Index by author
December 01, 2019; Volume 96,Issue 6
A
Adlere, Ilze
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Andersen, Signe
- You have accessConformational Changes in the 5-HT3A Receptor Extracellular Domain Measured by Voltage-Clamp FluorometryLachlan Munro, Lucy Kate Ladefoged, Vithushan Padmanathan, Signe Andersen, Birgit Schiøtt and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 720-734; DOI: https://doi.org/10.1124/mol.119.116657
Arimont, Marta
- Open AccessChemokine Receptor Crystal Structures: What Can Be Learned from Them?Marta Arimont, Carsten Hoffmann, Chris de Graaf and Rob LeursMolecular Pharmacology December 2019, 96 (6) 765-777; DOI: https://doi.org/10.1124/mol.119.117168
- Open AccessAntibodies Targeting Chemokine Receptors CXCR4 and ACKR3Vladimir Bobkov, Marta Arimont, Aurélien Zarca, Timo W.M. De Groof, Bas van der Woning, Hans de Haard and Martine J. SmitMolecular Pharmacology December 2019, 96 (6) 753-764; DOI: https://doi.org/10.1124/mol.119.116954
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
B
Bachelerie, Françoise
- You have accessAtypical Chemokine Receptor 3 (ACKR3): A Comprehensive Overview of its Expression and Potential Roles in the Immune SystemJoyce Koenen, Françoise Bachelerie, Karl Balabanian, Géraldine Schlecht-Louf and Carmen GallegoMolecular Pharmacology December 2019, 96 (6) 809-818; DOI: https://doi.org/10.1124/mol.118.115329
Baek, Yi-Yong
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Baker, Jillian G.
- You have accessComparative Docking to Distinct G Protein–Coupled Receptor Conformations Exclusively Yields Ligands with Agonist EfficacyMagdalena M. Scharf, Moritz Bünemann, Jillian G. Baker and Peter KolbMolecular Pharmacology December 2019, 96 (6) 851-861; DOI: https://doi.org/10.1124/mol.119.117515
Balabanian, Karl
- You have accessAtypical Chemokine Receptor 3 (ACKR3): A Comprehensive Overview of its Expression and Potential Roles in the Immune SystemJoyce Koenen, Françoise Bachelerie, Karl Balabanian, Géraldine Schlecht-Louf and Carmen GallegoMolecular Pharmacology December 2019, 96 (6) 809-818; DOI: https://doi.org/10.1124/mol.118.115329
Barrella, Lorenzo
- You have accessMutational Analysis and Modeling of Negative Allosteric Modulator Binding Sites in AMPA ReceptorsCharlotte Stenum-Berg, Maria Musgaard, Sergei Chavez-Abiega, Christine L. Thisted, Lorenzo Barrella, Philip C. Biggin and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 835-850; DOI: https://doi.org/10.1124/mol.119.116871
Biggin, Philip C.
- You have accessMutational Analysis and Modeling of Negative Allosteric Modulator Binding Sites in AMPA ReceptorsCharlotte Stenum-Berg, Maria Musgaard, Sergei Chavez-Abiega, Christine L. Thisted, Lorenzo Barrella, Philip C. Biggin and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 835-850; DOI: https://doi.org/10.1124/mol.119.116871
Bobkov, Vladimir
- Open AccessAntibodies Targeting Chemokine Receptors CXCR4 and ACKR3Vladimir Bobkov, Marta Arimont, Aurélien Zarca, Timo W.M. De Groof, Bas van der Woning, Hans de Haard and Martine J. SmitMolecular Pharmacology December 2019, 96 (6) 753-764; DOI: https://doi.org/10.1124/mol.119.116954
Briddon, Stephen
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Briddon, Stephen J.
