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Index by author

November 01, 2019; Volume 96,Issue 5

A

  1. Abe, Satoshi

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  2. Ambudkar, Suresh V.

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  3. Asai, Akira

    1. Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Jun-ichi Sawada, Hirosuke Ishii, Kenji Matsuno, Masayuki Sato, Yumiko Suzuki and Akira Asai
      Molecular Pharmacology November 2019, 96 (5) 609-618; DOI: https://doi.org/10.1124/mol.119.116624

  4. Austin, Caroline A.

    1. Open Access
      The Deubiquitinating Enzyme Inhibitor PR-619 is a Potent DNA Topoisomerase II Poison
      Ian G. Cowell, Elise M. Ling, Rebecca L. Swan, Matilda L.W. Brooks and Caroline A. Austin
      Molecular Pharmacology November 2019, 96 (5) 562-572; DOI: https://doi.org/10.1124/mol.119.117390

B

  1. Ben-Tal, Nir

    1. Metal Coordination Is Crucial for Geranylgeranyl Diphosphate Synthase–Bisphosphonate Interactions: A Crystallographic and Computational Analysis
      Michal Lisnyansky, Elon Yariv, Omri Segal, Milit Marom, Anat Loewenstein, Nir Ben-Tal, Moshe Giladi and Yoni Haitin
      Molecular Pharmacology November 2019, 96 (5) 580-588; DOI: https://doi.org/10.1124/mol.119.117499

  2. Bohn, Laura M.

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  3. Brimacombe, Kyle R.

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  4. Brooks, Matilda L.W.

    1. Open Access
      The Deubiquitinating Enzyme Inhibitor PR-619 is a Potent DNA Topoisomerase II Poison
      Ian G. Cowell, Elise M. Ling, Rebecca L. Swan, Matilda L.W. Brooks and Caroline A. Austin
      Molecular Pharmacology November 2019, 96 (5) 562-572; DOI: https://doi.org/10.1124/mol.119.117390

  5. Butcher, Neville J.

    1. Arylamine N-Acetyltransferase 1 Regulates Expression of Matrix Metalloproteinase 9 in Breast Cancer Cells: Role of Hypoxia-Inducible Factor 1-α
      Pengcheng Li, Neville J. Butcher and Rodney F. Minchin
      Molecular Pharmacology November 2019, 96 (5) 573-579; DOI: https://doi.org/10.1124/mol.119.117432

C

  1. Cao, Zhi-Xing

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  2. Chen, Jian-Ping

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  3. Chen, Lu

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  4. Conibear, Alexandra E.

    1. A Biased View of μ-Opioid Receptors?
      Alexandra E. Conibear and Eamonn Kelly
      Molecular Pharmacology November 2019, 96 (5) 542-549; DOI: https://doi.org/10.1124/mol.119.115956

  5. Correia, Maria Almira

    1. Induction via Functional Protein Stabilization of Hepatic Cytochromes P450 upon gp78/Autocrine Motility Factor Receptor (AMFR) Ubiquitin E3-Ligase Genetic Ablation in Mice: Therapeutic and Toxicological Relevance
      Doyoung Kwon, Sung-Mi Kim, Peyton Jacob, Yi Liu and Maria Almira Correia
      Molecular Pharmacology November 2019, 96 (5) 641-654; DOI: https://doi.org/10.1124/mol.119.117069

  6. Cowell, Ian G.

    1. Open Access
      The Deubiquitinating Enzyme Inhibitor PR-619 is a Potent DNA Topoisomerase II Poison
      Ian G. Cowell, Elise M. Ling, Rebecca L. Swan, Matilda L.W. Brooks and Caroline A. Austin
      Molecular Pharmacology November 2019, 96 (5) 562-572; DOI: https://doi.org/10.1124/mol.119.117390

E

  1. Egorova, Natalia S.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

F

  1. Fourmy, Daniel

    1. Understanding Peptide Binding in Class A G Protein-Coupled Receptors
      Irina G. Tikhonova, Veronique Gigoux and Daniel Fourmy
      Molecular Pharmacology November 2019, 96 (5) 550-561; DOI: https://doi.org/10.1124/mol.119.115915

G

  1. Gao, Fei

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  2. GC, Jeevan B.

