Table of Contents

Articles

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  Innovative Bioluminescence Resonance Energy Transfer Assay Reveals Differential Agonist-Induced D2 Receptor Intracellular Trafficking and Arrestin-3 Recruitment

  Luc De Vries, Frédéric Finana, Claudie Cathala, Brice Ronsin and Didier Cussac

  Molecular Pharmacology September 2019, 96 (3) 308-319; DOI: https://doi.org/10.1124/mol.119.115998
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  Steady-State Activation and Modulation of the Concatemeric α1β2γ2L GABA_A Receptor

  Allison L. Germann, Spencer R. Pierce, Ariel B. Burbridge, Joe Henry Steinbach and Gustav Akk

  Molecular Pharmacology September 2019, 96 (3) 320-329; DOI: https://doi.org/10.1124/mol.119.116913
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  Temperature Dependence of the Biophysical Mechanisms Underlying the Inhibition and Enhancement Effect of Amiodarone on hERG Channels

  Yung-Chen Lo and Chung-Chin Kuo

  Molecular Pharmacology September 2019, 96 (3) 330-344; DOI: https://doi.org/10.1124/mol.119.116400
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  Mechanistic Insights of Phenobarbital-Mediated Activation of Human but Not Mouse Pregnane X Receptor

  Linhao Li, Matthew A. Welch, Zhihui Li, Bryan Mackowiak, Scott Heyward, Peter W. Swaan and Hongbing Wang

  Molecular Pharmacology September 2019, 96 (3) 345-354; DOI: https://doi.org/10.1124/mol.119.116616
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  Mapping the Site of Action of Human P2X7 Receptor Antagonists AZ11645373, Brilliant Blue G, KN-62, Calmidazolium, and ZINC58368839 to the Intersubunit Allosteric Pocket

  Anfal Bin Dayel, Richard J. Evans and Ralf Schmid

  Molecular Pharmacology September 2019, 96 (3) 355-363; DOI: https://doi.org/10.1124/mol.119.116715
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  Characterization and Proteomic-Transcriptomic Investigation of Monocarboxylate Transporter 6 Knockout Mice: Evidence of a Potential Role in Glucose and Lipid Metabolism

  Robert S. Jones, Chengjian Tu, Ming Zhang, Jun Qu and Marilyn E. Morris

  Molecular Pharmacology September 2019, 96 (3) 364-376; DOI: https://doi.org/10.1124/mol.119.116731
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  Investigating the Influence of Tracer Kinetics on Competition-Kinetic Association Binding Assays: Identifying the Optimal Conditions for Assessing the Kinetics of Low-Affinity Compounds

  David A. Sykes, Palash Jain and Steven J. Charlton

  Molecular Pharmacology September 2019, 96 (3) 378-392; DOI: https://doi.org/10.1124/mol.119.116764
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  Inhibition of the Warm Temperature–Activated Ca²⁺-Permeable Transient Receptor Potential Vanilloid TRPV3 Channel Attenuates Atopic Dermatitis

  Yaxuan Qu, Gongxin Wang, Xiaoying Sun and KeWei Wang

  Molecular Pharmacology September 2019, 96 (3) 393-400; DOI: https://doi.org/10.1124/mol.119.116962
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  Dantrolene Requires Mg²⁺ and ATP To Inhibit the Ryanodine Receptor

  Gyula Diszházi, Zsuzsanna Édua Magyar, János András Mótyán, László Csernoch, István Jóna, Péter Pál Nánási and János Almássy

  Molecular Pharmacology September 2019, 96 (3) 401-407; DOI: https://doi.org/10.1124/mol.119.116475