Table of Contents

Articles

• Open Access

  Identification of Celecoxib-Targeted Proteins Using Label-Free Thermal Proteome Profiling on Rat Hippocampus

  Elham Gholizadeh, Reza Karbalaei, Ali Khaleghian, Mona Salimi, Kambiz Gilany, Rabah Soliymani, Ziaurrehman Tanoli, Hassan Rezadoost, Marc Baumann, Mohieddin Jafari and Jing Tang

  Molecular Pharmacology May 2021, 99 (5) 308-318; DOI: https://doi.org/10.1124/molpharm.120.000210
• Open Access

  Inhibition of Bitter Taste from Oral Tenofovir Alafenamide

  Erik Schwiebert, Yi Wang, Ranhui Xi, Katarzyna Choma, John Streiff, Linda J. Flammer, Natasha Rivers, Mehmet Hakan Ozdener, Robert F. Margolskee, Carol M. Christensen, Nancy E. Rawson, Peihua Jiang and Paul A. S. Breslin

  Molecular Pharmacology May 2021, 99 (5) 319-327; DOI: https://doi.org/10.1124/molpharm.120.000071
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  Positive Allosteric Modulators of Metabotropic Glutamate Receptor 5 as Tool Compounds to Study Signaling Bias

  Angela Arsova, Thor C. Møller, Shane D. Hellyer, Line Vedel, Simon R. Foster, Jakob L. Hansen, Hans Bräuner-Osborne and Karen J. Gregory

  Molecular Pharmacology May 2021, 99 (5) 328-341; DOI: https://doi.org/10.1124/molpharm.120.000185
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  The Negative Allosteric Modulator EU1794-4 Reduces Single-Channel Conductance and Ca²⁺ Permeability of GluN1/GluN2A N-Methyl-d-Aspartate Receptors

  Riley E. Perszyk, Zhaoshi Zheng, Tue G. Banke, Jing Zhang, Lingling Xie, Miranda J. McDaniel, Brooke M. Katzman, Stephen C. Pelly, Hongjie Yuan, Dennis C. Liotta and Stephen F. Traynelis

  Molecular Pharmacology May 2021, 99 (5) 399-411; DOI: https://doi.org/10.1124/molpharm.120.000218