    1. Does the Lipid Bilayer Orchestrate Access and Binding of Ligands to Transmembrane Orthosteric/Allosteric Sites of G Protein-Coupled Receptors?
      Does the Lipid Bilayer Orchestrate Access and Binding of Ligands to Transmembrane Orthosteric/Allosteric Sites of G Protein-Coupled Receptors?
      Christopher T. Szlenk, Jeevan B. GC and Senthil Natesan
      Molecular Pharmacology November 2019, 96 (5) 527-541; DOI: https://doi.org/10.1124/mol.118.115113

  3. Gigoux, Veronique

    1. Understanding Peptide Binding in Class A G Protein-Coupled Receptors
      Irina G. Tikhonova, Veronique Gigoux and Daniel Fourmy
      Molecular Pharmacology November 2019, 96 (5) 550-561; DOI: https://doi.org/10.1124/mol.119.115915

  4. Giladi, Moshe

    1. Metal Coordination Is Crucial for Geranylgeranyl Diphosphate Synthase–Bisphosphonate Interactions: A Crystallographic and Computational Analysis
      Michal Lisnyansky, Elon Yariv, Omri Segal, Milit Marom, Anat Loewenstein, Nir Ben-Tal, Moshe Giladi and Yoni Haitin
      Molecular Pharmacology November 2019, 96 (5) 580-588; DOI: https://doi.org/10.1124/mol.119.117499

  5. Gong, Dao-Yin

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  6. Gottesman, Michael M.

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  7. Grim, Travis W.

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  8. Guha, Rajarshi

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  9. Guo, Chuan-Jie

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

H

  1. Haitin, Yoni

    1. Metal Coordination Is Crucial for Geranylgeranyl Diphosphate Synthase–Bisphosphonate Interactions: A Crystallographic and Computational Analysis
      Michal Lisnyansky, Elon Yariv, Omri Segal, Milit Marom, Anat Loewenstein, Nir Ben-Tal, Moshe Giladi and Yoni Haitin
      Molecular Pharmacology November 2019, 96 (5) 580-588; DOI: https://doi.org/10.1124/mol.119.117499

  2. Hall, Matthew D.

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  3. He, Jun-Lin

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  4. Ho, Jo-Hao

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  5. Honkakoski, Paavo

    1. The Basis for Strain-Dependent Rat Aldehyde Dehydrogenase 1A7 (ALDH1A7) Gene Expression
      Katerina Touloupi, Jenni Küblbeck, Angeliki Magklara, Ferdinand Molnár, Mika Reinisalo, Maria Konstandi, Paavo Honkakoski and Periklis Pappas
      Molecular Pharmacology November 2019, 96 (5) 655-663; DOI: https://doi.org/10.1124/mol.119.117424

  6. Hua, Tian

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  7. Huang, Shen-Zhen

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

I

  1. Iagorshvili, Ia

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  2. Igarashi, Katsuhide

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  3. Ishii, Hirosuke

    1. Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Jun-ichi Sawada, Hirosuke Ishii, Kenji Matsuno, Masayuki Sato, Yumiko Suzuki and Akira Asai
      Molecular Pharmacology November 2019, 96 (5) 609-618; DOI: https://doi.org/10.1124/mol.119.116624

  4. Ivanov, Igor A.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

J

  1. Jacob, Peyton

    1. Induction via Functional Protein Stabilization of Hepatic Cytochromes P450 upon gp78/Autocrine Motility Factor Receptor (AMFR) Ubiquitin E3-Ligase Genetic Ablation in Mice: Therapeutic and Toxicological Relevance
      Doyoung Kwon, Sung-Mi Kim, Peyton Jacob, Yi Liu and Maria Almira Correia
      Molecular Pharmacology November 2019, 96 (5) 641-654; DOI: https://doi.org/10.1124/mol.119.117069

K

  1. Kanno, Jun

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  2. Kasheverov, Igor E.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  3. Katsarava, Ramaz

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  4. Kazuki, Yasuhiro

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  5. Kelly, Eamonn

    1. A Biased View of μ-Opioid Receptors?
      Alexandra E. Conibear and Eamonn Kelly
      Molecular Pharmacology November 2019, 96 (5) 542-549; DOI: https://doi.org/10.1124/mol.119.115956

