Binding parameters of (±)-[3H]DOB obtained from saturation experiments with CHOFA4 cells expressing human 5-HT2A receptors
| Kd | Bmax | |
|---|---|---|
| nM | fmol/mg of protein | |
| Control | 0.80 ± 0.16 | 62.85 ± 22.27 |
| 31.22 ± 11.41 | 307.63 ± 54.84 | |
| Plus 100μM Gpp(NH)p | 24.44 ± 7.34 | 346.20 ± 79.89 |
Values represent mean ± S.E.M. of three independent experiments performed with duplicate points.