Table of Contents

Articles

• Open Access

  Kinetic Analysis of the Early Signaling Steps of the Human Chemokine Receptor CXCR4

  Cristina Perpiñá-Viciano, Ali Işbilir, Aurélien Zarca, Birgit Caspar, Laura E. Kilpatrick, Stephen J. Hill, Martine J. Smit, Martin J. Lohse and Carsten Hoffmann

  Molecular Pharmacology August 2020, 98 (2) 72-87; DOI: https://doi.org/10.1124/mol.119.118448
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  Modulation of Human Arylamine N-Acetyltransferase 1 Activity by Lysine Acetylation: Role of p300/CREB-Binding Protein and Sirtuins 1 and 2

  Neville J. Butcher, Rachel Burow and Rodney F. Minchin

  Molecular Pharmacology August 2020, 98 (2) 88-95; DOI: https://doi.org/10.1124/mol.119.119008
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  Characterization of Meta-Iodobenzylguanidine (mIBG) Transport by Polyspecific Organic Cation Transporters: Implication for mIBG Therapy

  Antonio J. López Quiñones, David J. Wagner and Joanne Wang

  Molecular Pharmacology August 2020, 98 (2) 109-119; DOI: https://doi.org/10.1124/mol.120.119495
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  MicroRNA hsa-miR-1301-3p Regulates Human ADH6, ALDH5A1 and ALDH8A1 in the Ethanol-Acetaldehyde-Acetate Metabolic Pathway

  Xubing Wang, Yanjie Zhao, Jiao Luo, Lin Xu, Xinmei Li, Yuan Jin, Chuanhai Li, Meiyao Feng, Ying Wang, Jing Chen, Yufei Hou, Qianwen Zhao, Jinquan Zhao, Baitang Ning, Yuxin Zheng and Dianke Yu

  Molecular Pharmacology August 2020, 98 (2) 120-129; DOI: https://doi.org/10.1124/mol.120.119693
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  Novel c-Myc–Targeting Compound N, N-Bis (5-Ethyl-2-Hydroxybenzyl) Methylamine for Mediated c-Myc Ubiquitin-Proteasomal Degradation in Lung Cancer Cells

  Nicharat Sriratanasak, Korrakod Petsri, Apirat Laobuthee, Worawat Wattanathana, Chanida Vinayanuwattikun, Sudjit Luanpitpong and Pithi Chanvorachote

  Molecular Pharmacology August 2020, 98 (2) 130-142; DOI: https://doi.org/10.1124/mol.120.119719
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  The Phosphodiesterase Inhibitor IBMX Blocks the Potassium Channel THIK-1 from the Extracellular Side

  Xinle Zou, Linus J. Conrad, Kristin Koschinsky, Günter Schlichthörl, Regina Preisig-Müller, Eugen Netz, Jens Krüger, Jürgen Daut and Vijay Renigunta

  Molecular Pharmacology August 2020, 98 (2) 143-155; DOI: https://doi.org/10.1124/molpharm.120.000011
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  Structural Refinement of the Tubulin Ligand (+)-Discodermolide to Attenuate Chemotherapy-Mediated Senescence

  Boying Guo, Alicia Rodriguez-Gabin, Andrea E. Prota, Tobias Mühlethaler, Nan Zhang, Kenny Ye, Michel O. Steinmetz, Susan Band Horwitz, Amos B. Smith and Hayley M. McDaid

  Molecular Pharmacology August 2020, 98 (2) 156-167; DOI: https://doi.org/10.1124/mol.119.117457
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  A Methyl Scan of the Pyrrolidinium Ring of Nicotine Reveals Significant Differences in Its Interactions with α7 and α4β2 Nicotinic Acetylcholine Receptors

  Hong Xing, Kristin W. Andrud, Ferenc Soti, Anne Rouchaud, Stephan C. Jahn, Ziang Lu, Yeh-Hyon Cho, Sophia Habibi, Patrick Corsino, Svetoslav Slavov, James R. Rocca, Jon M. Lindstrom, Ron J. Lukas and William R. Kem

  Molecular Pharmacology August 2020, 98 (2) 168-180; DOI: https://doi.org/10.1124/mol.119.118786