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
Bünemann, Moritz
- You have accessComparative Docking to Distinct G Protein–Coupled Receptor Conformations Exclusively Yields Ligands with Agonist EfficacyMagdalena M. Scharf, Moritz Bünemann, Jillian G. Baker and Peter KolbMolecular Pharmacology December 2019, 96 (6) 851-861; DOI: https://doi.org/10.1124/mol.119.117515
C
Calhoun, Jacob
- You have accessFunctional RNAi Screens Define Distinct Protein Kinase Vulnerabilities in EGFR-Dependent HNSCC Cell LinesTrista K. Hinz, Emily K. Kleczko, Katherine R. Singleton, Jacob Calhoun, Lindsay A. Marek, Jihye Kim, Aik Choon Tan and Lynn E. HeasleyMolecular Pharmacology December 2019, 96 (6) 862-870; DOI: https://doi.org/10.1124/mol.119.117804
Capoferri, Davide
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
Caspar, Birgit
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
- Open AccessCXCR4/ACKR3 Phosphorylation and Recruitment of Interacting Proteins: Key Mechanisms Regulating Their Functional StatusAmos Fumagalli, Aurélien Zarca, Maria Neves, Birgit Caspar, Stephen J. Hill, Federico Mayor, Martine J. Smit and Philippe MarinMolecular Pharmacology December 2019, 96 (6) 794-808; DOI: https://doi.org/10.1124/mol.118.115360
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Chavez-Abiega, Sergei
- You have accessMutational Analysis and Modeling of Negative Allosteric Modulator Binding Sites in AMPA ReceptorsCharlotte Stenum-Berg, Maria Musgaard, Sergei Chavez-Abiega, Christine L. Thisted, Lorenzo Barrella, Philip C. Biggin and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 835-850; DOI: https://doi.org/10.1124/mol.119.116871
Chen, Gang
- Open AccessPotential Regulation of UGT2B10 and UGT2B7 by miR-485-5p in Human LiverAimee K. Sutliff, Jian Shi, Christy J.W. Watson, Martina S. Hunt, Gang Chen, Hao-Jie Zhu and Philip LazarusMolecular Pharmacology December 2019, 96 (6) 674-682; DOI: https://doi.org/10.1124/mol.119.115881
Chen, Lijuan
- You have accessThe Natural Compound Withaferin A Covalently Binds to Cys239 of β-Tubulin to Promote Tubulin DegradationJianhong Yang, Wei Yan, Yong Li, Lu Niu, Haoyu Ye and Lijuan ChenMolecular Pharmacology December 2019, 96 (6) 711-719; DOI: https://doi.org/10.1124/mol.119.117812
Choi, Seunghwan
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
D
de Esch, Iwan
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
de Graaf, Chris
- Open AccessChemokine Receptor Crystal Structures: What Can Be Learned from Them?Marta Arimont, Carsten Hoffmann, Chris de Graaf and Rob LeursMolecular Pharmacology December 2019, 96 (6) 765-777; DOI: https://doi.org/10.1124/mol.119.117168
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
De Groof, Timo W.M.
- Open AccessAntibodies Targeting Chemokine Receptors CXCR4 and ACKR3Vladimir Bobkov, Marta Arimont, Aurélien Zarca, Timo W.M. De Groof, Bas van der Woning, Hans de Haard and Martine J. SmitMolecular Pharmacology December 2019, 96 (6) 753-764; DOI: https://doi.org/10.1124/mol.119.116954
de Haard, Hans
- Open AccessAntibodies Targeting Chemokine Receptors CXCR4 and ACKR3Vladimir Bobkov, Marta Arimont, Aurélien Zarca, Timo W.M. De Groof, Bas van der Woning, Hans de Haard and Martine J. SmitMolecular Pharmacology December 2019, 96 (6) 753-764; DOI: https://doi.org/10.1124/mol.119.116954
Dekkers, Sebastian
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Durroux, Thierry
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
F
Fumagalli, Amos
- Open AccessCXCR4/ACKR3 Phosphorylation and Recruitment of Interacting Proteins: Key Mechanisms Regulating Their Functional StatusAmos Fumagalli, Aurélien Zarca, Maria Neves, Birgit Caspar, Stephen J. Hill, Federico Mayor, Martine J. Smit and Philippe MarinMolecular Pharmacology December 2019, 96 (6) 794-808; DOI: https://doi.org/10.1124/mol.118.115360
- You have accessThe Role of ACKR3 in Breast, Lung, and Brain CancerMaria Neves, Amos Fumagalli, Jelle van den Bor, Philippe Marin, Martine J. Smit and Federico MayorMolecular Pharmacology December 2019, 96 (6) 819-825; DOI: https://doi.org/10.1124/mol.118.115279
G
Gallego, Carmen
- You have accessAtypical Chemokine Receptor 3 (ACKR3): A Comprehensive Overview of its Expression and Potential Roles in the Immune SystemJoyce Koenen, Françoise Bachelerie, Karl Balabanian, Géraldine Schlecht-Louf and Carmen GallegoMolecular Pharmacology December 2019, 96 (6) 809-818; DOI: https://doi.org/10.1124/mol.118.115329
H
Ha, Kwon-Soo
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Heasley, Lynn E.
- You have accessFunctional RNAi Screens Define Distinct Protein Kinase Vulnerabilities in EGFR-Dependent HNSCC Cell LinesTrista K. Hinz, Emily K. Kleczko, Katherine R. Singleton, Jacob Calhoun, Lindsay A. Marek, Jihye Kim, Aik Choon Tan and Lynn E. HeasleyMolecular Pharmacology December 2019, 96 (6) 862-870; DOI: https://doi.org/10.1124/mol.119.117804
Heuninck, Joyce
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
Hill, Stephen
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Hill, Stephen J.
