Ligand | EC50 | ||
---|---|---|---|
cAMP | MAPK | ||
nM | |||
Isoproterenol | 4.99 ± 2.08 | 214.21 ± 90.73 | |
Labetalol | 6.76 ± 3.42 | 11.65 ± 5.58 | |
Bucindolol | > 10,000 | 0.95 ± 0.32 | |
Carvedilol | > 10,000 | 6.88 ± 4.09 | |
Propranolol | 2.32 ± 0.37 | 8.64 ± 2.84 | |
Metoprolol | 294.20 ± 95.58 | N.D. | |
Bisoprolol | 305.50 ± 131.48 | N.D. | |
Atenolol | 2400.80 ± 1342.00 | N.D. |
N.D., not determined.