Flumazenil | Flunitrazepam | β-CCM | CL218-872 | Zolpidem | Triazolam | Clonazepam | |
---|---|---|---|---|---|---|---|
μM | |||||||
α1β1γ1 | >50003-c | 37.74 ± 5.073-a | >50003-c | >50003-c | >50003-c | 25.65 ± 7.523-c | 150.0 ± 8.53-c |
α1β1γ2 | 0.91 ± 0.223-a | 3.90 ± 0.803-a | 0.45 ± 0.103-b | 46.75 ± 11.323-b | 40.23 ± 12.603-b | 0.45 ± 0.133-b | 1.03 ± 0.133-b |
α1β1γ3 | 2.80 ± 1.013-a | 150 ± 303-b | 5530 ± 13503-b | 6.04 ± 0.293-b | 25.95 ± 1.673-b | ||
α1β1γ1Δ2.2 | 3.07 ± 1.213-a | 9.75 ± 1.503-b | |||||
α1β1γ1Δ2.6 | 2.59 ± 1.853-a | 10.69 ± 2.453-b | 17.95 ± 2.523-b | ||||
α1β1γ1Δ2.7 | 1.62 ± 0.283-b | 38.94 ± 1.553-b | |||||
α1β1γ1ΔI79F | 3.13 ± 0.403-a | 44.64 ± 3.693-b | 0.71 ± 0.073-b | 27.22 ± 2.943-b | >50003-b | 3.44 ± 0.733-b | 14.58 ± 1.943-b |
α1β1γ1ΔL132M | >50003-c | 3.72 ± 0.573-a | 1390 ± 3003-c | >50003-c | >50003-c | 1.58 ± 0.363-c | 2.68 ± 0.593-c |
α1β1γ1ΔI79F, L132M | 10.56 ± 2.623-c | 6.98 ± 1.733-a | 1380 ± 2703-c | ||||
α1β1γ1ΔI79Y | 5.56 ± 2.193-a | >50003-b | |||||
α1β1γ2ΔF77I | 1420 ± 1903-a | 7.62 ± 1.183-b | 264.7 ± 19.13-b | >50003-b | >50003-b | ||
α1β1γ3ΔL133M | 3.90 ± 0.983-a | 33.19 ± 1.213-b | 330 ± 803-b | 1.49 ± 0.253-b | 4.80 ± 0.973-b |