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
- Open AccessCXCR4/ACKR3 Phosphorylation and Recruitment of Interacting Proteins: Key Mechanisms Regulating Their Functional StatusAmos Fumagalli, Aurélien Zarca, Maria Neves, Birgit Caspar, Stephen J. Hill, Federico Mayor, Martine J. Smit and Philippe MarinMolecular Pharmacology December 2019, 96 (6) 794-808; DOI: https://doi.org/10.1124/mol.118.115360
Hinz, Trista K.
- You have accessFunctional RNAi Screens Define Distinct Protein Kinase Vulnerabilities in EGFR-Dependent HNSCC Cell LinesTrista K. Hinz, Emily K. Kleczko, Katherine R. Singleton, Jacob Calhoun, Lindsay A. Marek, Jihye Kim, Aik Choon Tan and Lynn E. HeasleyMolecular Pharmacology December 2019, 96 (6) 862-870; DOI: https://doi.org/10.1124/mol.119.117804
Hoffmann, Carsten
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
- Open AccessChemokine Receptor Crystal Structures: What Can Be Learned from Them?Marta Arimont, Carsten Hoffmann, Chris de Graaf and Rob LeursMolecular Pharmacology December 2019, 96 (6) 765-777; DOI: https://doi.org/10.1124/mol.119.117168
Hunt, Martina S.
- Open AccessPotential Regulation of UGT2B10 and UGT2B7 by miR-485-5p in Human LiverAimee K. Sutliff, Jian Shi, Christy J.W. Watson, Martina S. Hunt, Gang Chen, Hao-Jie Zhu and Philip LazarusMolecular Pharmacology December 2019, 96 (6) 674-682; DOI: https://doi.org/10.1124/mol.119.115881
I
Işbilir, Ali
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
J
Jackson, William F.
- You have accessLoss-of-Function Mutations in Human Regulator of G Protein Signaling RGS2 Differentially Regulate Pharmacological Reactivity of Resistance VasculatureHoa T.N. Phan, William F. Jackson, Vincent S. Shaw, Stephanie W. Watts and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 826-834; DOI: https://doi.org/10.1124/mol.119.116822
Jeoung, Dooil
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
K
Kellam, Barrie
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Kim, Ji-Yoon
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Kim, Jihye
- You have accessFunctional RNAi Screens Define Distinct Protein Kinase Vulnerabilities in EGFR-Dependent HNSCC Cell LinesTrista K. Hinz, Emily K. Kleczko, Katherine R. Singleton, Jacob Calhoun, Lindsay A. Marek, Jihye Kim, Aik Choon Tan and Lynn E. HeasleyMolecular Pharmacology December 2019, 96 (6) 862-870; DOI: https://doi.org/10.1124/mol.119.117804
Kim, Joohwan
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Kim, Suji
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Kim, Taesam
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Kim, Young-Myeong
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Kleczko, Emily K.
- You have accessFunctional RNAi Screens Define Distinct Protein Kinase Vulnerabilities in EGFR-Dependent HNSCC Cell LinesTrista K. Hinz, Emily K. Kleczko, Katherine R. Singleton, Jacob Calhoun, Lindsay A. Marek, Jihye Kim, Aik Choon Tan and Lynn E. HeasleyMolecular Pharmacology December 2019, 96 (6) 862-870; DOI: https://doi.org/10.1124/mol.119.117804
Koenen, Joyce
- You have accessAtypical Chemokine Receptor 3 (ACKR3): A Comprehensive Overview of its Expression and Potential Roles in the Immune SystemJoyce Koenen, Françoise Bachelerie, Karl Balabanian, Géraldine Schlecht-Louf and Carmen GallegoMolecular Pharmacology December 2019, 96 (6) 809-818; DOI: https://doi.org/10.1124/mol.118.115329
Kolb, Peter
- You have accessComparative Docking to Distinct G Protein–Coupled Receptor Conformations Exclusively Yields Ligands with Agonist EfficacyMagdalena M. Scharf, Moritz Bünemann, Jillian G. Baker and Peter KolbMolecular Pharmacology December 2019, 96 (6) 851-861; DOI: https://doi.org/10.1124/mol.119.117515
Kristensen, Anders S.
