Elucidation of the Contribution of Active Site and Exosite Interactions to Affinity and Specificity of Peptidylic Serine Protease Inhibitors, using Non-natural Arginine Analogs

Masood Hosseini; Longguang Jiang; Hans Peter Sorensen; Jan K Jensen; Anni Christensen; Sarah Fogh; Cai Yuan; Lisbeth M. Andersen; Mingdong Huang; Peter A. Andreasen; Knud J. Jensen

doi:10.1124/mol.111.072280

Research ArticleArticle

Elucidation of the Contribution of Active Site and Exosite Interactions to Affinity and Specificity of Peptidylic Serine Protease Inhibitors, using Non-natural Arginine Analogs

Masood Hosseini, Longguang Jiang, Hans Peter Sorensen, Jan K Jensen, Anni Christensen, Sarah Fogh, Cai Yuan, Lisbeth M. Andersen, Mingdong Huang, Peter A. Andreasen and Knud J. Jensen

Molecular Pharmacology July 5, 2011, mol.111.072280; DOI: https://doi.org/10.1124/mol.111.072280

Masood Hosseini

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Longguang Jiang

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Hans Peter Sorensen

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Jan K Jensen

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Anni Christensen

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Sarah Fogh

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Cai Yuan

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Lisbeth M. Andersen

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Mingdong Huang

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Peter A. Andreasen

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Knud J. Jensen

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Research ArticleArticle

Elucidation of the Contribution of Active Site and Exosite Interactions to Affinity and Specificity of Peptidylic Serine Protease Inhibitors, using Non-natural Arginine Analogs

Masood Hosseini, Longguang Jiang, Hans Peter Sorensen, Jan K Jensen, Anni Christensen, Sarah Fogh, Cai Yuan, Lisbeth M. Andersen, Mingdong Huang, Peter A. Andreasen and Knud J. Jensen

Molecular Pharmacology July 5, 2011, mol.111.072280; DOI: https://doi.org/10.1124/mol.111.072280

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Research ArticleArticle

Elucidation of the Contribution of Active Site and Exosite Interactions to Affinity and Specificity of Peptidylic Serine Protease Inhibitors, using Non-natural Arginine Analogs

Masood Hosseini, Longguang Jiang, Hans Peter Sorensen, Jan K Jensen, Anni Christensen, Sarah Fogh, Cai Yuan, Lisbeth M. Andersen, Mingdong Huang, Peter A. Andreasen and Knud J. Jensen

Molecular Pharmacology July 5, 2011, mol.111.072280; DOI: https://doi.org/10.1124/mol.111.072280

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