Compound | Luciferase-DMSO (Agonist Mode) | Luciferase-Rifampicin (Antagonist Mode) | ||||
---|---|---|---|---|---|---|
EC50 | Maximum Activation Observed | EC50 | Maximum Activation Observed | |||
μM | % | μM | % | |||
CDD3508 | 4.4 | 73 | 23.9 | 108 | ||
CDD3530 | 1.5 | 70 | 14.3 | 110 | ||
CDD3532 | 1.3 | 81 | 14.4 | 110 | ||
CDD3538 | 1.4 | 92 | 18.4 | 108 | ||
CDD3540 | 1.9 | 56 | 15.8 | 110 | ||
Clotrimazole | 1.1 | 96 | 16.7 | 107 |