- You have accessConformational Changes in the 5-HT3A Receptor Extracellular Domain Measured by Voltage-Clamp FluorometryLachlan Munro, Lucy Kate Ladefoged, Vithushan Padmanathan, Signe Andersen, Birgit Schiøtt and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 720-734; DOI: https://doi.org/10.1124/mol.119.116657
- You have accessMutational Analysis and Modeling of Negative Allosteric Modulator Binding Sites in AMPA ReceptorsCharlotte Stenum-Berg, Maria Musgaard, Sergei Chavez-Abiega, Christine L. Thisted, Lorenzo Barrella, Philip C. Biggin and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 835-850; DOI: https://doi.org/10.1124/mol.119.116871
Kunselman, Jennifer M.
- You have accessHomologous Regulation of Mu Opioid Receptor Recycling by Gβγ, Protein Kinase C, and Receptor PhosphorylationJennifer M. Kunselman, Amanda S. Zajac, Zara Y. Weinberg and Manojkumar A. PuthenveeduMolecular Pharmacology December 2019, 96 (6) 702-710; DOI: https://doi.org/10.1124/mol.119.117267
Kwon, Young-Guen
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
L
Ladefoged, Lucy Kate
- You have accessConformational Changes in the 5-HT3A Receptor Extracellular Domain Measured by Voltage-Clamp FluorometryLachlan Munro, Lucy Kate Ladefoged, Vithushan Padmanathan, Signe Andersen, Birgit Schiøtt and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 720-734; DOI: https://doi.org/10.1124/mol.119.116657
Lazarus, Philip
- Open AccessPotential Regulation of UGT2B10 and UGT2B7 by miR-485-5p in Human LiverAimee K. Sutliff, Jian Shi, Christy J.W. Watson, Martina S. Hunt, Gang Chen, Hao-Jie Zhu and Philip LazarusMolecular Pharmacology December 2019, 96 (6) 674-682; DOI: https://doi.org/10.1124/mol.119.115881
Lee, Hansoo
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Leurs, Rob
- Open AccessChemokine Receptor Crystal Structures: What Can Be Learned from Them?Marta Arimont, Carsten Hoffmann, Chris de Graaf and Rob LeursMolecular Pharmacology December 2019, 96 (6) 765-777; DOI: https://doi.org/10.1124/mol.119.117168
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Li, Yong
- You have accessThe Natural Compound Withaferin A Covalently Binds to Cys239 of β-Tubulin to Promote Tubulin DegradationJianhong Yang, Wei Yan, Yong Li, Lu Niu, Haoyu Ye and Lijuan ChenMolecular Pharmacology December 2019, 96 (6) 711-719; DOI: https://doi.org/10.1124/mol.119.117812
Lohse, Martin J.
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
M
Marek, Lindsay A.
- You have accessFunctional RNAi Screens Define Distinct Protein Kinase Vulnerabilities in EGFR-Dependent HNSCC Cell LinesTrista K. Hinz, Emily K. Kleczko, Katherine R. Singleton, Jacob Calhoun, Lindsay A. Marek, Jihye Kim, Aik Choon Tan and Lynn E. HeasleyMolecular Pharmacology December 2019, 96 (6) 862-870; DOI: https://doi.org/10.1124/mol.119.117804
Marin, Philippe
- Open AccessCXCR4/ACKR3 Phosphorylation and Recruitment of Interacting Proteins: Key Mechanisms Regulating Their Functional StatusAmos Fumagalli, Aurélien Zarca, Maria Neves, Birgit Caspar, Stephen J. Hill, Federico Mayor, Martine J. Smit and Philippe MarinMolecular Pharmacology December 2019, 96 (6) 794-808; DOI: https://doi.org/10.1124/mol.118.115360
- You have accessThe Role of ACKR3 in Breast, Lung, and Brain CancerMaria Neves, Amos Fumagalli, Jelle van den Bor, Philippe Marin, Martine J. Smit and Federico MayorMolecular Pharmacology December 2019, 96 (6) 819-825; DOI: https://doi.org/10.1124/mol.118.115279
Mayor, Federico
- Open AccessCXCR4/ACKR3 Phosphorylation and Recruitment of Interacting Proteins: Key Mechanisms Regulating Their Functional StatusAmos Fumagalli, Aurélien Zarca, Maria Neves, Birgit Caspar, Stephen J. Hill, Federico Mayor, Martine J. Smit and Philippe MarinMolecular Pharmacology December 2019, 96 (6) 794-808; DOI: https://doi.org/10.1124/mol.118.115360
- You have accessThe Role of ACKR3 in Breast, Lung, and Brain CancerMaria Neves, Amos Fumagalli, Jelle van den Bor, Philippe Marin, Martine J. Smit and Federico MayorMolecular Pharmacology December 2019, 96 (6) 819-825; DOI: https://doi.org/10.1124/mol.118.115279
Milligan, Graeme
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
Mohammadi, Mohammadjavad
- You have accessAn Interhelical Salt Bridge Controls Flexibility and Inhibitor Potency for Regulators of G-protein Signaling Proteins 4, 8, and 19Vincent S. Shaw, Mohammadjavad Mohammadi, Josiah A. Quinn, Harish Vashisth and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 683-691; DOI: https://doi.org/10.1124/mol.119.117176
Munro, Lachlan
- You have accessConformational Changes in the 5-HT3A Receptor Extracellular Domain Measured by Voltage-Clamp FluorometryLachlan Munro, Lucy Kate Ladefoged, Vithushan Padmanathan, Signe Andersen, Birgit Schiøtt and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 720-734; DOI: https://doi.org/10.1124/mol.119.116657
Musgaard, Maria
- You have accessMutational Analysis and Modeling of Negative Allosteric Modulator Binding Sites in AMPA ReceptorsCharlotte Stenum-Berg, Maria Musgaard, Sergei Chavez-Abiega, Christine L. Thisted, Lorenzo Barrella, Philip C. Biggin and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 835-850; DOI: https://doi.org/10.1124/mol.119.116871
N
Neubig, Richard R.
