Table of Contents

Articles

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  Structure of Cytochrome P450 2C9*2 in Complex with Losartan: Insights into the Effect of Genetic Polymorphism

  Sonia J. Parikh, Chiara M. Evans, Juliet O. Obi, Qinghai Zhang, Keiko Maekawa, Karen C. Glass and Manish B. Shah

  Molecular Pharmacology November 2020, 98 (5) 529-539; DOI: https://doi.org/10.1124/molpharm.120.000042
• Open Access

  GS-967 and Eleclazine Block Sodium Channels in Human Induced Pluripotent Stem Cell–Derived Cardiomyocytes

  Franck Potet, Defne E. Egecioglu, Paul W. Burridge and Alfred L. George

  Molecular Pharmacology November 2020, 98 (5) 540-547; DOI: https://doi.org/10.1124/molpharm.120.000048
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  Regulation of Kappa Opioid Receptor Inactivation Depends on Sex and Cellular Site of Antagonist Action

  Kathryn L. Reichard, Keionna A. Newton, Zeena M.G. Rivera, Paulo M. Sotero de Menezes, Selena S. Schattauer, Benjamin B. Land and Charles Chavkin

  Molecular Pharmacology November 2020, 98 (5) 548-558; DOI: https://doi.org/10.1124/molpharm.120.000124
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  Transient Receptor Potential Ankyrin-1 and Vanilloid-3 Differentially Regulate Endoplasmic Reticulum Stress and Cytotoxicity in Human Lung Epithelial Cells After Pneumotoxic Wood Smoke Particle Exposure

  Nam D. Nguyen, Tosifa A. Memon, Katherine L. Burrell, Marysol Almestica-Roberts, Emmanuel Rapp, Lili Sun, Abigail F. Scott, Joseph E. Rower, Cassandra E. Deering-Rice and Christopher A. Reilly

  Molecular Pharmacology November 2020, 98 (5) 586-597; DOI: https://doi.org/10.1124/molpharm.120.000047
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  Open Access

  Arrestin Recruitment to C-C Chemokine Receptor 5: Potent C-C Chemokine Ligand 5 Analogs Reveal Differences in Dependence on Receptor Phosphorylation and Isoform-Specific Recruitment Bias

  Elsa Martins, Hellena Brodier, Irène Rossitto-Borlat, Ilke Ilgaz, Mélanie Villard and Oliver Hartley

  Molecular Pharmacology November 2020, 98 (5) 599-611; DOI: https://doi.org/10.1124/molpharm.120.000036
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  Antiepileptic Drug–Activated Constitutive Androstane Receptor Inhibits Peroxisome Proliferator–Activated Receptor α and Peroxisome Proliferator–Activated Receptor γ Coactivator 1α–Dependent Gene Expression to Increase Blood Triglyceride Levels

  Ryota Shizu, Yuta Otsuka, Kanako Ezaki, Chizuru Ishii, Shingo Arakawa, Yuto Amaike, Taiki Abe, Takuomi Hosaka, Takamitsu Sasaki, Yuichiro Kanno, Masaaki Miyata, Yasushi Yamazoe and Kouichi Yoshinari

  Molecular Pharmacology November 2020, 98 (5) 634-647; DOI: https://doi.org/10.1124/molpharm.120.000103