pEC50 | |||
---|---|---|---|
M2 mAChR | A1R | ||
+10 μM Atropine | +100 μM Carbachol | +10 μM DPCPX | |
LUF5484 | 5.33 ± 0.22 | 5.53 ± 0.06 | N.D. |
PD81,723 | 4.98 ± 0.25 | 4.97 ± 0.07 | N.D. |
T62 | 5.68 ± 0.26 | 5.60 ± 0.10 | 5.23 ± 0.08 |
VCP520 | 5.78 ± 0.21 | 5.78 ± 0.08 | N.A. |
VCP333 | 5.77 ± 0.25 | 5.60 ± 0.07 | 5.67 ± 0.13 |
N.D., not determined; N.A., not applicable.