TABLE 2
Kinetics of HNK inhibition
Data are means and 95% confidence intervals.
KET
HNK
k
on
0.6 (95% CI −0.6 to 1.5) × 10
6
M
−1
s
−1
0.006 (95% CI 0.002–0.01) × 10
6
M
−1
s
−1
*
k
off
0.7 (95% CI 0.2–1.3) s
−1
1.3 (95% CI 1.28–1.3) s
−1
K
D
0.6 µM
203 µM
*
↵
*
P
= 0.02 relative to KET.