Peptide | IC50 (95% CI) | ||||
---|---|---|---|---|---|
T. californica nAChR | α7 nAChR | α9 LBD | L. stagnalis AChBP | A. californica AChBP | |
μM | |||||
R3 | >40 | >40 | >60 | >40 | >40 |
WR2 | > 20 | >40 | >60 | >40 | >40 |
W2R4 | 4.18 (3.32–5.26) | >40 | 15.5 (12.5–19.1) | >40 | >40 |
R6 | 1.21 (0.94–1.56) | >40 | 4.75 (3.31–6.82) | >40 | >40 |
R8 | 0.401 (0.376–0.442) | 22.4 (20.7–24.2) | 1.31 (1.20–1.43) | >20 | >40 |
R16 | 0.036 (0.028–0.045) | 7.66 (5.44–10.79) | 0.16 (0.14–0.18) | 1.44 (1.21–1.74) | >40 |