  6. Kim, Sung-Mi

    1. Induction via Functional Protein Stabilization of Hepatic Cytochromes P450 upon gp78/Autocrine Motility Factor Receptor (AMFR) Ubiquitin E3-Ligase Genetic Ablation in Mice: Therapeutic and Toxicological Relevance
      Doyoung Kwon, Sung-Mi Kim, Peyton Jacob, Yi Liu and Maria Almira Correia
      Molecular Pharmacology November 2019, 96 (5) 641-654; DOI: https://doi.org/10.1124/mol.119.117069

  7. Kitajima, Satoshi

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  8. Klumpp-Thomas, Carleen

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  9. Kobayashi, Kaoru

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  10. Konstandi, Maria

    1. The Basis for Strain-Dependent Rat Aldehyde Dehydrogenase 1A7 (ALDH1A7) Gene Expression
      Katerina Touloupi, Jenni Küblbeck, Angeliki Magklara, Ferdinand Molnár, Mika Reinisalo, Maria Konstandi, Paavo Honkakoski and Periklis Pappas
      Molecular Pharmacology November 2019, 96 (5) 655-663; DOI: https://doi.org/10.1124/mol.119.117424

  11. Korde, Anisha

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  12. Kryukova, Elena V.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  13. Küblbeck, Jenni

    1. The Basis for Strain-Dependent Rat Aldehyde Dehydrogenase 1A7 (ALDH1A7) Gene Expression
      Katerina Touloupi, Jenni Küblbeck, Angeliki Magklara, Ferdinand Molnár, Mika Reinisalo, Maria Konstandi, Paavo Honkakoski and Periklis Pappas
      Molecular Pharmacology November 2019, 96 (5) 655-663; DOI: https://doi.org/10.1124/mol.119.117424

  14. Kudryavtsev, Denis S.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  15. Kuze, Jiro

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  16. Kwon, Doyoung

    1. Induction via Functional Protein Stabilization of Hepatic Cytochromes P450 upon gp78/Autocrine Motility Factor Receptor (AMFR) Ubiquitin E3-Ligase Genetic Ablation in Mice: Therapeutic and Toxicological Relevance
      Doyoung Kwon, Sung-Mi Kim, Peyton Jacob, Yi Liu and Maria Almira Correia
      Molecular Pharmacology November 2019, 96 (5) 641-654; DOI: https://doi.org/10.1124/mol.119.117069

L

  1. Laprairie, Robert B.

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  2. Lebedev, Dmitry S.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  3. Lee, Olivia W.

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  4. Lee, Tobie D.

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  5. Li, Pengcheng

    1. Arylamine N-Acetyltransferase 1 Regulates Expression of Matrix Metalloproteinase 9 in Breast Cancer Cells: Role of Hypoxia-Inducible Factor 1-α
      Pengcheng Li, Neville J. Butcher and Rodney F. Minchin
      Molecular Pharmacology November 2019, 96 (5) 573-579; DOI: https://doi.org/10.1124/mol.119.117432

  6. Li, Yu-Zhi

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  7. Ling, Elise M.

    1. Open Access
      The Deubiquitinating Enzyme Inhibitor PR-619 is a Potent DNA Topoisomerase II Poison
      Ian G. Cowell, Elise M. Ling, Rebecca L. Swan, Matilda L.W. Brooks and Caroline A. Austin
      Molecular Pharmacology November 2019, 96 (5) 562-572; DOI: https://doi.org/10.1124/mol.119.117390

  8. Lisnyansky, Michal

    1. Metal Coordination Is Crucial for Geranylgeranyl Diphosphate Synthase–Bisphosphonate Interactions: A Crystallographic and Computational Analysis
      Michal Lisnyansky, Elon Yariv, Omri Segal, Milit Marom, Anat Loewenstein, Nir Ben-Tal, Moshe Giladi and Yoni Haitin
      Molecular Pharmacology November 2019, 96 (5) 580-588; DOI: https://doi.org/10.1124/mol.119.117499

