Agonist | t1/2 (95% CI) | Extent of Desensitization (95% CI) |
---|---|---|
min | % | |
Endomorphin-2 (30 μM) | 1.58 (1.52–1.64) | 47.9 (47.4–48.4) |
DAMGO (10 μM) | 2.98 (2.76–3.23) | 52.7 (51.1–54.3) |
Etorphine (1 μM) | 5.04 (4.10–6.55) | 54.6 (47.4–61.8) |
Morphine (30 μM) | 3.38 (3.16–3.63) | 30.2 (29.1–31.3) |
CI, confidence interval.