Table of Contents

Articles

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  Cannabinoid CB2 Agonist AM1710 Differentially Suppresses Distinct Pathological Pain States and Attenuates Morphine Tolerance and Withdrawal

  Ai-Ling Li, Xiaoyan Lin, Amey S. Dhopeshwarkar, Ana Carla Thomaz, Lawrence M. Carey, Yingpeng Liu, Spyros P. Nikas, Alexandros Makriyannis, Ken Mackie and Andrea G. Hohmann

  Molecular Pharmacology February 2019, 95 (2) 155-168; DOI: https://doi.org/10.1124/mol.118.113233
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  Rat Organic Cation Transporter 1 Contains Three Binding Sites for Substrate 1-Methyl-4-phenylpyridinium per Monomer

  Thorsten Keller, Valentin Gorboulev, Thomas D. Mueller, Volker Dötsch, Frank Bernhard and Hermann Koepsell

  Molecular Pharmacology February 2019, 95 (2) 169-182; DOI: https://doi.org/10.1124/mol.118.113498
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  Efavirenz and Efavirenz-like Compounds Activate Human, Murine, and Macaque Hepatic IRE1α-XBP1

  Carley J. S. Heck, Allyson N. Hamlin and Namandjé N. Bumpus

  Molecular Pharmacology February 2019, 95 (2) 183-195; DOI: https://doi.org/10.1124/mol.118.113647
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  Open Access

  Design, Synthesis, and Evaluation of a Diazirine Photoaffinity Probe for Ligand-Based Receptor Capture Targeting G Protein–Coupled Receptors

  Frederike M. Müskens, Richard J. Ward, Dominik Herkt, Helmus van de Langemheen, Andrew B. Tobin, Rob M. J. Liskamp and Graeme Milligan

  Molecular Pharmacology February 2019, 95 (2) 196-209; DOI: https://doi.org/10.1124/mol.118.114249
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  Ginsenosides Act As Positive Modulators of P2X4 Receptors

  Kshitija Dhuna, Matthew Felgate, Stefan M. Bidula, Samuel Walpole, Lucka Bibic, Brett A. Cromer, Jesus Angulo, Julie Sanderson, Martin J. Stebbing and Leanne Stokes

  Molecular Pharmacology February 2019, 95 (2) 210-221; DOI: https://doi.org/10.1124/mol.118.113696
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  Preclinical Evaluation of AZ12601011 and AZ12799734, Inhibitors of Transforming Growth Factor β Superfamily Type 1 Receptors

  Lindsay C. Spender, G. John Ferguson, Gareth D. Hughes, Barry R. Davies, Frederick W. Goldberg, Blanca Herrera, Richard G. Taylor, Lauren S. Strathearn, Owen J. Sansom, Simon T. Barry and Gareth J. Inman

  Molecular Pharmacology February 2019, 95 (2) 222-234; DOI: https://doi.org/10.1124/mol.118.112946