  9. Liu, Qing-Qing

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  10. Liu, Yi

    1. Induction via Functional Protein Stabilization of Hepatic Cytochromes P450 upon gp78/Autocrine Motility Factor Receptor (AMFR) Ubiquitin E3-Ligase Genetic Ablation in Mice: Therapeutic and Toxicological Relevance
      Doyoung Kwon, Sung-Mi Kim, Peyton Jacob, Yi Liu and Maria Almira Correia
      Molecular Pharmacology November 2019, 96 (5) 641-654; DOI: https://doi.org/10.1124/mol.119.117069

  11. Liu, Zhi-Jie

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  12. Loewenstein, Anat

    1. Metal Coordination Is Crucial for Geranylgeranyl Diphosphate Synthase–Bisphosphonate Interactions: A Crystallographic and Computational Analysis
      Michal Lisnyansky, Elon Yariv, Omri Segal, Milit Marom, Anat Loewenstein, Nir Ben-Tal, Moshe Giladi and Yoni Haitin
      Molecular Pharmacology November 2019, 96 (5) 580-588; DOI: https://doi.org/10.1124/mol.119.117499

  13. Lusvarghi, Sabrina

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

M

  1. Magklara, Angeliki

    1. The Basis for Strain-Dependent Rat Aldehyde Dehydrogenase 1A7 (ALDH1A7) Gene Expression
      Katerina Touloupi, Jenni Küblbeck, Angeliki Magklara, Ferdinand Molnár, Mika Reinisalo, Maria Konstandi, Paavo Honkakoski and Periklis Pappas
      Molecular Pharmacology November 2019, 96 (5) 655-663; DOI: https://doi.org/10.1124/mol.119.117424

  2. Makriyannis, Alexandros

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  3. Marom, Milit

    1. Metal Coordination Is Crucial for Geranylgeranyl Diphosphate Synthase–Bisphosphonate Interactions: A Crystallographic and Computational Analysis
      Michal Lisnyansky, Elon Yariv, Omri Segal, Milit Marom, Anat Loewenstein, Nir Ben-Tal, Moshe Giladi and Yoni Haitin
      Molecular Pharmacology November 2019, 96 (5) 580-588; DOI: https://doi.org/10.1124/mol.119.117499

  4. Matsuno, Kenji

    1. Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Jun-ichi Sawada, Hirosuke Ishii, Kenji Matsuno, Masayuki Sato, Yumiko Suzuki and Akira Asai
      Molecular Pharmacology November 2019, 96 (5) 609-618; DOI: https://doi.org/10.1124/mol.119.116624

  5. Minchin, Rodney F.

    1. Arylamine N-Acetyltransferase 1 Regulates Expression of Matrix Metalloproteinase 9 in Breast Cancer Cells: Role of Hypoxia-Inducible Factor 1-α
      Pengcheng Li, Neville J. Butcher and Rodney F. Minchin
      Molecular Pharmacology November 2019, 96 (5) 573-579; DOI: https://doi.org/10.1124/mol.119.117432

  6. Minegishi, Genki

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  7. Molnár, Ferdinand

    1. The Basis for Strain-Dependent Rat Aldehyde Dehydrogenase 1A7 (ALDH1A7) Gene Expression
      Katerina Touloupi, Jenni Küblbeck, Angeliki Magklara, Ferdinand Molnár, Mika Reinisalo, Maria Konstandi, Paavo Honkakoski and Periklis Pappas
      Molecular Pharmacology November 2019, 96 (5) 655-663; DOI: https://doi.org/10.1124/mol.119.117424

N

  1. Natesan, Senthil

    1. Does the Lipid Bilayer Orchestrate Access and Binding of Ligands to Transmembrane Orthosteric/Allosteric Sites of G Protein-Coupled Receptors?
      Does the Lipid Bilayer Orchestrate Access and Binding of Ligands to Transmembrane Orthosteric/Allosteric Sites of G Protein-Coupled Receptors?
      Christopher T. Szlenk, Jeevan B. GC and Senthil Natesan
      Molecular Pharmacology November 2019, 96 (5) 527-541; DOI: https://doi.org/10.1124/mol.118.115113

O

  1. Oshimura, Mitsuo

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

P

  1. Pappas, Periklis

    1. The Basis for Strain-Dependent Rat Aldehyde Dehydrogenase 1A7 (ALDH1A7) Gene Expression
      Katerina Touloupi, Jenni Küblbeck, Angeliki Magklara, Ferdinand Molnár, Mika Reinisalo, Maria Konstandi, Paavo Honkakoski and Periklis Pappas
      Molecular Pharmacology November 2019, 96 (5) 655-663; DOI: https://doi.org/10.1124/mol.119.117424