- You have accessAn Interhelical Salt Bridge Controls Flexibility and Inhibitor Potency for Regulators of G-protein Signaling Proteins 4, 8, and 19Vincent S. Shaw, Mohammadjavad Mohammadi, Josiah A. Quinn, Harish Vashisth and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 683-691; DOI: https://doi.org/10.1124/mol.119.117176
- You have accessLoss-of-Function Mutations in Human Regulator of G Protein Signaling RGS2 Differentially Regulate Pharmacological Reactivity of Resistance VasculatureHoa T.N. Phan, William F. Jackson, Vincent S. Shaw, Stephanie W. Watts and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 826-834; DOI: https://doi.org/10.1124/mol.119.116822
Neves, Maria
- Open AccessCXCR4/ACKR3 Phosphorylation and Recruitment of Interacting Proteins: Key Mechanisms Regulating Their Functional StatusAmos Fumagalli, Aurélien Zarca, Maria Neves, Birgit Caspar, Stephen J. Hill, Federico Mayor, Martine J. Smit and Philippe MarinMolecular Pharmacology December 2019, 96 (6) 794-808; DOI: https://doi.org/10.1124/mol.118.115360
- You have accessThe Role of ACKR3 in Breast, Lung, and Brain CancerMaria Neves, Amos Fumagalli, Jelle van den Bor, Philippe Marin, Martine J. Smit and Federico MayorMolecular Pharmacology December 2019, 96 (6) 819-825; DOI: https://doi.org/10.1124/mol.118.115279
Niu, Lu
- You have accessThe Natural Compound Withaferin A Covalently Binds to Cys239 of β-Tubulin to Promote Tubulin DegradationJianhong Yang, Wei Yan, Yong Li, Lu Niu, Haoyu Ye and Lijuan ChenMolecular Pharmacology December 2019, 96 (6) 711-719; DOI: https://doi.org/10.1124/mol.119.117812
P
Padmanathan, Vithushan
- You have accessConformational Changes in the 5-HT3A Receptor Extracellular Domain Measured by Voltage-Clamp FluorometryLachlan Munro, Lucy Kate Ladefoged, Vithushan Padmanathan, Signe Andersen, Birgit Schiøtt and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 720-734; DOI: https://doi.org/10.1124/mol.119.116657
Park, Minsik
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Park, Wonjin
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Perpiñá Viciano, Cristina
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
Phan, Hoa T.N.
- You have accessLoss-of-Function Mutations in Human Regulator of G Protein Signaling RGS2 Differentially Regulate Pharmacological Reactivity of Resistance VasculatureHoa T.N. Phan, William F. Jackson, Vincent S. Shaw, Stephanie W. Watts and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 826-834; DOI: https://doi.org/10.1124/mol.119.116822
Pin, Jean-Philippe
- Open AccessContext-Dependent Signaling of CXC Chemokine Receptor 4 and Atypical Chemokine Receptor 3Joyce Heuninck, Cristina Perpiñá Viciano, Ali Işbilir, Birgit Caspar, Davide Capoferri, Stephen J. Briddon, Thierry Durroux, Stephen J. Hill, Martin J. Lohse, Graeme Milligan, Jean-Philippe Pin and Carsten HoffmannMolecular Pharmacology December 2019, 96 (6) 778-793; DOI: https://doi.org/10.1124/mol.118.115477
Puthenveedu, Manojkumar A.
