Compound | Structure | Drug Class | Kir4.1 IC50 | Reference |
---|---|---|---|---|
µM | ||||
Fluoxetine | SSRI | 15 | Ohno et al. (2007) | |
Amitriptyline | TCA | 89 | This study | |
Chloroquine | Antimalarial | 7 | Marmolejo-Murillo et al. (2017b) | |
Nortriptyline | TCA | 16–38a | Su et al. (2007) | |
Pentamidine | Antimicrobial | 0.097b | Takanari et al. (2013), Aréchiga-Figueroa et al. (2017) | |
Quinacrine | Antimalarial | ∼3 | Marmolejo-Murillo et al. (2017a) | |
VU717 | None | 6 | Raphemot et al. (2013) | |
VU0134992 | None | 0.97 | This study |