Target Inhibitor (dose) | MDA-231 (ERBB2-/ER-) | SKBr3 (ERBB2+/ER-) | BT474 (ERBB2+/ER+) | MCF7 (ERBB2-/ER+) |
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ErbB2 kinase | - | + | + | - |
AG825 (25 μM) | ||||
MEK1/2 | + | + | + | + |
AZD6244 (100 nM) | ||||
PI3K | - | + | + | - |
LY294002 (10 μM) | ||||
Hsp90 | - | - | - | - |
17AAG (50 nM) | ||||
HDACs | + | - | - | + |
LAQ824 (10 nM) |
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