- You have accessHomologous Regulation of Mu Opioid Receptor Recycling by Gβγ, Protein Kinase C, and Receptor PhosphorylationJennifer M. Kunselman, Amanda S. Zajac, Zara Y. Weinberg and Manojkumar A. PuthenveeduMolecular Pharmacology December 2019, 96 (6) 702-710; DOI: https://doi.org/10.1124/mol.119.117267
Q
Quinn, Josiah A.
- You have accessAn Interhelical Salt Bridge Controls Flexibility and Inhibitor Potency for Regulators of G-protein Signaling Proteins 4, 8, and 19Vincent S. Shaw, Mohammadjavad Mohammadi, Josiah A. Quinn, Harish Vashisth and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 683-691; DOI: https://doi.org/10.1124/mol.119.117176
S
Scharf, Magdalena M.
- You have accessComparative Docking to Distinct G Protein–Coupled Receptor Conformations Exclusively Yields Ligands with Agonist EfficacyMagdalena M. Scharf, Moritz Bünemann, Jillian G. Baker and Peter KolbMolecular Pharmacology December 2019, 96 (6) 851-861; DOI: https://doi.org/10.1124/mol.119.117515
Schiøtt, Birgit
- You have accessConformational Changes in the 5-HT3A Receptor Extracellular Domain Measured by Voltage-Clamp FluorometryLachlan Munro, Lucy Kate Ladefoged, Vithushan Padmanathan, Signe Andersen, Birgit Schiøtt and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 720-734; DOI: https://doi.org/10.1124/mol.119.116657
Schlecht-Louf, Géraldine
- You have accessAtypical Chemokine Receptor 3 (ACKR3): A Comprehensive Overview of its Expression and Potential Roles in the Immune SystemJoyce Koenen, Françoise Bachelerie, Karl Balabanian, Géraldine Schlecht-Louf and Carmen GallegoMolecular Pharmacology December 2019, 96 (6) 809-818; DOI: https://doi.org/10.1124/mol.118.115329
Shaw, Vincent S.
- You have accessAn Interhelical Salt Bridge Controls Flexibility and Inhibitor Potency for Regulators of G-protein Signaling Proteins 4, 8, and 19Vincent S. Shaw, Mohammadjavad Mohammadi, Josiah A. Quinn, Harish Vashisth and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 683-691; DOI: https://doi.org/10.1124/mol.119.117176
- You have accessLoss-of-Function Mutations in Human Regulator of G Protein Signaling RGS2 Differentially Regulate Pharmacological Reactivity of Resistance VasculatureHoa T.N. Phan, William F. Jackson, Vincent S. Shaw, Stephanie W. Watts and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 826-834; DOI: https://doi.org/10.1124/mol.119.116822
Shi, Jian
- Open AccessPotential Regulation of UGT2B10 and UGT2B7 by miR-485-5p in Human LiverAimee K. Sutliff, Jian Shi, Christy J.W. Watson, Martina S. Hunt, Gang Chen, Hao-Jie Zhu and Philip LazarusMolecular Pharmacology December 2019, 96 (6) 674-682; DOI: https://doi.org/10.1124/mol.119.115881
Singleton, Katherine R.
- You have accessFunctional RNAi Screens Define Distinct Protein Kinase Vulnerabilities in EGFR-Dependent HNSCC Cell LinesTrista K. Hinz, Emily K. Kleczko, Katherine R. Singleton, Jacob Calhoun, Lindsay A. Marek, Jihye Kim, Aik Choon Tan and Lynn E. HeasleyMolecular Pharmacology December 2019, 96 (6) 862-870; DOI: https://doi.org/10.1124/mol.119.117804
Smit, Martine J.
- You have accessFrom Insight to Modulation of CXCR4 and ACKR3 (CXCR7) FunctionMartine J. Smit and Jacqueline E. van Muijlwijk-KoezenMolecular Pharmacology December 2019, 96 (6) 735-736; DOI: https://doi.org/10.1124/mol.119.118364
- Open AccessCXCR4/ACKR3 Phosphorylation and Recruitment of Interacting Proteins: Key Mechanisms Regulating Their Functional StatusAmos Fumagalli, Aurélien Zarca, Maria Neves, Birgit Caspar, Stephen J. Hill, Federico Mayor, Martine J. Smit and Philippe MarinMolecular Pharmacology December 2019, 96 (6) 794-808; DOI: https://doi.org/10.1124/mol.118.115360
- Open AccessAntibodies Targeting Chemokine Receptors CXCR4 and ACKR3Vladimir Bobkov, Marta Arimont, Aurélien Zarca, Timo W.M. De Groof, Bas van der Woning, Hans de Haard and Martine J. SmitMolecular Pharmacology December 2019, 96 (6) 753-764; DOI: https://doi.org/10.1124/mol.119.116954
- You have accessThe Role of ACKR3 in Breast, Lung, and Brain CancerMaria Neves, Amos Fumagalli, Jelle van den Bor, Philippe Marin, Martine J. Smit and Federico MayorMolecular Pharmacology December 2019, 96 (6) 819-825; DOI: https://doi.org/10.1124/mol.118.115279
Stenum-Berg, Charlotte
- You have accessMutational Analysis and Modeling of Negative Allosteric Modulator Binding Sites in AMPA ReceptorsCharlotte Stenum-Berg, Maria Musgaard, Sergei Chavez-Abiega, Christine L. Thisted, Lorenzo Barrella, Philip C. Biggin and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 835-850; DOI: https://doi.org/10.1124/mol.119.116871
Stocks, Michael
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Stuijt, Jeffrey
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Sutliff, Aimee K.
