Example | MW | PPB fu | CLInt | CLhep | CLogP | |||
---|---|---|---|---|---|---|---|---|
h | r | h | r | h | r | |||
ml/min per kg | ||||||||
1 (VU0652925) | 460.53 | <0.001 | <0.001 | 2.17 | 2.14 | 1.91 | 16.4 | 5.44 |
2 (VU0661247) | 407.44 | 0.001 | 0.003 | 17.7 | 37.9 | 9.62 | 24.6 | 5.09 |
3 (VU0661245) | 331.35 | 0.008 | 0.031 | 20.7 | 61.5 | 10.4 | 32.7 | 3.32 |
4 (VU0807074) | 301.32 | 0.007 | 0.03 | 133 | 336 | 18.1 | 57.9 | 3.23 |
5 (VU0807081) | 301.32 | 0.015 | 0.022 | 65.3 | 210 | 15.9 | 52.5 | 3.23 |
6 (VU0806526) | 271.04 | 0.01 | 0.047 | 89.4 | 285 | 17 | 56.2 | 3.31 |
cLogP, octanol/water partition coefficient; fu, unbound fraction; MW, molecular weight; PPB, plasma protein binding.