Table 1

IC50 values for selected nTAA compounds against [3H]TEA transport in hOCT1-expressing HeLa cells (mean ± S.E.M.; n = 3 to 4).

CompoundCLog PIC50
μM
TEA−3.14167.5  ± 25.9
TPrA−1.0222.0  ± 4.1
TBA1.096.5  ± 1.5
TPeA3.211.8  ± 0.2