  2. Peng, Cheng

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

R

  1. Reinisalo, Mika

    1. The Basis for Strain-Dependent Rat Aldehyde Dehydrogenase 1A7 (ALDH1A7) Gene Expression
      Katerina Touloupi, Jenni Küblbeck, Angeliki Magklara, Ferdinand Molnár, Mika Reinisalo, Maria Konstandi, Paavo Honkakoski and Periklis Pappas
      Molecular Pharmacology November 2019, 96 (5) 655-663; DOI: https://doi.org/10.1124/mol.119.117424

  2. Robey, Robert W.

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

S

  1. Sato, Masayuki

    1. Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Jun-ichi Sawada, Hirosuke Ishii, Kenji Matsuno, Masayuki Sato, Yumiko Suzuki and Akira Asai
      Molecular Pharmacology November 2019, 96 (5) 609-618; DOI: https://doi.org/10.1124/mol.119.116624

  2. Sawada, Jun-ichi

    1. Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Jun-ichi Sawada, Hirosuke Ishii, Kenji Matsuno, Masayuki Sato, Yumiko Suzuki and Akira Asai
      Molecular Pharmacology November 2019, 96 (5) 609-618; DOI: https://doi.org/10.1124/mol.119.116624

  3. Segal, Omri

    1. Metal Coordination Is Crucial for Geranylgeranyl Diphosphate Synthase–Bisphosphonate Interactions: A Crystallographic and Computational Analysis
      Michal Lisnyansky, Elon Yariv, Omri Segal, Milit Marom, Anat Loewenstein, Nir Ben-Tal, Moshe Giladi and Yoni Haitin
      Molecular Pharmacology November 2019, 96 (5) 580-588; DOI: https://doi.org/10.1124/mol.119.117499

  4. Shen, Min

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  5. Siniavin, Andrei E.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  6. Spirova, Ekaterina N.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  7. Stahl, Edward L.

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  8. Stevens, Raymond C.

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

  9. Suzuki, Yumiko

    1. Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Selective Inhibition of Spindle Microtubules by a Tubulin-Binding Quinazoline Derivative
      Jun-ichi Sawada, Hirosuke Ishii, Kenji Matsuno, Masayuki Sato, Yumiko Suzuki and Akira Asai
      Molecular Pharmacology November 2019, 96 (5) 609-618; DOI: https://doi.org/10.1124/mol.119.116624

  10. Swan, Rebecca L.

    1. Open Access
      The Deubiquitinating Enzyme Inhibitor PR-619 is a Potent DNA Topoisomerase II Poison
      Ian G. Cowell, Elise M. Ling, Rebecca L. Swan, Matilda L.W. Brooks and Caroline A. Austin
      Molecular Pharmacology November 2019, 96 (5) 562-572; DOI: https://doi.org/10.1124/mol.119.117390

  11. Szlenk, Christopher T.

    1. Does the Lipid Bilayer Orchestrate Access and Binding of Ligands to Transmembrane Orthosteric/Allosteric Sites of G Protein-Coupled Receptors?
      Does the Lipid Bilayer Orchestrate Access and Binding of Ligands to Transmembrane Orthosteric/Allosteric Sites of G Protein-Coupled Receptors?
      Christopher T. Szlenk, Jeevan B. GC and Senthil Natesan
      Molecular Pharmacology November 2019, 96 (5) 527-541; DOI: https://doi.org/10.1124/mol.118.115113

T

  1. Takehara, Shoko

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  2. Tebase, Bethilehem G.

