HEK α4β2 pEC50 [Max-fold]a | HEK α3β4 pEC50 [Max-fold]a | |
---|---|---|
PNU-120596 | N.A. [0.89 ± 0.11]b (n = 4) | N.A. [0.80 ± 0.08]b (n = 4) |
TQS | 5.3 ± 0.2 [0.27 ± 0.04] (n = 4) | N.A. [0.89 ± 0.07]c (n = 4) |
5-HI | 3.4 ± 0.1 [0.21 ± 2.7] (n = 6) | 2.9 ± 0.2 [0.28 ± 2.7] (n = 4) |
Genistein | N.A. [0.60 ± 0.07]d (n = 6) | N.A. [0.63 ± 0.10]d (n = 4) |