Drug | pKi(Ki) | |||
---|---|---|---|---|
WT | V2.53L | WT2C | WT2A | |
nM | ||||
SNF | 7.76 ± 0.05 (17) | 6.64 ± 0.07d (230) | 7.16 ± 0.07 (69) | 5.74 ± 0.08 (1,800) |
RNF | 7.21 ± 0.04 (62) | 6.84 ± 0.07d (140) | 7.07 ± 0.08 (85) | 5.85 ± 0.07 (1,400) |
α-Desmethyl-NF | 7.26 ± 0.06a (55) | 6.58 ± 0.05bd (260) | 7.06 ± 0.07 (87) | 5.87 ± 0.06 (1,300) |
α-Ethyl-NF | 6.11 ± 0.08abc (780) | 6.44 ± 0.08abcd (360) | 6.0 ± 0.1abc (1,000) | 5.0 ± 0.1abc (10.000) |