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Michaelis-Menten quantification of ligand signalling bias applied to the promiscuous Vasopressin V2 receptor
Franziska Marie Heydenreich, Bianca Plouffe, Aurelien Rizk, Dalibor Milic, Joris Zhou, Billy Breton, Christian Le Gouill, Asuka Inoue, Michel Bouvier and Dmitry Veprintsev
Molecular Pharmacology July 2, 2022, MOLPHARM-AR-2022-000497; DOI: https://doi.org/10.1124/molpharm.122.000497
Franziska Marie Heydenreich
1Structural Studies, MRC Laboratory of Molecular Biology, United Kingdom
Bianca Plouffe
2Wellcome-Wolfson Institute for Experimental Medicine, Queen's University Belfast, United Kingdom
Aurelien Rizk
3InterAx Biotech AG, Switzerland
Dalibor Milic
4Department of Structural and Computational Biology, University of Vienna, Austria
Joris Zhou
5Institute for Research in Immunology and Cancer, University of Montreal, Canada
Billy Breton
5Institute for Research in Immunology and Cancer, University of Montreal, Canada
Christian Le Gouill
6University of Montreal, Canada
Asuka Inoue
7Tohoku University, Japan
Michel Bouvier
8Department of Biochemistry and Molec ular Medicine, University of Montreal, Canada
Dmitry Veprintsev
9School of Life Sciences, University of Nottingham, United Kingdom
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Molecular Pharmacology
Vol. 105, Issue 4
1 Apr 2024
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Michaelis Menten quantification of GPCR-G protein signalling
Franziska Marie Heydenreich, Bianca Plouffe, Aurelien Rizk, Dalibor Milic, Joris Zhou, Billy Breton, Christian Le Gouill, Asuka Inoue, Michel Bouvier and Dmitry Veprintsev
Molecular Pharmacology July 2, 2022, MOLPHARM-AR-2022-000497; DOI: https://doi.org/10.1124/molpharm.122.000497
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Michaelis Menten quantification of GPCR-G protein signalling
Franziska Marie Heydenreich, Bianca Plouffe, Aurelien Rizk, Dalibor Milic, Joris Zhou, Billy Breton, Christian Le Gouill, Asuka Inoue, Michel Bouvier and Dmitry Veprintsev
Molecular Pharmacology July 2, 2022, MOLPHARM-AR-2022-000497; DOI: https://doi.org/10.1124/molpharm.122.000497
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