TABLE 3
p
K
i
values from competitive fit
Compound
p
K
i-GTP coupling
(95% CI)
p
K
i-
β
arr2 recruitment
(95% CI)
6′-GNTI
8.7 (9.1 to 8.4)
8.5 (8.8 to 8.1)
Nalbuphine
6.8 (7.0 to 6.6)
7.1 (7.4 to 6.9)
Nalmefene
9.1 (9.4 to 8.9)
9.0 (9.4 to 8.7)