    1. A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein
      Tobie D. Lee, Olivia W. Lee, Kyle R. Brimacombe, Lu Chen, Rajarshi Guha, Sabrina Lusvarghi, Bethilehem G. Tebase, Carleen Klumpp-Thomas, Robert W. Robey, Suresh V. Ambudkar, Min Shen, Michael M. Gottesman and Matthew D. Hall
      Molecular Pharmacology November 2019, 96 (5) 629-640; DOI: https://doi.org/10.1124/mol.119.115964

  3. Tikhonova, Irina G.

    1. Understanding Peptide Binding in Class A G Protein-Coupled Receptors
      Irina G. Tikhonova, Veronique Gigoux and Daniel Fourmy
      Molecular Pharmacology November 2019, 96 (5) 550-561; DOI: https://doi.org/10.1124/mol.119.115915

  4. Timofeev, Nikita D.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  5. Touloupi, Katerina

    1. The Basis for Strain-Dependent Rat Aldehyde Dehydrogenase 1A7 (ALDH1A7) Gene Expression
      Katerina Touloupi, Jenni Küblbeck, Angeliki Magklara, Ferdinand Molnár, Mika Reinisalo, Maria Konstandi, Paavo Honkakoski and Periklis Pappas
      Molecular Pharmacology November 2019, 96 (5) 655-663; DOI: https://doi.org/10.1124/mol.119.117424

  6. Tsetlin, Victor I.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  7. Tufanova, Elizaveta Yu.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  8. Tzartos, Socrates J.

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

V

  1. Vemuri, Kiran

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

W

  1. Wen, Yi

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  2. Wu, Yiran

    1. Probing the CB1 Cannabinoid Receptor Binding Pocket with AM6538, a High-Affinity Irreversible Antagonist
      Robert B. Laprairie, Kiran Vemuri, Edward L. Stahl, Anisha Korde, Jo-Hao Ho, Travis W. Grim, Tian Hua, Yiran Wu, Raymond C. Stevens, Zhi-Jie Liu, Alexandros Makriyannis and Laura M. Bohn
      Molecular Pharmacology November 2019, 96 (5) 619-628; DOI: https://doi.org/10.1124/mol.119.116483

Y

  1. Yamamoto, Takushi

    1. CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
      Kaoru Kobayashi, Jiro Kuze, Satoshi Abe, Shoko Takehara, Genki Minegishi, Katsuhide Igarashi, Satoshi Kitajima, Jun Kanno, Takushi Yamamoto, Mitsuo Oshimura and Yasuhiro Kazuki
      Molecular Pharmacology November 2019, 96 (5) 600-608; DOI: https://doi.org/10.1124/mol.119.117333

  2. Yariv, Elon

    1. Metal Coordination Is Crucial for Geranylgeranyl Diphosphate Synthase–Bisphosphonate Interactions: A Crystallographic and Computational Analysis
      Michal Lisnyansky, Elon Yariv, Omri Segal, Milit Marom, Anat Loewenstein, Nir Ben-Tal, Moshe Giladi and Yoni Haitin
      Molecular Pharmacology November 2019, 96 (5) 580-588; DOI: https://doi.org/10.1124/mol.119.117499

Z

  1. Zavradashvili, Nino

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713

  2. Zhang, Ruo-Qi

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  3. Zheng, Shu-Wen

    1. Isoliquiritigenin, an Orally Available Natural FLT3 Inhibitor from Licorice, Exhibits Selective Anti–Acute Myeloid Leukemia Efficacy In Vitro and In Vivo
      Zhi-Xing Cao, Yi Wen, Jun-Lin He, Shen-Zhen Huang, Fei Gao, Chuan-Jie Guo, Qing-Qing Liu, Shu-Wen Zheng, Dao-Yin Gong, Yu-Zhi Li, Ruo-Qi Zhang, Jian-Ping Chen and Cheng Peng
      Molecular Pharmacology November 2019, 96 (5) 589-599; DOI: https://doi.org/10.1124/mol.119.116129

  4. Zouridakis, Marios

    1. Oligoarginine Peptides, a New Family of Nicotinic Acetylcholine Receptor Inhibitors
      Dmitry S. Lebedev, Elena V. Kryukova, Igor A. Ivanov, Natalia S. Egorova, Nikita D. Timofeev, Ekaterina N. Spirova, Elizaveta Yu. Tufanova, Andrei E. Siniavin, Denis S. Kudryavtsev, Igor E. Kasheverov, Marios Zouridakis, Ramaz Katsarava, Nino Zavradashvili, Ia Iagorshvili, Socrates J. Tzartos and Victor I. Tsetlin
      Molecular Pharmacology November 2019, 96 (5) 664-673; DOI: https://doi.org/10.1124/mol.119.117713
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