi.org/10.1124/mol.117.111443
Philip J. Sandoval
Department of Physiology, College of Medicine, University of Arizona, Tucson, Arizona (P.J.S., S.H.W.); Collaborations Pharmaceuticals, Inc., Raleigh, North Carolina (K.M.Z., S.E.); and Molecular Materials Informatics, Inc., Montreal, Quebec, Canada (A.M.C.)
Kimberley M. Zorn
Department of Physiology, College of Medicine, University of Arizona, Tucson, Arizona (P.J.S., S.H.W.); Collaborations Pharmaceuticals, Inc., Raleigh, North Carolina (K.M.Z., S.E.); and Molecular Materials Informatics, Inc., Montreal, Quebec, Canada (A.M.C.)
Alex M. Clark
Department of Physiology, College of Medicine, University of Arizona, Tucson, Arizona (P.J.S., S.H.W.); Collaborations Pharmaceuticals, Inc., Raleigh, North Carolina (K.M.Z., S.E.); and Molecular Materials Informatics, Inc., Montreal, Quebec, Canada (A.M.C.)
Sean Ekins
Department of Physiology, College of Medicine, University of Arizona, Tucson, Arizona (P.J.S., S.H.W.); Collaborations Pharmaceuticals, Inc., Raleigh, North Carolina (K.M.Z., S.E.); and Molecular Materials Informatics, Inc., Montreal, Quebec, Canada (A.M.C.)
Stephen H. Wright
Department of Physiology, College of Medicine, University of Arizona, Tucson, Arizona (P.J.S., S.H.W.); Collaborations Pharmaceuticals, Inc., Raleigh, North Carolina (K.M.Z., S.E.); and Molecular Materials Informatics, Inc., Montreal, Quebec, Canada (A.M.C.)
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Research ArticleArticle
Substrate Dependence of OCT2 Inhibition
Philip J. Sandoval, Kimberley M. Zorn, Alex M. Clark, Sean Ekins and Stephen H. Wright
Molecular Pharmacology September 1, 2018, 94 (3) 1057-1068; DOI: https://doi.org/10.1124/mol.117.111443
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