- Open AccessPotential Regulation of UGT2B10 and UGT2B7 by miR-485-5p in Human LiverAimee K. Sutliff, Jian Shi, Christy J.W. Watson, Martina S. Hunt, Gang Chen, Hao-Jie Zhu and Philip LazarusMolecular Pharmacology December 2019, 96 (6) 674-682; DOI: https://doi.org/10.1124/mol.119.115881
T
Tan, Aik Choon
- You have accessFunctional RNAi Screens Define Distinct Protein Kinase Vulnerabilities in EGFR-Dependent HNSCC Cell LinesTrista K. Hinz, Emily K. Kleczko, Katherine R. Singleton, Jacob Calhoun, Lindsay A. Marek, Jihye Kim, Aik Choon Tan and Lynn E. HeasleyMolecular Pharmacology December 2019, 96 (6) 862-870; DOI: https://doi.org/10.1124/mol.119.117804
Thisted, Christine L.
- You have accessMutational Analysis and Modeling of Negative Allosteric Modulator Binding Sites in AMPA ReceptorsCharlotte Stenum-Berg, Maria Musgaard, Sergei Chavez-Abiega, Christine L. Thisted, Lorenzo Barrella, Philip C. Biggin and Anders S. KristensenMolecular Pharmacology December 2019, 96 (6) 835-850; DOI: https://doi.org/10.1124/mol.119.116871
V
van den Bor, Jelle
- You have accessThe Role of ACKR3 in Breast, Lung, and Brain CancerMaria Neves, Amos Fumagalli, Jelle van den Bor, Philippe Marin, Martine J. Smit and Federico MayorMolecular Pharmacology December 2019, 96 (6) 819-825; DOI: https://doi.org/10.1124/mol.118.115279
van der Woning, Bas
- Open AccessAntibodies Targeting Chemokine Receptors CXCR4 and ACKR3Vladimir Bobkov, Marta Arimont, Aurélien Zarca, Timo W.M. De Groof, Bas van der Woning, Hans de Haard and Martine J. SmitMolecular Pharmacology December 2019, 96 (6) 753-764; DOI: https://doi.org/10.1124/mol.119.116954
van Muijlwijk-Koezen, Jacqueline E.
- You have accessFrom Insight to Modulation of CXCR4 and ACKR3 (CXCR7) FunctionMartine J. Smit and Jacqueline E. van Muijlwijk-KoezenMolecular Pharmacology December 2019, 96 (6) 735-736; DOI: https://doi.org/10.1124/mol.119.118364
Vashisth, Harish
- You have accessAn Interhelical Salt Bridge Controls Flexibility and Inhibitor Potency for Regulators of G-protein Signaling Proteins 4, 8, and 19Vincent S. Shaw, Mohammadjavad Mohammadi, Josiah A. Quinn, Harish Vashisth and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 683-691; DOI: https://doi.org/10.1124/mol.119.117176
Visser, Kirsten
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
W
Watson, Christy J.W.
- Open AccessPotential Regulation of UGT2B10 and UGT2B7 by miR-485-5p in Human LiverAimee K. Sutliff, Jian Shi, Christy J.W. Watson, Martina S. Hunt, Gang Chen, Hao-Jie Zhu and Philip LazarusMolecular Pharmacology December 2019, 96 (6) 674-682; DOI: https://doi.org/10.1124/mol.119.115881
Watts, Stephanie W.
- You have accessLoss-of-Function Mutations in Human Regulator of G Protein Signaling RGS2 Differentially Regulate Pharmacological Reactivity of Resistance VasculatureHoa T.N. Phan, William F. Jackson, Vincent S. Shaw, Stephanie W. Watts and Richard R. NeubigMolecular Pharmacology December 2019, 96 (6) 826-834; DOI: https://doi.org/10.1124/mol.119.116822
Weinberg, Zara Y.
