Table of Contents

Articles

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  Mexiletine Block of Voltage-Gated Sodium Channels: Isoform- and State-Dependent Drug–Pore Interactions

  Hiroki Nakagawa, Tatsuo Munakata and Akihiko Sunami

  Molecular Pharmacology March 2019, 95 (3) 236-244; DOI: https://doi.org/10.1124/mol.118.114025
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  Molecular Basis of Action of a Small-Molecule Positive Allosteric Modulator Agonist at the Type 1 Cholecystokinin Holoreceptor

  Aditya J. Desai, Ingrid Mechin, Karthigeyan Nagarajan, Celine Valant, Denise Wootten, Polo C. H. Lam, Andrew Orry, Ruben Abagyan, Anil Nair, Patrick M. Sexton, Arthur Christopoulos and Laurence J. Miller

  Molecular Pharmacology March 2019, 95 (3) 245-259; DOI: https://doi.org/10.1124/mol.118.114082
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  Repeated Exposure to 4-Methyl-2,4-bis(4-hydroxyphenyl)pent-1-ene (MBP), an Active Metabolite of Bisphenol A, Aggressively Stimulates Breast Cancer Cell Growth in an Estrogen Receptor β (ERβ)–Dependent Manner

  Masayo Hirao-Suzuki, Shuso Takeda, Katsuhiro Okuda, Masufumi Takiguchi and Shin’ichi Yoshihara

  Molecular Pharmacology March 2019, 95 (3) 260-268; DOI: https://doi.org/10.1124/mol.118.114124
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  S29434, a Quinone Reductase 2 Inhibitor: Main Biochemical and Cellular Characterization

  Jean A. Boutin, Frederic Bouillaud, Elzbieta Janda, István Gacsalyi, Gérald Guillaumet, Etienne C. Hirsch, Daniel A. Kane, Françoise Nepveu, Karine Reybier, Philippe Dupuis, Marc Bertrand, Monivan Chhour, Thierry Le Diguarher, Mathias Antoine, Karen Brebner, Hervé Da Costa, Pierre Ducrot, Adeline Giganti, Vishalgiri Goswami, Hala Guedouari, Patrick P. Michel, Aakash Patel, Jérôme Paysant, Johann Stojko, Marie-Claude Viaud-Massuard and Gilles Ferry

  Molecular Pharmacology March 2019, 95 (3) 269-285; DOI: https://doi.org/10.1124/mol.118.114231
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  Structural Basis of p97 Inhibition by the Site-Selective Anticancer Compound CB-5083

  Wai Kwan Tang, Taivan Odzorig, Whitney Jin and Di Xia

  Molecular Pharmacology March 2019, 95 (3) 286-293; DOI: https://doi.org/10.1124/mol.118.114256
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  Inhibition of Interleukin 10 Transcription through the SMAD2/3 Signaling Pathway by Ca²⁺-Activated K⁺ Channel K_Ca3.1 Activation in Human T-Cell Lymphoma HuT-78 Cells

  Miki Matsui, Junko Kajikuri, Hiroaki Kito, Kyoko Endo, Yuki Hasegawa, Shinya Murate and Susumu Ohya

  Molecular Pharmacology March 2019, 95 (3) 294-302; DOI: https://doi.org/10.1124/mol.118.114405
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  Hyperforin-Induced Activation of the Pregnane X Receptor Is Influenced by the Organic Anion-Transporting Polypeptide 2B1

  Anima M. Schäfer, Olivier Potterat, Isabell Seibert, Orlando Fertig and Henriette E. Meyer zu Schwabedissen

  Molecular Pharmacology March 2019, 95 (3) 313-323; DOI: https://doi.org/10.1124/mol.118.114066
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  Belinostat, at Its Clinically Relevant Concentrations, Inhibits Rifampicin-Induced CYP3A4 and MDR1 Gene Expression

  Kodye L. Abbott, Chloe S. Chaudhury, Aneesh Chandran, Saraswathi Vishveshwara, Zdenek Dvorak, Eva Jiskrova, Karolina Poulikova, Barbora Vyhlidalova, Sridhar Mani and Satyanarayana R. Pondugula

  Molecular Pharmacology March 2019, 95 (3) 324-334; DOI: https://doi.org/10.1124/mol.118.114587