Table of Contents

Articles

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  Pyrimidinyl Biphenylureas Act as Allosteric Modulators to Activate Cannabinoid Receptor 1 and Initiate β-Arrestin–Dependent Responses

  Caitlin A. D. Jagla, Caitlin E. Scott, Yaliang Tang, Changjiang Qiao, Gabriel E. Mateo-Semidey, Guillermo A. Yudowski, Dai Lu and Debra A. Kendall

  Molecular Pharmacology January 2019, 95 (1) 1-10; DOI: https://doi.org/10.1124/mol.118.112854
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  Regulation of an Opioid Receptor Chaperone Protein, RTP4, by Morphine

  Wakako Fujita, Mini Yokote, Ivone Gomes, Achla Gupta, Hiroshi Ueda and Lakshmi A. Devi

  Molecular Pharmacology January 2019, 95 (1) 11-19; DOI: https://doi.org/10.1124/mol.118.112987
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  Subcellular Localization and Activity of the Mitogen-Activated Protein Kinase Kinase 7 (MKK7) γ Isoform are Regulated through Binding to the Phosphatase Calcineurin

  Emily S. Gibson, Kevin M. Woolfrey, Huiming Li, Patrick G. Hogan, Raphael A. Nemenoff, Lynn E. Heasley and Mark L. Dell’Acqua

  Molecular Pharmacology January 2019, 95 (1) 20-32; DOI: https://doi.org/10.1124/mol.118.113159
• Open Access

  Substrate-Induced Motion between TM4 and TM7 of the Glutamate Transporter EAAT1 Revealed by Paired Cysteine Mutagenesis

  Wenlong Zhang, Xiuping Zhang and Shaogang Qu

  Molecular Pharmacology January 2019, 95 (1) 33-42; DOI: https://doi.org/10.1124/mol.118.113183
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  Macroscopic and Microscopic Activation of α7 Nicotinic Acetylcholine Receptors by the Structurally Unrelated Allosteric Agonist-Positive Allosteric Modulators (ago-PAMs) B-973B and GAT107

  Marta Quadri, Sumanta Garai, Ganesh A. Thakur, Clare Stokes, Alican Gulsevin, Nicole A. Horenstein and Roger L. Papke

  Molecular Pharmacology January 2019, 95 (1) 43-61; DOI: https://doi.org/10.1124/mol.118.113340
• Open Access

  N-Phthalyl-l-Tryptophan (RG108), like Clozapine (CLO), Induces Chromatin Remodeling in Brains of Prenatally Stressed Mice

  Erbo Dong, Valentina Locci, Eleonora Gatta, Dennis R. Grayson and Alessandro Guidotti

  Molecular Pharmacology January 2019, 95 (1) 62-69; DOI: https://doi.org/10.1124/mol.118.113415
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  Analysis of GABA_A Receptor Activation by Combinations of Agonists Acting at the Same or Distinct Binding Sites

  Daniel J. Shin, Allison L. Germann, Douglas F. Covey, Joe Henry Steinbach and Gustav Akk

  Molecular Pharmacology January 2019, 95 (1) 70-81; DOI: https://doi.org/10.1124/mol.118.113464
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  A Modified Tripeptide Motif of RS1 (RSC1A1) Down-Regulates Exocytotic Pathways of Human Na⁺-d-glucose Cotransporters SGLT1, SGLT2, and Glucose Sensor SGLT3 in the Presence of Glucose

  Nadine Schäfer, Prashanth Reddy Rikkala, Maike Veyhl-Wichmann, Thorsten Keller, Christian Ferdinand Jurowich, Dietmar Geiger and Hermann Koepsell

  Molecular Pharmacology January 2019, 95 (1) 82-96; DOI: https://doi.org/10.1124/mol.118.113514
• Open Access

  Constitutive Androstane Receptor 1 is Constitutively Bound to Chromatin and 'Primed' for Transactivation in Hepatocytes

  Michael McMahon, Shaohong Ding, Lourdes Acosta Jimenez, Remi Terranova, Marie-Apolline Gerard, Antonio Vitobello, Jonathan Moggs, Colin J. Henderson and C. Roland Wolf

  Molecular Pharmacology January 2019, 95 (1) 97-105; DOI: https://doi.org/10.1124/mol.118.113555
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  Cell Cycle and Apoptosis Regulator 1, CCAR1, Regulates Enhancer-Dependent Nuclear Receptor CAR Transactivation

  Yuichiro Kanno, Shuai Zhao, Naoya Yamashita, Nao Saito, Aoi Ujiie, Rie Iijima, Nami Kikawa, Kiyomitsu Nemoto and Yoshio Inouye

  Molecular Pharmacology January 2019, 95 (1) 120-126; DOI: https://doi.org/10.1124/mol.118.114272
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  Lysosome Membrane Permeabilization and Disruption of the Molecular Target of Rapamycin (mTOR)-Lysosome Interaction Are Associated with the Inhibition of Lung Cancer Cell Proliferation by a Chloroquinoline Analog

  Juan Sironi, Evelyn Aranda, Lars Ulrik Nordstrøm and Edward L. Schwartz

  Molecular Pharmacology January 2019, 95 (1) 127-138; DOI: https://doi.org/10.1124/mol.118.113118
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  Identification of Peracetylated Quercetin as a Selective 12-Lipoxygenase Pathway Inhibitor in Human Platelets

  Marco S. Doucet, Jean-Luc Jougleux, Samuel J. Poirier, Marc Cormier, Jacob L. Léger, Marc E. Surette, Nicolas Pichaud, Mohamed Touaibia and Luc H. Boudreau

  Molecular Pharmacology January 2019, 95 (1) 139-150; DOI: https://doi.org/10.1124/mol.118.113480