- You have accessHomologous Regulation of Mu Opioid Receptor Recycling by Gβγ, Protein Kinase C, and Receptor PhosphorylationJennifer M. Kunselman, Amanda S. Zajac, Zara Y. Weinberg and Manojkumar A. PuthenveeduMolecular Pharmacology December 2019, 96 (6) 702-710; DOI: https://doi.org/10.1124/mol.119.117267
Wijtmans, Maikel
- Open AccessModulators of CXCR4 and CXCR7/ACKR3 FunctionIlze Adlere, Birgit Caspar, Marta Arimont, Sebastian Dekkers, Kirsten Visser, Jeffrey Stuijt, Chris de Graaf, Michael Stocks, Barrie Kellam, Stephen Briddon, Maikel Wijtmans, Iwan de Esch, Stephen Hill and Rob LeursMolecular Pharmacology December 2019, 96 (6) 737-752; DOI: https://doi.org/10.1124/mol.119.117663
Won, Moo-Ho
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Y
Yan, Wei
- You have accessThe Natural Compound Withaferin A Covalently Binds to Cys239 of β-Tubulin to Promote Tubulin DegradationJianhong Yang, Wei Yan, Yong Li, Lu Niu, Haoyu Ye and Lijuan ChenMolecular Pharmacology December 2019, 96 (6) 711-719; DOI: https://doi.org/10.1124/mol.119.117812
Yang, Jianhong
- You have accessThe Natural Compound Withaferin A Covalently Binds to Cys239 of β-Tubulin to Promote Tubulin DegradationJianhong Yang, Wei Yan, Yong Li, Lu Niu, Haoyu Ye and Lijuan ChenMolecular Pharmacology December 2019, 96 (6) 711-719; DOI: https://doi.org/10.1124/mol.119.117812
Ye, Haoyu
- You have accessThe Natural Compound Withaferin A Covalently Binds to Cys239 of β-Tubulin to Promote Tubulin DegradationJianhong Yang, Wei Yan, Yong Li, Lu Niu, Haoyu Ye and Lijuan ChenMolecular Pharmacology December 2019, 96 (6) 711-719; DOI: https://doi.org/10.1124/mol.119.117812
Yun, Jung-A
- Open AccessN-Terminal Modification of the Tetrapeptide Arg-Leu-Tyr-Glu, a Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2) Antagonist, Improves Antitumor Activity by Increasing its Stability against Serum PeptidasesJung-A Yun, Joohwan Kim, Yi-Yong Baek, Wonjin Park, Minsik Park, Suji Kim, Taesam Kim, Seunghwan Choi, Dooil Jeoung, Hansoo Lee, Moo-Ho Won, Ji-Yoon Kim, Kwon-Soo Ha, Young-Guen Kwon and Young-Myeong KimMolecular Pharmacology December 2019, 96 (6) 692-701; DOI: https://doi.org/10.1124/mol.119.117234
Z
Zajac, Amanda S.
- You have accessHomologous Regulation of Mu Opioid Receptor Recycling by Gβγ, Protein Kinase C, and Receptor PhosphorylationJennifer M. Kunselman, Amanda S. Zajac, Zara Y. Weinberg and Manojkumar A. PuthenveeduMolecular Pharmacology December 2019, 96 (6) 702-710; DOI: https://doi.org/10.1124/mol.119.117267
Zarca, Aurélien
- Open AccessCXCR4/ACKR3 Phosphorylation and Recruitment of Interacting Proteins: Key Mechanisms Regulating Their Functional StatusAmos Fumagalli, Aurélien Zarca, Maria Neves, Birgit Caspar, Stephen J. Hill, Federico Mayor, Martine J. Smit and Philippe MarinMolecular Pharmacology December 2019, 96 (6) 794-808; DOI: https://doi.org/10.1124/mol.118.115360
- Open AccessAntibodies Targeting Chemokine Receptors CXCR4 and ACKR3Vladimir Bobkov, Marta Arimont, Aurélien Zarca, Timo W.M. De Groof, Bas van der Woning, Hans de Haard and Martine J. SmitMolecular Pharmacology December 2019, 96 (6) 753-764; DOI: https://doi.org/10.1124/mol.119.116954
Zhu, Hao-Jie
- Open AccessPotential Regulation of UGT2B10 and UGT2B7 by miR-485-5p in Human LiverAimee K. Sutliff, Jian Shi, Christy J.W. Watson, Martina S. Hunt, Gang Chen, Hao-Jie Zhu and Philip LazarusMolecular Pharmacology December 2019, 96 (6) 674-682; DOI: https://doi.org/10.1124/mol.119.115881
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